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Mechanistic and Structural Insights on Difluoromethyl-1,3,4-oxadiazole Inhibitors of HDAC6

International Journal of Molecular Sciences
2024-05-28 | Journal article
Contributors: Edoardo Cellupica; Aureliano Gaiassi; Ilaria Rocchio; Grazia Rovelli; Roberta Pomarico; Giovanni Sandrone; Gianluca Caprini; Paola Cordella; Cyprian Cukier; Gianluca Fossati et al.
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Difluoromethyl-1,3,4-oxadiazoles are slow-binding substrate analog inhibitors of histone deacetylase 6 with unprecedented isotype selectivity

Journal of Biological Chemistry
2023-01 | Journal article
Contributors: Edoardo Cellupica; Gianluca Caprini; Paola Cordella; Cyprian Cukier; Gianluca Fossati; Mattia Marchini; Ilaria Rocchio; Giovanni Sandrone; Maria Antonietta Vanoni; Barbara Vergani et al.
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