Personal information

France

Activities

Works (27)

Cholesterol Oxime Olesoxime Assessed as a Potential Ligand of Human Cholinesterases

Biomolecules
2024-05 | Journal article | Author
Contributors: Dora Kolić; Goran Šinko; Ludovic Jean; Mourad Chioua; José Dias; José Marco-Contelles; Zrinka Kovarik
Source: check_circle
Multidisciplinary Digital Publishing Institute

The risk associated with organophosphorus nerve agents: from their discovery to their unavoidable threat, current medical countermeasures and perspectives.

Chemico-biological interactions
2024-04-02 | Journal article
Contributors: Voros C; Dias J; Timperley CM; Nachon F; Brown RCD; Baati R
Source: Self-asserted source
José Dias

Inhibition of Human Cholinesterases and in vitro β‐Amyloid Aggregation by Rationally Designed Peptides

ChemMedChem
2023-06-15 | Journal article
Part of ISSN: 1860-7179
Part of ISSN: 1860-7187
Contributors: Ivan Sanchis; Roque Spinelli; José Dias; Xavier Brazzolotto; Álvaro Rietmann; Florencia Aimaretti; Alvaro Siano
Source: Self-asserted source
José Dias

Grid‐Type Quaternary Metallosupramolecular Compounds Inhibit Human Cholinesterases through Dynamic Multivalent Interactions

ChemBioChem
2022-12-05 | Journal article
Part of ISSN: 1439-4227
Part of ISSN: 1439-7633
Contributors: Florian Nachon; Xavier BRAZZOLOTTO; José Dias; Charlotte Courageux; Wojciech Drożdż; Xiao‐Yu Cao; Artur R. Stefankiewicz; Jean‐Marie Lehn
Source: Self-asserted source
José Dias

A New Class of Bi- and Trifunctional Sugar Oximes as Antidotes against Organophosphorus Poisoning

Journal of Medicinal Chemistry
2022-03-24 | Journal article
Part of ISSN: 0022-2623
Part of ISSN: 1520-4804
Contributors: José Dias
Source: Self-asserted source
José Dias

From tryptophan-based amides to tertiary amines: Optimization of a butyrylcholinesterase inhibitor series.

European journal of medicinal chemistry
2022-03-07 | Journal article
Contributors: José Dias
Source: Self-asserted source
José Dias

Discovery of multifunctional anti-Alzheimer's agents with a unique mechanism of action including inhibition of the enzyme butyrylcholinesterase and γ-aminobutyric acid transporters.

European journal of medicinal chemistry
2021-03-31 | Journal article
Contributors: José Dias
Source: Self-asserted source
José Dias

Fine-Tuning the Biological Profile of Multitarget Mitochondriotropic Antioxidants for Neurodegenerative Diseases

Antioxidants
2021-02 | Journal article | Author
Contributors: Daniel Chavarria; Ophelie DA SILVA; Sofia Benfeito; Sandra Barreiro; Jorge Garrido; Cagide-Fagín, Fernando; Cagide, Fernando; Pedro Soares; Fernando Remião; Xavier BRAZZOLOTTO; Florian Nachon et al.
Source: check_circle
Multidisciplinary Digital Publishing Institute

Discovery of drug-like acetylcholinesterase inhibitors by rapid virtual screening of a 6.9 million compound database.

Chemical biology & drug design
2021-02-02 | Journal article
Contributors: José Dias
Source: Self-asserted source
José Dias

Development of versatile and potent monoquaternary reactivators of acetylcholinesterase.

Archives of toxicology
2021-01-31 | Journal article
Contributors: José Dias
Source: Self-asserted source
José Dias

Efficacy assessment of an uncharged reactivator of nop-inhibited acetylcholinesterase based on tetrahydroacridine pyridine-aldoxime hybrid in mouse compared to pralidoxime

Biomolecules
2020 | Journal article
EID:

2-s2.0-85086045322

Part of ISBN:

2218273X

Contributors: Calas, A.-G.; Hanak, A.-S.; Jaffré, N.; Nervo, A.; Dias, J.; Rousseau, C.; Courageux, C.; Brazzolotto, X.; Villa, P.; Obrecht, A. et al.
Source: Self-asserted source
José Dias via Scopus - Elsevier

Chemoselective Hydrogenation of 6-Alkynyl-3-fluoro-2-pyridinaldoximes: Access to First-in-Class 6-Alkyl-3-Fluoro-2-pyridinaldoxime Scaffolds as New Reactivators of Sarin-Inhibited Human Acetylcholinesterase with Increased Blood-Brain Barrier Permeability.

Chemistry (Weinheim an der Bergstrasse, Germany)
2020-10-20 | Journal article
Contributors: José Dias
Source: Self-asserted source
José Dias

Rapid discovery of a selective butyrylcholinesterase inhibitor using structure-based virtual screening.

Bioorganic & medicinal chemistry letters
2020-10-08 | Journal article
Contributors: José Dias
Source: Self-asserted source
José Dias

New evidence for dual binding site inhibitors of acetylcholinesterase as improved drugs for treatment of Alzheimer's disease

Neuropharmacology
2019 | Journal article
EID:

2-s2.0-85066340195

Part of ISBN:

18737064 00283908

Contributors: Zueva, I.; Dias, J.; Lushchekina, S.; Semenov, V.; Mukhamedyarov, M.; Pashirova, T.; Babaev, V.; Nachon, F.; Petrova, N.; Nurullin, L. et al.
Source: Self-asserted source
José Dias via Scopus - Elsevier

Characterization of association of human mitochondrial lysyl-tRNA synthetase with HIV-1 Pol and tRNA<inf>3</inf><sup>Lys</sup>

BMC Biochemistry
2018 | Journal article
EID:

2-s2.0-85044199146

Part of ISBN:

14712091

Contributors: Khoder-Agha, F.; Dias, J.M.; Comisso, M.; Mirande, M.
Source: Self-asserted source
José Dias via Scopus - Elsevier

Structure-Based Optimization of Nonquaternary Reactivators of Acetylcholinesterase Inhibited by Organophosphorus Nerve Agents

Journal of Medicinal Chemistry
2018 | Journal article
EID:

2-s2.0-85052988306

Part of ISBN:

15204804 00222623

Contributors: Santoni, G.; De Sousa, J.; De La Mora, E.; Dias, J.; Jean, L.; Sussman, J.L.; Silman, I.; Renard, P.-Y.; Brown, R.C.D.; Weik, M. et al.
Source: Self-asserted source
José Dias via Scopus - Elsevier

An easy method for the determination of active concentrations of cholinesterase reactivators in blood samples: Application to the efficacy assessment of non quaternary reactivators compared to HI-6 and pralidoxime in VX-poisoned mice

Chemico-Biological Interactions
2017 | Journal article
EID:

2-s2.0-85014772179

Contributors: Calas, A.-G.; Dias, J.; Rousseau, C.; Arboléas, M.; Touvrey-Loiodice, M.; Mercey, G.; Jean, L.; Renard, P.-Y.; Nachon, F.
Source: Self-asserted source
José Dias via Scopus - Elsevier

Association of human mitochondrial lysyl-tRNA synthetase with HIV-1 GagPol does not require other viral proteins

Biochimie Open
2016 | Journal article
EID:

2-s2.0-84961958184

Contributors: Kobbi, L.; Dias, J.; Comisso, M.; Mirande, M.
Source: Self-asserted source
José Dias via Scopus - Elsevier

Synthesis and in vitro evaluation of donepezil-based reactivators and analogues for nerve agent-inhibited human acetylcholinesterase

RSC Advances
2016 | Journal article
EID:

2-s2.0-84959018896

Contributors: Renou, J.; Dias, J.; Mercey, G.; Verdelet, T.; Rousseau, C.; Gastellier, A.-J.; Arboléas, M.; Touvrey-Loiodice, M.; Baati, R.; Jean, L. et al.
Source: Self-asserted source
José Dias via Scopus - Elsevier

Small-angle X-ray solution scattering study of the multi-aminoacyl-tRNA synthetase complex reveals an elongated and multi-armed particle

Journal of Biological Chemistry
2013 | Journal article
EID:

2-s2.0-84882310444

Contributors: Dias, J.; Renault, L.; Pérez, J.; Mirande, M.
Source: Self-asserted source
José Dias via Scopus - Elsevier

Activation of Human Mitochondrial Lysyl-tRNA Synthetase upon Maturation of Its Premitochondrial Precursor

Biochemistry
2012 | Journal article
EID:

2-s2.0-84856439541

Contributors: Dias, J.; Octobre, G.; Kobbi, L.; Comisso, M.; Flisiak, S.; Mirande, M.
Source: Self-asserted source
José Dias via Scopus - Elsevier

Association of mitochondrial lysyl-tRNA synthetase with HIV-1 GagPol involves catalytic domain of the synthetase and transframe and integrase domains of pol

Journal of Molecular Biology
2011 | Journal article
EID:

2-s2.0-79960369440

Contributors: Kobbi, L.; Octobre, G.; Dias, J.; Comisso, M.; Mirande, M.
Source: Self-asserted source
José Dias via Scopus - Elsevier

Association of mitochondrial lysyl-tRNA synthetase with HIV-1 GagPol involves catalytic domain of the synthetase and transframe and integrase domains of Pol

2011 | Other
EID:

2-s2.0-80455162293

Contributors: Kobbi, L.; Dias, J.; Octobre, G.; Comisso, M.; Kaminska, M.; Shalak, V.F.; Mirande, M.
Source: Self-asserted source
José Dias via Scopus - Elsevier

Effects of small molecule modulators on ATP binding to skeletal ryanodine receptor

Protein Journal
2009 | Journal article
EID:

2-s2.0-69549084454

Contributors: Dias, J.M.; Vogel, P.D.
Source: Self-asserted source
José Dias via Scopus - Elsevier

Characteristics of l-carnitine import into heart cells

Biochimie
2008 | Journal article
EID:

2-s2.0-39049170302

Contributors: Rigault, C.; Dias, J.V.; Demarquoy, J.; Le Borgne, F.
Source: Self-asserted source
José Dias via Scopus - Elsevier

Insights into the regulation of the ryanodine receptor: Differential effects of Mg<sup>2+</sup> and Ca<sup>2+</sup> on ATP binding

Biochemistry
2006 | Journal article
EID:

2-s2.0-33747097488

Contributors: Dias, J.M.; Szegedi, C.; Jóna, I.; Vogel, P.D.
Source: Self-asserted source
José Dias via Scopus - Elsevier

Thyroid hormone controls carnitine status through modifications of γ-butyrobetaine hydroxylase activity and gene expression

Cellular and Molecular Life Sciences
2002 | Journal article
EID:

2-s2.0-0036202551

Contributors: Galland, S.; Georges, B.; Le Borgne, F.; Conductier, G.; Viana Dias, J.; Demarquoy, J.
Source: Self-asserted source
José Dias via Scopus - Elsevier