Personal information

fluorous chemistry, process chemistry, organic synthetic chemistry
Japan

Activities

Employment (3)

Meijo Daigaku Nogakubu Daigakuin Nogaku Kenkyuka: Nagoya, Aichi, JP

2005-04-01 to present | Professor (Department of Applied Biological Chemistry)
Employment
Source: Self-asserted source
Masato Matsugi

Osaka University: Suita, JP

2000-04-01 to 2004-03-31 | Assistant Professor (Graduate School of Engineering)
Employment
Source: Self-asserted source
Masato Matsugi

Otsuka Seiyaku Kabushiki Kaisha Tokushima Kenkyujo: Tokushima, JP

1990-04-01 to 2000-03-31
Employment
Source: Self-asserted source
Masato Matsugi

Professional activities (5)

Koeki Shadan Hojin Nihon Nogei Kagakukai: Bunkyo-ku, Tokyo, JP

2008-04-01 to present
Service
Source: Self-asserted source
Masato Matsugi

American Chemical Society: Washington, DC, US

2005-06-14 to present
Membership
Source: Self-asserted source
Masato Matsugi

The Sciety of Synthetic Organic Chemistry Japan: Tokyo, JP

2000-04-01 to present
Membership
Source: Self-asserted source
Masato Matsugi

Nihon Yakugakukai: Shibuya-ku, Tokyo, JP

1997-04-01 to present
Membership
Source: Self-asserted source
Masato Matsugi

Koeki Shadan Hojin Nihon Kagakukai: Chiyoda-ku, Tokyo, JP

1990-04-01 to present
Membership
Source: Self-asserted source
Masato Matsugi

Works (50 of 77)

Items per page:
Page 1 of 2

Synthesis of Sparsomycin via Regioselective Oxidation of Disulfide Intermediate Employing Titanium Mandelate Complex

Synlett
2025-02-12 | Journal article
Contributors: Taichi Kano; Shogo Hata; Shizuku Senoh; Nina Gotoh; Ryusuke Okamoto; Yamato Kato; Masato Matsugi
Source: check_circle
Crossref

Metal-Free Selective Air-Oxidation of Sulfides to Sulfoxides Using 2,2′-Azobis-(2,4-dimethyl-4-methoxyvaleronitrile) (V-70) and Isobutyraldehyde

Synlett
2024-11-15 | Journal article
Contributors: Masato Matsugi; Yamato Kato; Miho Kanoh; Takayuki Shioiri
Source: check_circle
Crossref

Practical Epoxidation of Olefins Using Air and Ubiquitous Iron-Based Fluorous Salen Complex

Molecules
2024-02-22 | Journal article
Contributors: Yamato Kato; Miho Kanoh; Hina Kobayashi; Takayuki Shioiri; Masato Matsugi
Source: check_circle
Crossref
grade
Preferred source (of 2)‎

Asymmetric Henry Reaction Using Cobalt Complexes with Bisoxazoline Ligands Bearing Two Fluorous Tags

Molecules
2023-11-16 | Journal article
Contributors: Kazuki Ishihara; Yamato Kato; Narisa Takeuchi; Yuka Hayashi; Yuna Hagiwara; Shyota Shibuya; Tohya Natsume; Masato Matsugi
Source: check_circle
Crossref
grade
Preferred source (of 2)‎

Cutting edge of diphenyl phosphorazidate (DPPA) as a synthetic reagent – A fifty-year odyssey

Organic Chemistry Frontiers
2022 | Journal article
Contributors: Takayuki Shioiri; Kotaro Ishihara; Masato Matsugi
Source: check_circle
Crossref

Practical synthesis of tetrazoles from amides and phosphorazidates in the presence of aromatic bases

Tetrahedron
2022 | Journal article
EID:

2-s2.0-85123721659

Part of ISSN: 14645416 00404020
Contributors: Ishihara, K.; Ishihara, K.; Tanaka, Y.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Synthesis of carbamoyl azides via the Lossen rearrangement utilizing diphenyl phosphorazidate

Tetrahedron Letters
2022 | Journal article
EID:

2-s2.0-85126883784

Part of ISSN: 18733581 00404039
Contributors: Ishihara, K.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Synthesis of 1,5-Disubstituted Tetrazoles from Nitrones by Using Bis(p-nitrophenyl) Phosphorazidate in the Presence of 4-(Dimethylamino)pyridine

Synlett
2022-05 | Journal article
Part of ISSN: 0936-5214
Part of ISSN: 1437-2096
Source: Self-asserted source
Masato Matsugi

A fluorous proline catalyst immobilized on teflon<sup>®</sup> for highly stereoselective asymmetric aldol reactions

Heterocycles
2021 | Journal article
EID:

2-s2.0-85108372440

Part of ISSN: 18810942 03855414
Contributors: Ishihara, K.; Obayashi, R.; Ohira, M.; Kobayashi, Y.; Ishihara, K.; Kato, Y.; Takeuchi, N.; Mizuno, R.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

A recyclable and highly stereoselective multi-fluorous proline catalyst for asymmetric aldol reactions

Tetrahedron Letters
2020 | Journal article
EID:

2-s2.0-85079186062

Part of ISSN: 18733581 00404039
Contributors: Ishihara, K.; Obayashi, R.; Gotoh, M.; Watanabe, Y.; Kobayashi, Y.; Ishihara, K.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

An Expeditious Approach to Tetrazoles from Amides Utilizing Phosphorazidates

Organic Letters
2020-08-21 | Journal article
Contributors: Kotaro Ishihara; Takayuki Shioiri; Masato Matsugi
Source: check_circle
Crossref
grade
Preferred source (of 2)‎

SNAr azidation of phenolic functions utilizing diphenyl phosphorazidate

Tetrahedron Letters
2020-02 | Journal article
Contributors: Kotaro Ishihara; Takayuki Shioiri; Masato Matsugi
Source: check_circle
Crossref
grade
Preferred source (of 2)‎

Stereospecific synthesis of 1,5-disubstituted tetrazoles from ketoximes via a Beckmann rearrangement facilitated by diphenyl phosphorazidate

Tetrahedron Letters
2019-05 | Journal article
Contributors: Kotaro Ishihara; Takayuki Shioiri; Masato Matsugi
Source: check_circle
Crossref
grade
Preferred source (of 2)‎

Unprecedented Asymmetric Epoxidation of Isolated Carbon-Carbon Double Bonds by a Chiral Fluorous Fe(III) Salen Complex: Exploiting Fluorophilic Effect for Catalyst Design

European Journal of Organic Chemistry
2019-04-09 | Journal article
Part of ISSN: 1434-193X
Source: Self-asserted source
Masato Matsugi
grade
Preferred source (of 3)‎

Activation of grubbs-hoveyda second-generation catalysts employing aromatic ligands bearing a widespread aryl substituent

Heterocycles
2018 | Journal article
EID:

2-s2.0-85064491559

Part of ISSN: 18810942 03855414
Contributors: Kobayashi, Y.; Igarashi, R.; Ishikawa, Y.; Inukai, S.; Shimowaki, K.; Sugiyama, Y.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

A Practical Synthesis of 5-Substituted 1H-Tetrazoles from Aldoximes Employing the Azide Anion from Diphenyl Phosphorazidate

Synthesis
2018-03 | Journal article
Part of ISSN: 0039-7881
Part of ISSN: 1437-210X
Source: Self-asserted source
Masato Matsugi
grade
Preferred source (of 2)‎

Concise synthesis of peptide analogs using a fluorous-fmoc protection strategy

New Horizons of Process Chemistry: Scalable Reactions and Technologies
2017 | Book
EID:

2-s2.0-85034952675

Contributors: Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Grubbs-Hoveyda Second-Generation Catalysts Activated by the Introduction of a Light Fluorous Tag onto the Bidentate Ligands

Synthesis (Germany)
2017 | Journal article
EID:

2-s2.0-85009964742

Contributors: Kobayashi, Y.; Suzumura, N.; Tsuchiya, Y.; Goto, M.; Sugiyama, Y.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Pummerer rearrangement using bis(p-nitrophenyl) phosphorazidate as an azidation reagent: A novel synthesis of azidomethyl sulfides

Tetrahedron Letters
2017 | Journal article
EID:

2-s2.0-85029438177

Contributors: Ishihara, K.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Fluorous Mixture Synthesis of Tripeptides and Pentapeptides Using­ a Fluorous-Fmoc Protection Strategy

Synthesis
2017-02-06 | Journal article
Part of ISSN: 0039-7881
Part of ISSN: 1437-210X
Source: Self-asserted source
Masato Matsugi
grade
Preferred source (of 2)‎

Highly Activated Second-Generation Grubbs-Hoveyda Catalyst Driven by Intramolecular Steric Strain

Synlett
2016 | Journal article
EID:

2-s2.0-84978531778

Contributors: Kobayashi, Y.; Miyazaki, H.; Inukai, S.; Takagi, C.; Makino, R.; Shimowaki, K.; Igarashi, R.; Sugiyama, Y.; Nakamura, S.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Synthesis of 5-Substituted 1 H -Tetrazoles from Aldoximes Using Diphenyl Phosphorazidate

Synlett
2016 | Journal article
EID:

2-s2.0-84976254331

Contributors: Ishihara, K.; Kawashima, M.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

A medium fluorous Grubbs-Hoveyda 2nd generation catalyst for phase transfer catalysis of ring closing metathesis reactions

Tetrahedron Letters
2015 | Journal article
EID:

2-s2.0-84923632904

Contributors: Kobayashi, Y.; Inukai, S.; Kondo, N.; Watanabe, T.; Sugiyama, Y.; Hamamoto, H.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Concise Synthesis of All Stereoisomers of Dendroamide A by Fluorous Mixture Synthesis Based on Fluorous‐Fmoc Protection of Amino Acids

European Journal of Organic Chemistry
2015 | Journal article
EID:

2-s2.0-85027955139

Contributors: Takahashi, H.; Endo, N.; Takanose, H.; Sugiyama, Y.; Eguchi, F.; Oguri, K.; Hamamoto, H.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Development of efficient processes for multi-gram scale and divergent preparation of fluorous-Fmoc reagents

Tetrahedron
2015 | Journal article
EID:

2-s2.0-84931008124

Contributors: Sugiyama, Y.; Endo, N.; Ishihara, K.; Kobayashi, Y.; Hamamoto, H.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Enhancement of stereoselectivities in asymmetric synthesis using fluorinated solvents, auxiliaries, and catalysts

RSC Advances
2015 | Journal article
EID:

2-s2.0-84923869720

Contributors: Sugiishi, T.; Matsugi, M.; Hamamoto, H.; Amii, H.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

S<sub>N</sub>2 displacement at the quaternary carbon center: A novel entry to the synthesis of α,α-disubstituted α-amino acids This Letter is dedicated to the late Professor Harry Wasserman, a great chemist as well as a splendid artist

Tetrahedron Letters
2015 | Journal article
EID:

2-s2.0-84929574032

Contributors: Ishihara, K.; Hamamoto, H.; Matsugi, M.; Shioiri, T.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

A comparative study of the asymmetric epoxidation of aromatic olefins using the first generation manganese salen epoxidation catalysts and their light fluorous variants: An interesting discovery on the use of benzotrifluoride as a cosolvent We dedicate this paper to Prof. Yasuyuki Kita on the occasion of his 70th birthday

Tetrahedron Asymmetry
2014 | Journal article
EID:

2-s2.0-85027924173

Contributors: Kobayashi, Y.; Inukai, S.; Asai, N.; Oyamada, M.; Ikegawa, S.; Sugiyama, Y.; Hamamoto, H.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

A nonenzymatic kinetic resolution of (±)-trans-2-arylcyclohexanols via esterification using polymer-supported DCC, DMAP, and 3 β- acetoxyetienic acid

Synthetic Communications
2013 | Journal article
EID:

2-s2.0-84876189161

Contributors: Shamoto, K.; Miyazaki, A.; Matsukura, M.; Kobayashi, Y.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

A synthesis of all stereoisomers of tenuecyclamide A employing a fluorous-Fmoc strategy

Journal of Organic Chemistry
2013 | Journal article
EID:

2-s2.0-84886379973

Contributors: Sugiyama, Y.; Eguchi, F.; Miyazaki, A.; Hayashi, K.; Takahashi, H.; Hamamoto, H.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Fluorous mixture synthesis of fluorous-Fmoc reagents using a one-pot double tagging strategy

Tetrahedron Letters
2013 | Journal article
EID:

2-s2.0-84875232218

Contributors: Sugiyama, Y.; Ishihara, K.; Masuda, Y.; Kobayashi, Y.; Hamamoto, H.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Liquid-phase split-type combinatorial synthesis of tripeptide derivatives encoded by fluorous fmoc reagents

Synlett
2013 | Journal article
EID:

2-s2.0-84889879796

Contributors: Sugiyama, Y.; Hirose, M.; Matsui, J.; Endo, N.; Hamamoto, H.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

The systematic structure-activity relationship to predict how flavones bind to human androgen receptor for their antagonistic activity

Bioorganic and Medicinal Chemistry
2013 | Journal article
EID:

2-s2.0-84877834098

Contributors: Tamura, H.; Yoshioka, M.; Hasegawa, M.; Hosoda, A.; Matsugi, M.; Akamatsu, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

A fluorous Mukaiyama coupling reagent for a concise condensation reaction: Utility of medium-fluorous strategy

Tetrahedron
2012 | Journal article
EID:

2-s2.0-84859801839

Contributors: Sugiyama, Y.; Kurata, Y.; Kunda, Y.; Miyazaki, A.; Matsui, J.; Nakamura, S.; Hamamoto, H.; Shioiri, T.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

An effective synthesis of 5,4′-disubstituted flavones via a cesium enolate assisted intramolecular ipso-substitution reaction

Chemical and Pharmaceutical Bulletin
2010 | Journal article
EID:

2-s2.0-77955393526

Contributors: Matsugi, M.; Takeda, M.; Takahashi, A.; Tazaki, T.; Tamura, H.; Shioiri, T.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Pronounced rate enhancements in condensation reactions attributed to the fluorous tag in modified Mukaiyama reagents

Tetrahedron Letters
2010 | Journal article
EID:

2-s2.0-70649094342

Contributors: Matsugi, M.; Nakamura, S.; Kunda, Y.; Sugiyama, Y.; Shioiri, T.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Synthesis and RCM reactions using a recyclable grubbs-hoveyda metathesis catalyst activated by a light fluorous tag

Journal of Organic Chemistry
2010 | Journal article
EID:

2-s2.0-78449252048

Contributors: Matsugi, M.; Kobayashi, Y.; Suzumura, N.; Tsuchiya, Y.; Shioiri, T.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

An alternative and facile purification procedure of amidation and esterification reactions using a medium fluorous Mukaiyama reagent

Tetrahedron Letters
2008 | Journal article
EID:

2-s2.0-52949085062

Contributors: Matsugi, M.; Suganuma, M.; Yoshida, S.; Hasebe, S.; Kunda, Y.; Hagihara, K.; Oka, S.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Direct perfluoroalkylation of non-activated aromatic C-H bonds of phenols

Tetrahedron Letters
2008 | Journal article
EID:

2-s2.0-44149100929

Contributors: Matsugi, M.; Hasegawa, M.; Hasebe, S.; Takai, S.; Suyama, R.; Wakita, Y.; Kudo, K.; Imamura, H.; Hayashi, T.; Haga, S.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Simplification of an organic synthetic process based on a light-fluorous strategy

Yuki Gosei Kagaku Kyokaishi/Journal of Synthetic Organic Chemistry
2008 | Journal article
EID:

2-s2.0-52049123871

Contributors: Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Preparation and condensation reactions of a new light-fluorous Mukaiyama reagent: reliable purification with fluorous solid phase extraction for esters and amides

Tetrahedron Letters
2007 | Journal article
EID:

2-s2.0-34247858969

Contributors: Matsugi, M.; Hasegawa, M.; Sadachika, D.; Okamoto, S.; Tomioka, M.; Ikeya, Y.; Masuyama, A.; Mori, Y.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Synthesis of fluorous-FMOC reagents and purification of protected dipeptides with fluorous solid phase extraction

QSAR and Combinatorial Science
2006 | Journal article
EID:

2-s2.0-33749037122

Contributors: Matsugi, M.; Yamanaka, K.; Inomata, I.; Takekoshi, N.; Hasegawa, M.; Curran, D.P.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Efficient synthesis of thioesters and amides from aldehydes by using an intermolecular radical reaction in water

Chemistry - A European Journal
2005 | Journal article
EID:

2-s2.0-12444342979

Contributors: Nambu, H.; Hata, K.; Matsugi, M.; Kita, Y.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Synthesis, reaction, and recycle of light fluorous Grubbs-Hoveyda catalysts for alkene metathesis

Journal of Organic Chemistry
2005 | Journal article
EID:

2-s2.0-14544270505

Contributors: Matsugi, M.; Curran, D.P.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

A novel separation technique of diastereomeric esters of pyridylethanols by extraction: Formal total synthesis of PNU-142721, HIV-1 reverse transcriptase inhibitor

Tetrahedron
2004 | Journal article
EID:

2-s2.0-1642265128

Contributors: Matsugi, M.; Itoh, K.; Nojima, M.; Hagimoto, Y.; Kita, Y.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Fluorous columns are superior to cyclodextrin columns for demixing in fluorous mixture synthesis: When and why to use fluorous silica gel

Synlett
2004 | Journal article
EID:

2-s2.0-3943071029

Contributors: Curran, D.P.; Dandapani, S.; Werner, S.; Matsugi, M.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Reverse fluorous solid-phase extraction: A new technique for rapid separation of fluorous compounds

Organic Letters
2004 | Journal article
EID:

2-s2.0-4344641834

Contributors: Matsugi, M.; Curran, D.P.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

A simple determination method of the absolute configuration of 1-arylethanthiols by an intramolecular CH/π shielding effect in <sup>1</sup>H-NMR of diastereomeric thiol esters

Chemical and Pharmaceutical Bulletin
2003 | Journal article
EID:

2-s2.0-0242349137

Contributors: Matsugi, M.; Hagimoto, Y.; Itoh, K.; Nojima, M.; Kita, Y.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

An efficient methodology for the C-C bond forming radical cyclization of hydrophobic substrates in water: Effect of additive on radical reaction in water

Tetrahedron
2003 | Journal article
EID:

2-s2.0-0037213655

Contributors: Nambu, H.; Anilkumar, G.; Matsugi, M.; Kita, Y.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier

Effective nonenzymatic kinetic resolution of (±)-trans-2-arylcyclohexanols using 3β-acetoxyetienic acid, DCC, and DMAP

Organic Process Research and Development
2003 | Journal article
EID:

2-s2.0-0043246691

Contributors: Matsugi, M.; Hagimoto, Y.; Nojima, M.; Kita, Y.
Source: Self-asserted source
Masato Matsugi via Scopus - Elsevier
Items per page:
Page 1 of 2

Peer review (16 reviews for 9 publications/grants)

Review activity for ACS omega. (1)
Review activity for ACS sustainable chemistry & engineering. (1)
Review activity for Chemistry - an Asian journal. (1)
Review activity for European journal of organic chemistry. (1)
Review activity for Journal of organic chemistry. (4)
Review activity for Organic letters. (4)
Review activity for Organic process research & development. (2)
Review activity for Tetrahedron chem. (1)
Review activity for Tetrahedron letters. (1)