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Scopus Author ID: 7005870313

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Works (47)

Synthesis and Antiviral Evaluation of 5-(4-Aryl-1,3-butadiyn-1-yl)-uridines and Their Phosphoramidate Pronucleotides

Molecules
2024-12 | Journal article | Author
DOI: 10.3390/molecules30010096
Contributors: Evan Saillard; otmane bourzikat; Koffi Assa; vincent; Luigi AGROFOGLIO
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Multidisciplinary Digital Publishing Institute

Antibiotics and Antibiotic Resistance—Mur Ligases as an Antibacterial Target

Molecules
2023-12 | Journal article | Author
DOI: 10.3390/molecules28248076
Contributors: Vincent Hervin; vincent; Luigi AGROFOGLIO
Source: check_circle
Multidisciplinary Digital Publishing Institute

Synthesis and Antiviral Evaluation of (1,4-Disubstituted-1,2,3-Triazol)-(<i>E</i>)-2-Methyl-but-2-Enyl Nucleoside Phosphonate Prodrugs

Molecules
2021-03 | Journal article | Author
DOI: 10.3390/molecules26051493
Contributors: Tuniyazi Abuduaini; vincent; Julien Marlet; Catherine Gaudy-Graffin; Denys Brand; Cécile Baronti; Franck Touret; Bruno Coutard; Tamara R. McBrayer; Raymond F. Schinazi et al.
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Multidisciplinary Digital Publishing Institute

Design and Synthesis of Various 5′-Deoxy-5′-(4-Substituted-1,2,3-Triazol-1-yl)-Uridine Analogues as Inhibitors of <i>Mycobacterium tuberculosis</i> Mur Ligases

Molecules
2020-10 | Journal article | Author
DOI: 10.3390/molecules25214953
Contributors: Vincent Hervin; Ritu Arora; Jyoti Rani; Srinivasan Ramchandran; Urmi Bajpai; Luigi AGROFOGLIO; vincent
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Multidisciplinary Digital Publishing Institute

Highly convergent synthesis and antiviral activity of (E)-but-2-enyl nucleoside phosphonoamidates

European Journal of Medicinal Chemistry
2018 | Journal article
DOI: 10.1016/j.ejmech.2018.01.086
EID:

2-s2.0-85041599355
Contributors: Bessières, M.; Hervin, V.; Roy, V.; Chartier, A.; Snoeck, R.; Andrei, G.; Lohier, J.-F.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Selective inhibition of human cathepsin S by 2,4,6-trisubstituted 1,3,5-triazine analogs

Bioorganic and Medicinal Chemistry
2018 | Journal article
DOI: 10.1016/j.bmc.2018.07.032
EID:

2-s2.0-85050193428
Contributors: Tber, Z.; Wartenberg, M.; Jacques, J.-E.; Roy, V.; Lecaille, F.; Warszycki, D.; Bojarski, A.J.; Lalmanach, G.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Synthesis and characterization of various 5′-dye-labeled ribonucleosides

Organic and Biomolecular Chemistry
2018 | Journal article
DOI: 10.1039/c8ob01606b
EID:

2-s2.0-85053548532
Contributors: De Schutter, C.; Roy, V.; Favetta, P.; Pavageau, C.; Maisonneuve, S.; Bogliotti, N.; Xie, J.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Synthesis of 5,5-difluoro-5-phosphono-pent-2-en-1-yl nucleosides as potential antiviral agents

RSC Advances
2017 | Journal article
DOI: 10.1039/c7ra05153k
EID:

2-s2.0-85021772321
Contributors: Chevrier, F.; Chamas, Z.; Lequeux, T.; Pfund, E.; Andrei, G.; Snoeck, R.; Roy, V.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Tailor-Made Molecularly Imprinted Polymer for Selective Recognition of the Urinary Tumor Marker Pseudouridine

Macromolecular Bioscience
2017 | Journal article
DOI: 10.1002/mabi.201700250
EID:

2-s2.0-85034108737
Contributors: Krstulja, A.; Lettieri, S.; Hall, A.J.; Roy, V.; Favetta, P.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Sonication-Assisted Synthesis of (E)-2-Methyl-but-2-enyl Nucleoside Phosphonate Prodrugs

ChemistrySelect
2016 | Journal article
DOI: 10.1002/slct.201600879
EID:

2-s2.0-85021731181
Contributors: Bessières, M.; Sari, O.; Roy, V.; Warszycki, D.; Bojarski, A.J.; Nolan, S.P.; Snoeck, R.; Andrei, G.; Schinazi, R.F.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Straightforward synthesis of 2,4,6-trisubstituted 1,3,5-triazine compounds targeting cysteine cathepsins K and S

European Journal of Medicinal Chemistry
2016 | Journal article
DOI: 10.1016/j.ejmech.2016.05.009
EID:

2-s2.0-84969668259
Contributors: Plebanek, E.; Chevrier, F.; Roy, V.; Garenne, T.; Lecaille, F.; Warszycki, D.; Bojarski, A.J.; Lalmanach, G.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Active site labeling of cysteine cathepsins by a straightforward diazomethylketone probe derived from the N-terminus of human cystatin C

Biochemical and Biophysical Research Communications
2015 | Journal article
DOI: 10.1016/j.bbrc.2015.03.020
EID:

2-s2.0-84937758444
Contributors: Garenne, T.; Saidi, A.; Gilmore, B.F.; Niemiec, E.; Roy, V.; Agrofoglio, L.A.; Kasabova, M.; Lecaille, F.; Lalmanach, G.
Source: Self-asserted source
vincent via Scopus - Elsevier

Recent progress for the synthesis of selected carbocyclic nucleosides

Future Medicinal Chemistry
2015 | Journal article
DOI: 10.4155/fmc.15.105
EID:

2-s2.0-84944382753
Contributors: Bessières, M.; Chevrier, F.; Roy, V.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Synthesis of dihydropyrimidine α,mu;3-diketobutanoic acid derivatives targeting HIV integrase

European Journal of Medicinal Chemistry
2015 | Journal article
DOI: 10.1016/j.ejmech.2015.09.015
EID:

2-s2.0-84944045760
Contributors: Sari, O.; Roy, V.; Métifiot, M.; Marchand, C.; Pommier, Y.; Bourg, S.; Bonnet, P.; Schinazi, R.F.; Agrofoglio, L.A.
Source: Self-asserted source
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Synthesis of fluorine-containing 3,3-disubstituted oxetanes and alkylidene oxetanes

European Journal of Organic Chemistry
2015 | Journal article
DOI: 10.1002/ejoc.201500172
EID:

2-s2.0-84928803395
Contributors: Laporte, R.; Prunier, A.; Pfund, E.; Roy, V.; Agrofoglio, L.A.; Lequeux, T.
Source: Self-asserted source
vincent via Scopus - Elsevier

A convenient, highly selective and eco-friendly N-Boc protection of pyrimidines under microwave irradiation

RSC Advances
2014 | Journal article
DOI: 10.1039/c4ra13033b
EID:

2-s2.0-84911994560
Contributors: Bessières, M.; Roy, V.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Detection of urinary modified nucleosides by a bulk acoustic wave MIP sensor - Results and future work

IRBM
2014 | Journal article
DOI: 10.1016/j.irbm.2014.02.009
EID:

2-s2.0-84898043439
Contributors: Agrofoglio, L.A.; Krstulja, A.; De Schutter, C.; Favetta, P.; Delépée, R.; Roy, V.; Dejous, C.; Hallil, H.; Lachaud, J.-L.; Lebal, N. et al.
Source: Self-asserted source
vincent via Scopus - Elsevier

Development of nucleoside analogs under microwave irradiation

Microwaves in Drug Discovery and Development: Recent Advances
2014 | Book
Part of DOI: 10.4155/FSEB2013.13.126
EID:

2-s2.0-84957381825
Contributors: Niemiec, E.; Bessieres, M.; Roy, V.; Agrofoglio, L.A.Luigi A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Olefin cross-metathesis for the synthesis of alkenyl acyclonucleoside phosphonates

Current Protocols in Nucleic Acid Chemistry
2014 | Journal article
DOI: 10.1002/0471142700.nc1411s59
EID:

2-s2.0-84949293246
Contributors: Bessières, M.; De Schutter, C.; Roy, V.; Agofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Nucleosides Modified at the Base Moiety

Chemical Synthesis of Nucleoside Analogues
2013 | Book
Part of DOI: 10.1002/9781118498088.ch2
EID:

2-s2.0-84886833261
Contributors: Sari, O.; Roy, V.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Synthesis and broad spectrum antiviral evaluation of bis(POM) prodrugs of novel acyclic nucleosides

European Journal of Medicinal Chemistry
2013 | Journal article
DOI: 10.1016/j.ejmech.2013.06.053
EID:

2-s2.0-84880902014
Contributors: Hamada, M.; Roy, V.; McBrayer, T.R.; Whitaker, T.; Urbina-Blanco, C.; Nolan, S.P.; Balzarini, J.; Snoeck, R.; Andrei, G.; Schinazi, R.F. et al.
Source: Self-asserted source
vincent via Scopus - Elsevier

The preparation of trisubstituted alkenyl nucleoside phosphonates under ultrasound-assisted olefin cross-metathesis

Organic Letters
2013 | Journal article
DOI: 10.1021/ol401922r
EID:

2-s2.0-84883746443
Contributors: Sari, O.; Hamada, M.; Roy, V.; Nolan, S.P.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Synthesis and antiviral evaluation of bis(POM) prodrugs of (E)-[4′-phosphono-but-2′-en-1′-yl]purine nucleosides

European Journal of Medicinal Chemistry
2012 | Journal article
DOI: 10.1016/j.ejmech.2012.08.042
EID:

2-s2.0-84866976536
Contributors: Pradère, U.; Roy, V.; Montagu, A.; Sari, O.; Hamada, M.; Balzarini, J.; Snoeck, R.; Andrei, G.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Synthesis and antiviral evaluation of C5-substituted-(1,3-diyne)-2′- deoxyuridines

European Journal of Medicinal Chemistry
2012 | Journal article
DOI: 10.1016/j.ejmech.2012.04.001
EID:

2-s2.0-84861581552
Contributors: Sari, O.; Roy, V.; Balzarini, J.; Snoeck, R.; Andrei, G.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Expeditious convergent procedure for the preparation of bis(POC) prodrugs of new (E)-4-phosphono-but-2-en-1-yl nucleosides

Tetrahedron
2011 | Journal article
DOI: 10.1016/j.tet.2011.05.017
EID:

2-s2.0-79958770577
Contributors: Montagu, A.; Pradére, U.; Roy, V.; Nolan, S.P.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

In situ one-step method for synthesis of "click"-functionalized monolithic stationary phase for capillary electrochromatography

Macromolecular Chemistry and Physics
2011 | Journal article
DOI: 10.1002/macp.201100526
EID:

2-s2.0-83455164716
Contributors: Salwiński, A.; Roy, V.; Agrofoglio, L.A.; Delépée, R.
Source: Self-asserted source
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Novel antiviral C5-substituted pyrimidine acyclic nucleoside phosphonates selected as human thymidylate kinase substrates

Journal of Medicinal Chemistry
2011 | Journal article
DOI: 10.1021/jm1011462
EID:

2-s2.0-78651091005
Contributors: Topalis, D.; Pradère, U.; Roy, V.; Caillat, C.; Azzouzi, A.; Broggi, J.; Snoeck, R.; Andrei, G.; Lin, J.; Eriksson, S. et al.
Source: Self-asserted source
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Synthesis and anti-HIV evaluation of 3′-triazolo nucleosides

Nucleosides, Nucleotides and Nucleic Acids
2011 | Journal article
DOI: 10.1080/15257770.2011.580291
EID:

2-s2.0-79957789729
Contributors: Roy, V.; Obikhod, A.; Zhang, H.-W.; Coats, S.J.; Herman, B.D.; Sluis-Cremer, N.; Agrofoglio, L.A.; Schinazi, R.F.
Source: Self-asserted source
vincent via Scopus - Elsevier

Synthesis of new C5-(1-substituted-1,2,3-triazol-4 or 5-yl)-2′- deoxyuridines and their antiviral evaluation

European Journal of Medicinal Chemistry
2011 | Journal article
DOI: 10.1016/j.ejmech.2010.12.017
EID:

2-s2.0-79151483228
Contributors: Montagu, A.; Roy, V.; Balzarini, J.; Snoeck, R.; Andrei, G.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

The shortest strategy for generating phosphonate prodrugs by olefin cross-metathesis - Application to acyclonucleoside phosphonates

European Journal of Organic Chemistry
2011 | Journal article
DOI: 10.1002/ejoc.201101111
EID:

2-s2.0-82955223239
Contributors: Pradère, U.; Clavier, H.; Roy, V.; Nolan, S.P.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

3′-(1,2,3-Triazol-1-yl)-3′-deoxythymidine analogs as substrates for human and Ureaplasma parvum thymidine kinase for structure-activity investigations

Bioorganic and Medicinal Chemistry
2010 | Journal article
DOI: 10.1016/j.bmc.2010.03.023
EID:

2-s2.0-77951296059
Contributors: Lin, J.; Roy, V.; Wang, L.; You, L.; Agrofoglio, L.A.; Deville-Bonne, D.; McBrayer, T.R.; Coats, S.J.; Schinazi, R.F.; Eriksson, S.
Source: Self-asserted source
vincent via Scopus - Elsevier

Microwave-assisted syntheses of nucleosides and their precursors

Future Medicinal Chemistry
2010 | Journal article
DOI: 10.4155/fmc.09.156
EID:

2-s2.0-77953390041
Contributors: Roy, V.; Pradère, U.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Preparation of carbocyclic C-nucleosides from α-chlorooxime precursor

European Journal of Organic Chemistry
2010 | Journal article
DOI: 10.1002/ejoc.200900950
EID:

2-s2.0-74949127969
Contributors: Pradere, U.; Kumamoto, H.; Roy, V.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Preparation of cyclonucleosides

Chemical Reviews
2010 | Journal article
DOI: 10.1021/cr900329y
EID:

2-s2.0-77951232654
Contributors: Mieczkowski, A.; Roy, V.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Preparation of C-5-substituted 6,5′-O-anhydrouridine by Sn-Pd transmetallation-coupling process and their use

Tetrahedron
2009 | Journal article
DOI: 10.1016/j.tet.2009.09.075
EID:

2-s2.0-70349972668
Contributors: Mieczkowski, A.; Blu, J.; Roy, V.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Microwave-assisted silylation-amination of uracil acyclonucleosides to 4-alkylamino-2(1H)-pyrimidinone analogues

Synthesis
2008 | Journal article
DOI: 10.1055/s-2008-1067094
EID:

2-s2.0-47349122417
Contributors: Roy, V.; Mieczkowski, A.; Topalis, D.; Berteina-Raboin, S.; Deville-Bonne, D.; Nolan, S.P.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

Preparation of acyclo nucleoside phosphonate analogues based on cross-metathesis

Tetrahedron
2008 | Journal article
DOI: 10.1016/j.tet.2008.01.140
EID:

2-s2.0-39849086493
Contributors: Kumamoto, H.; Topalis, D.; Broggi, J.; Pradère, U.; Roy, V.; Berteina-Raboin, S.; Nolan, S.P.; Deville-Bonne, D.; Andrei, G.; Snoeck, R. et al.
Source: Self-asserted source
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Preparation of ribavirin analogues by copper- and ruthenium-catalyzed azide-alkyne 1,3-dipolar cycloaddition

Tetrahedron
2008 | Journal article
DOI: 10.1016/j.tet.2008.07.007
EID:

2-s2.0-48549095314
Contributors: Pradere, U.; Roy, V.; McBrayer, T.R.; Schinazi, R.F.; Agrofoglio, L.A.
Source: Self-asserted source
vincent via Scopus - Elsevier

A cryptophane biosensor for the detection of specific nucleotide targets through xenon NMR spectroscopy

ChemPhysChem
2007 | Journal article
DOI: 10.1002/cphc.200700384
EID:

2-s2.0-35348955844
Contributors: Roy, V.; Brotin, T.; Dutasta, J.-P.; Charles, M.-H.; Delair, T.; Mallet, F.; Huber, G.; Desvaux, H.; Boulard, Y.; Berthault, P.
Source: Self-asserted source
vincent via Scopus - Elsevier

Cross-metathesis mediated synthesis of new acyclic nucleoside phosphonates

Nucleosides, Nucleotides and Nucleic Acids
2007 | Journal article
DOI: 10.1080/15257770701534196
EID:

2-s2.0-36949034699
Contributors: Roy, V.; Kumamoto, H.; Berteina-Raboin, S.; Nolan, S.P.; Topalis, D.; Deville-Bonne, D.; Balzarini, J.; Neyts, J.; Andrei, G.; Snoeck, R. et al.
Source: Self-asserted source
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Synthesis and antiviral evaluation of AZT analogues with a spacer arm between glucidic and base moieties. Part II

Nucleosides, Nucleotides and Nucleic Acids
2007 | Journal article
DOI: 10.1080/15257770701426153
EID:

2-s2.0-34250702028
Contributors: Roy, V.; Zerrouki, R.; Krausz, P.; Laumond, G.; Aubertin, A.M.
Source: Self-asserted source
vincent via Scopus - Elsevier

Cross-metathesis in the synthesis of bioactive phosphonates

Chimica Oggi
2006 | Journal article
EID:

2-s2.0-33846307095
Contributors: Agrofoglio, L.A.; Kumamoto, H.; Roy, V.
Source: Self-asserted source
vincent via Scopus - Elsevier

Improved synthesis of functional CTVs and cryptophanes using Sc(OTf)<inf>3</inf>as catalyst

Journal of Organic Chemistry
2005 | Journal article
DOI: 10.1021/jo050495g
EID:

2-s2.0-23044487193
Contributors: Brotin, T.; Roy, V.; Dutasta, J.-P.
Source: Self-asserted source
vincent via Scopus - Elsevier

New dinucleoside analogues via cross-coupling metathesis

Nucleosides, Nucleotides and Nucleic Acids
2005 | Journal article
DOI: 10.1081/NCN-60595
EID:

2-s2.0-22044439161
Contributors: Roy, V.; Zerrouki, R.; Krausz, P.
Source: Self-asserted source
vincent via Scopus - Elsevier

One step selective 5′-O-allylation of thymidine using microwave or ultrasound activation

Carbohydrate Research
2004 | Journal article
DOI: 10.1016/j.carres.2004.04.008
EID:

2-s2.0-3042608729
Contributors: Roy, V.; Colombeau, L.; Zerrouki, R.; Krausz, P.
Source: Self-asserted source
vincent via Scopus - Elsevier

Selective deprotection of fully benzoylated nucleoside derivatives

Journal of Carbohydrate Chemistry
2004 | Journal article
DOI: 10.1081/CAR-200030095
EID:

2-s2.0-28244455815
Contributors: Zerrouki, R.; Roy, V.; Hadj-Bouazza, A.; Krausz, P.
Source: Self-asserted source
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Synthesis and antiviral evaluation of D4T analogues with a spacer arm between glucidic and base moieties

Nucleosides, Nucleotides and Nucleic Acids
2004 | Journal article
DOI: 10.1081/NCN-200031457
EID:

2-s2.0-9644254200
Contributors: Roy, V.; Zerrouki, R.; Krausz, P.; Schmidt, S.; Aubertin, A.M.
Source: Self-asserted source
vincent via Scopus - Elsevier
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