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Japan

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Employment (3)

Kumamoto University: Kumamoto , JP

2016-10-01 to present | Post-doctor Research fellow (Bioorganic & Medicinal Chemistry)
Employment
Source: Self-asserted source
Mohamed

Kumamoto University: Kumamoto, JP

2013-04-01 to 2013-09-31 | Research Student (Bioorganic & Medicinal Chemistry)
Employment
Source: Self-asserted source
Mohamed

National Research Centre: Giza, EG

2009 to 2013-03-31 | Researcher assistant (Chemistry of Natural Compounds)
Employment
Source: Self-asserted source
Mohamed

Education and qualifications (1)

Kumamoto University: Kumamoto, JP

2013-10-01 to 2016-09-26 | PhD (Bioorganic & Medicinal Chemistry)
Education
Source: Self-asserted source
Mohamed

Works (50 of 52)

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Page 1 of 2

Beyond Psychotropic: Potential Repurposing of Fluoxetine toward Cancer Therapy

International Journal of Molecular Sciences
2024-06-07 | Journal article
Contributors: Sultan F. Kadasah; Abdulaziz M. S. Alqahtani; Abdullah Alkhammash; Mohamed O. Radwan
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Discovery of cytotoxic truncated vitamin D derivatives against both bortezomib‐sensitive and bortezomib‐resistant multiple myeloma phenotypes

Medicinal Chemistry Research
2024-05 | Journal article
Contributors: Mohamed O. Radwan; Sawa Sakai; Alaa N. Hassan; Momoko Uesugi; Masaharu Sakamoto; Tsugumasa Toma; Mohammed A. S. Abourehab; Mostafa M. Badran; Hiroshi Tateishi; Nao Nishimura et al.
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Beyond Psychotropic: Repurposing of Fluoxetine Toward Cancer Management and Its Molecular Mechanisms

2024-02-12 | Preprint
Contributors: Sultan F. Kadasah; Abdulaziz M. S. Alqahtani; Mohamed O. Radwan
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Structural Characterization of TRAF6 N-Terminal for Therapeutic Uses and Computational Studies on New Derivatives

Pharmaceuticals
2023-11 | Journal article | Author
Contributors: Omur Guven; Belgin Sever; Faika Başoğlu; Abdulilah Ece; HIROSHI TATEISHI; Ryoko Koga; Mohamed; Nefise Demir; Mustafa Can; Mutlu Dilsiz Aytemir et al.
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Multidisciplinary Digital Publishing Institute

Overview of Ursolic Acid Potential for the Treatment of Metabolic Disorders, Autoimmune Diseases, and Cancers via Nuclear Receptor Pathways

Biomedicines
2023-10-19 | Journal article
Contributors: Sultan F. Kadasah; Mohamed O. Radwan
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Harnessing Oleanolic Acid and Its Derivatives as Modulators of Metabolic Nuclear Receptors

Biomolecules
2023-09-28 | Journal article
Contributors: Mohamed O. Radwan; Sultan F. Kadasah; Salha M. Aljubiri; Abdulmajeed F. Alrefaei; Mahmoud H. El-Maghrabey; Mohamed A. El Hamd; Hiroshi Tateishi; Masami Otsuka; Mikako Fujita
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Gypsogenin Battling for a Front Position in the Pentacyclic Triterpenes Game of Thrones on Anti-Cancer Therapy: A Critical Review—Dedicated to the Memory of Professor Hanaa M. Rady

Molecules
2023-07-27 | Journal article
Contributors: Mohamed O. Radwan; Howaida I. Abd-Alla; Azhaar T. Alsaggaf; Hatem El-Mezayen; Mohammed A. S. Abourehab; Mohamed E. El-Beeh; Hiroshi Tateishi; Masami Otsuka; Mikako Fujita
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New insight into the bioactivity of substituted benzimidazole derivatives: Repurposing from anti-HIV activity to cell migration inhibition targeting hnRNP M

Bioorganic & Medicinal Chemistry
2023-05 | Journal article
Contributors: Mohamed O. Radwan; Tsugumasa Toma; Yuiichi Arakaki; Masahiro Kamo; Naoya Inoue; Ryoko Koga; Masami Otsuka; Hiroshi Tateishi; Mikako Fujita
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In vitro acetylcholinesterase, tyrosinase inhibitory potentials of secondary metabolites from Euphorbia schimperiana and Euphorbia balsamifera

Zeitschrift für Naturforschung C
2023-05-25 | Journal article
Contributors: Salha M. Aljubiri; Eman Abd Elsalam; Faten K. Abd El Hady; Mohamed O. Radwan; Abdulrahman I. Almansour; Kamel H. Shaker
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Design, synthesis, in vitro and in silico characterization of plastoquinone analogs containing piperidine moiety as antimicrobial agents

Journal of Molecular Structure
2023-04 | Journal article
Contributors: Mahmut Yıldız; Hatice Yıldırım; Nilüfer Bayrak; Selin Melis Çakmak; Emel Mataracı-Kara; Berna Özbek-Çelik; Masami Otsuka; Mikako Fujita; Mohamed O. Radwan; Amaç Fatih TuYuN
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A New 1,2-Naphthoquinone Derivative with Anti-lung Cancer Activity

Chemical and Pharmaceutical Bulletin
2022 | Journal article
EID:

2-s2.0-85133295759

Part of ISSN: 13475223 00092363
Contributors: Nakagawa, R.; Tateishi, H.; Radwan, M.O.; Chinen, T.; Ciftci, H.; Iwamaru, K.; Baba, N.; Tominaga, Y.; Koga, R.; Toma, T. et al.
Source: Self-asserted source
Mohamed via Scopus - Elsevier

A vitamin D C/D ring-derived compound with cytotoxicity

Medicinal Chemistry Research
2022 | Journal article
EID:

2-s2.0-85124074961

Part of ISSN: 15548120 10542523
Contributors: Hassan, A.N.; Toma, T.; Ciftci, H.; Biswas, T.; Tahara, Y.; Radwan, M.O.; Tateishi, H.; Fujita, M.; Otsuka, M.
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Mohamed via Scopus - Elsevier

Design, semi-synthesis and examination of new gypsogenin derivatives against leukemia via Abl tyrosine kinase inhibition and apoptosis induction

International Journal of Biological Macromolecules
2022 | Journal article
EID:

2-s2.0-85139361496

Part of ISSN: 18790003 01418130
Contributors: Ulusoy, N.G.; Emirdağ, S.; Sözer, E.; Radwan, M.O.; Çiftçi, H.; Aksel, M.; Bölükbaşı, S.Ş.; Özmen, A.; Yaylı, N.; Karayıldırım, T. et al.
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Mohamed via Scopus - Elsevier

In Vitro and in Silico Study to Assess Toxic Mechanisms of Hybrid Molecules of Quinone-Benzocaine as Plastoquinone Analogues in Breast Cancer Cells

ACS Omega
2022 | Journal article
EID:

2-s2.0-85136691343

Part of ISSN: 24701343
Contributors: Yilmaz Goler, A.M.; Jannuzzi, A.T.; Bayrak, N.; Ylldlz, M.; Ylldlrlm, H.; Otsuka, M.; Fujita, M.; Radwan, M.O.; Tuyun, A.F.
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Mohamed via Scopus - Elsevier

Natural-product-inspired design and synthesis of thiolated coenzyme Q analogs as promising agents against Gram-positive bacterial strains: insights into structure–activity relationship, activity profile, mode of action, and molecular docking

RSC Advances
2022 | Journal article
Contributors: Hatice Yıldırım; Mahmut Yıldız; Nilüfer Bayrak; Emel Mataracı-Kara; Berna Özbek-Çelik; Masami Otsuka; Mikako Fujita; Mohamed O. Radwan; Amaç Fatih TuYuN
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Tranilast-tyrosine hybrid molecule exhibits dual activity: suppression of epithelial-mesenchymal transition and induction of cytotoxicity in cancer cells

Medicinal Chemistry Research
2022 | Journal article
EID:

2-s2.0-85135260960

Part of ISSN: 15548120 10542523
Contributors: Toma, T.; Yamashita, J.; Radwan, M.O.; Badran, M.M.; Masunaga, T.; Kamo, M.; Koga, R.; Okamoto, Y.; Tateishi, H.; Otsuka, M. et al.
Source: Self-asserted source
Mohamed via Scopus - Elsevier

New Insights into the Structural Requirements of Isatin-Derived Pro-Apoptotic Agents against Acute Myeloid Leukemia

Pharmaceuticals
2022-12-17 | Journal article
Contributors: Ahmed K. Hamdy; Takashi Sakamoto; Tsugumasa Toma; Masaharu Sakamoto; Mohammed A. S. Abourehab; Masami Otsuka; Mikako Fujita; Hiroshi Tateishi; Mohamed O. Radwan
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Promising Antibacterial and Antifungal Agents Based on Thiolated Vitamin K3 Analogs: Synthesis, Bioevaluation, Molecular Docking

Pharmaceuticals
2022-05-10 | Journal article
Contributors: Hatice Yıldırım; Mahmut Yıldız; Nilüfer Bayrak; Emel Mataracı-Kara; Mohamed Osman Radwan; Ayse Tarbin Jannuzzi; Masami Otsuka; Mikako Fujita; Amaç Fatih TuYuN
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Discovery of Azaindolin-2-One as a Dual Inhibitor of GSK3β and Tau Aggregation with Potential Neuroprotective Activity

Pharmaceuticals
2022-03-31 | Journal article
Contributors: Taha F. S. Ali; Halil I. Ciftci; Mohamed O. Radwan; Eslam Roshdy; Ahmed M. Shawky; Mohammed A. S. Abourehab; Hiroshi Tateishi; Masami Otsuka; Mikako Fujita
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A new inhibitor of ADAM17 composed of a zinc-binding dithiol moiety and a specificity pocket-binding appendage

Chemical and Pharmaceutical Bulletin
2021 | Journal article
EID:

2-s2.0-85119120620

Part of ISSN: 13475223 00092363
Contributors: Tateishi, H.; Tateishi, M.; Radwan, M.O.; Masunaga, T.; Kawatashiro, K.; Oba, Y.; Oyama, M.; Inoue-Kitahashi, N.; Fujita, M.; Okamoto, Y. et al.
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Mohamed via Scopus - Elsevier

A new series of antileukemic agents: Design, synthesis, in vitro and in silico evaluation of thiazole-based ABL1 kinase inhibitors

Anti-Cancer Agents in Medicinal Chemistry
2021 | Journal article
EID:

2-s2.0-85100658187

Part of ISSN: 18755992 18715206
Contributors: Zeytün, E.; Altıntop, M.D.; Sever, B.; Özdemir, A.; Ellakwa, D.E.; Ocak, Z.; Ciftci, H.I.; Otsuka, M.; Fujita, M.; Radwan, M.O.
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Mohamed via Scopus - Elsevier

New quinoline/1,2,4-triazole hybrids as dual inhibitors of COX-2/5-LOX and inflammatory cytokines: Design, synthesis, and docking study

Journal of Molecular Structure
2021 | Journal article
EID:

2-s2.0-85109201616

Part of ISSN: 00222860
Contributors: Mohassab, A.M.; Hassan, H.A.; Abdelhamid, D.; Gouda, A.M.; Gomaa, H.A.M.; Youssif, B.G.M.; Radwan, M.O.; Fujita, M.; Otsuka, M.; Abdel-Aziz, M.
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Mohamed via Scopus - Elsevier

Genus Sophora: a comprehensive review on secondary chemical metabolites and their biological aspects from past achievements to future perspectives

Archives of Pharmacal Research
2021-11 | Journal article
Contributors: Howaida I. Abd-Alla; Dalila Souguir; Mohamed O. Radwan
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Selective SIRT2 inhibitors as promising anticancer therapeutics: An update from 2016 to 2020

European Journal of Medicinal Chemistry
2021-11 | Journal article
Contributors: Eslam Roshdy; Muhamad Mustafa; Abd El-Rahman Shaltout; Mohamed O. Radwan; Mahmoud A.A. Ibrahim; Mahmoud E. Soliman; Mikako Fujita; Masami Otsuka; Taha F.S. Ali
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EGFR-Targeted Pentacyclic Triterpene Analogues for Glioma Therapy

International Journal of Molecular Sciences
2021-10-11 | Journal article
Contributors: Halil I. Ciftci; Mohamed O. Radwan; Belgin Sever; Ahmed K. Hamdy; Safiye Emirdağ; N. Gokce Ulusoy; Ece Sozer; Mustafa Can; Nurettin Yayli; Norie Araki et al.
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First in class (S,E)-11-[2-(arylmethylene)hydrazono]-PBD analogs as selective CB2 modulators targeting neurodegenerative disorders

Medicinal Chemistry Research
2021-01-04 | Journal article
Contributors: David Mingle; Meirambek Ospanov; Mohamed O. Radwan; Nicole Ashpole; Masami Otsuka; Samir A. Ross; Larry A. Walker; Abbas G. Shilabin; Mohamed A. Ibrahim
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Anticancer activity of Turkish marine extracts: a purple sponge extract induces apoptosis with multitarget kinase inhibition activity

Investigational New Drugs
2020 | Journal article
EID:

2-s2.0-85079719943

Contributors: Ciftci, H.I.; Can, M.; Ellakwa, D.E.; Suner, S.C.; Ibrahim, M.A.; Oral, A.; Sekeroglu, N.; Özalp, B.; Otsuka, M.; Fujita, M. et al.
Source: Self-asserted source
Mohamed via Scopus - Elsevier

Interruption of Vif/Elongin C interaction: In silico and experimental elucidation of the underlying molecular mechanism of benzimidazole-based APOBEC3G stabilizers

Bioorganic and Medicinal Chemistry
2020 | Journal article
EID:

2-s2.0-85081245580

Contributors: Radwan, M.O.; Takaya, D.; Koga, R.; Iwamaru, K.; Tateishi, H.; Ali, T.F.S.; Takaori-Kondo, A.; Otsuka, M.; Honma, T.; Fujita, M.
Source: Self-asserted source
Mohamed via Scopus - Elsevier

Pentabromobenzyl-RP versus triazole-HILIC columns for separation of the polar basic analytes famotidine and famotidone: LC method development combined with in silico tools to follow the potential consequences of famotidine gastric instability

Journal of Pharmaceutical and Biomedical Analysis
2020 | Journal article
EID:

2-s2.0-85083769885

Part of ISSN: 1873264X 07317085
Contributors: El-Shaheny, R.; Radwan, M.O.; Belal, F.; Yamada, K.
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Mohamed via Scopus - Elsevier

In Vitro and In Silico Evaluation of Anticancer Activity of New Indole-Based 1,3,4-Oxadiazoles as EGFR and COX-2 Inhibitors

Molecules
2020-11-07 | Journal article
Contributors: Belgin Sever; Mehlika Dilek Altıntop; Ahmet Özdemir; Gülşen Akalın Çiftçi; Doha E. Ellakwa; Hiroshi Tateishi; Mohamed O. Radwan; Mahmoud A. A. Ibrahim; Masami Otsuka; Mikako Fujita et al.
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Structure activity study of S-trityl-cysteamine dimethylaminopyridine derivatives as SIRT2 inhibitors: Improvement of SIRT2 binding and inhibition

Bioorganic & Medicinal Chemistry Letters
2020-10 | Journal article
Contributors: Mohamed O. Radwan; Halil I. Ciftci; Taha F.S. Ali; Ryoko Koga; Hiroshi Tateishi; Akiko Nakata; Akihiro Ito; Minoru Yoshida; Mikako Fujita; Masami Otsuka
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HSP70 induction by bleomycin metal core analogs

Bioorganic & Medicinal Chemistry Letters
2020-04 | Journal article
Contributors: Taha F.S. Ali; Naomi Taira; Kana Iwamaru; Ryoko Koga; Masahiro Kamo; Mohamed O. Radwan; Hiroshi Tateishi; Hiromasa Kurosaki; Mohamed Abdel-Aziz; Gamal El-Din A.A. Abuo-Rahma et al.
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A novel series of chlorinated plastoquinone analogs: Design, synthesis, and evaluation of anticancer activity

Chemical Biology & Drug Design
2020-03 | Journal article
Contributors: Nilüfer Bayrak; Hatice Yıldırım; Mahmut Yıldız; Mohamed O. Radwan; Masami Otsuka; Mikako Fujita; Halil I. Ciftci; Amaç Fatih Tuyun
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Complementary HPLC, in silico toxicity, and molecular docking studies for investigation of the potential influences of gastric acidity and nitrite content on paracetamol safety

Microchemical Journal
2019 | Journal article
EID:

2-s2.0-85072272679

Contributors: El-Shaheny, R.; Fuchigami, T.; Yoshida, S.; Radwan, M.O.; Nakayama, M.
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Mohamed via Scopus - Elsevier

Design, synthesis, and biological activity of Plastoquinone analogs as a new class of anticancer agents

Bioorganic Chemistry
2019 | Journal article
EID:

2-s2.0-85072526037

Contributors: Bayrak, N.; Yıldırım, H.; Yıldız, M.; Radwan, M.O.; Otsuka, M.; Fujita, M.; Tuyun, A.F.; Ciftci, H.I.
Source: Self-asserted source
Mohamed via Scopus - Elsevier

New SIRT2 inhibitors: Histidine-based bleomycin spin-off

Bioorganic and Medicinal Chemistry
2019 | Journal article
EID:

2-s2.0-85062844025

Contributors: Ali, T.F.S.; Ciftci, H.I.; Radwan, M.O.; Koga, R.; Ohsugi, T.; Okiyama, Y.; Honma, T.; Nakata, A.; Ito, A.; Yoshida, M. et al.
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Mohamed via Scopus - Elsevier

Discovery and structure–activity relationship of plastoquinone analogs as anticancer agents against chronic myelogenous leukemia cells

Archiv der Pharmazie
2019-12 | Journal article
Contributors: Halil I. Ciftci; Nilüfer Bayrak; Hatice Yıldırım; Mahmut Yıldız; Mohamed O. Radwan; Masami Otsuka; Mikako Fujita; Amaç F. Tuyun
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Design, synthesis and biological evaluation of a new series of thiazolyl-pyrazolines as dual EGFR and HER2 inhibitors

European Journal of Medicinal Chemistry
2019-11 | Journal article
Contributors: Belgin Sever; Mehlika Dilek Altıntop; Mohamed O. Radwan; Ahmet Özdemir; Masami Otsuka; Mikako Fujita; Halil I. Ciftci
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Estimation of nizatidine gastric nitrosatability and product toxicity via an integrated approach combining HILIC, in silico toxicology, and molecular docking

Journal of Food and Drug Analysis
2019-10 | Journal article
Contributors: Rania El-Shaheny; Mohamed Radwan; Koji Yamada; Mahmoud El-Maghrabey
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Novel p97/VCP inhibitor induces endoplasmic reticulum stress and apoptosis in both bortezomib‐sensitive and ‐resistant multiple myeloma cells

Cancer Science
2019-10 | Journal article
Contributors: Nao Nishimura; Mohamed O. Radwan; Masayuki Amano; Shinya Endo; Eri Fujii; Hironori Hayashi; Shikiko Ueno; Niina Ueno; Hiro Tatetsu; Hiroyuki Hata et al.
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Antileukemic Activity of Twig Components of Caucasian Beech in Turkey

Molecules
2019-10-25 | Journal article
Contributors: Wataru Shida; Hiroshi Tateishi; Yurika Tahara; Mikako Fujita; Doaa Husham Majeed Alsaadi; Masato Watanabe; Ryoko Koga; Mohamed O. Radwan; Halil I. Ciftci; Sevgi Gezici et al.
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Design, Synthesis and Biological Evaluation of Pentacyclic Triterpene Derivatives: Optimization of Anti-ABL Kinase Activity

Molecules
2019-09-30 | Journal article
Contributors: Halil I. Ciftci; Mohamed O. Radwan; Safiye E. Ozturk; N. Gokce Ulusoy; Ece Sozer; Doha E. Ellakwa; Zeynep Ocak; Mustafa Can; Taha F.S. Ali; Howaida I. Abd-Alla et al.
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Antiproliferative S-Trityl-l-Cysteine -Derived Compounds as SIRT2 Inhibitors: Repurposing and Solubility Enhancement

Molecules
2019-09-10 | Journal article
Contributors: Mohamed O. Radwan; Halil I. Ciftci; Taha F. S. Ali; Doha E. Ellakwa; Ryoko Koga; Hiroshi Tateishi; Akiko Nakata; Akihiro Ito; Minoru Yoshida; Yoshinari Okamoto et al.
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Minimum structural requirements for inhibitors of the zinc finger protein TRAF6

Bioorganic & Medicinal Chemistry Letters
2019-06 | Journal article
Contributors: Mohamed O. Radwan; Ryoko Koga; Tomohiro Hida; Tomohiko Ejima; Yosuke Kanemaru; Hiroshi Tateishi; Yoshinari Okamoto; Jun-ichiro Inoue; Mikako Fujita; Masami Otsuka
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Design, synthesis, and biological evaluation of novel 1,3,4-thiadiazole derivatives as potential antitumor agents against chronic myelogenous leukemia: Striking effect of nitrothiazole moiety

Molecules
2018 | Journal article
EID:

2-s2.0-85039799160

Contributors: Altıntop, M.D.; Ciftci, H.I.; Radwan, M.O.; Sever, B.; Kaplancıklı, Z.A.; Ali, T.F.S.; Koga, R.; Fujita, M.; Otsuka, M.; Zdemir, A.
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Mohamed via Scopus - Elsevier
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The first pentacyclic triterpenoid gypsogenin derivative exhibiting anti-ABL1 kinase and anti-chronic myelogenous leukemia activities

Biological and Pharmaceutical Bulletin
2018 | Journal article
EID:

2-s2.0-85045006057

Contributors: Ciftci, H.I.; Ozturk, S.E.; Ali, T.F.S.; Radwan, M.O.; Tateishi, H.; Koga, R.; Ocak, Z.; Can, M.; Otsuka, M.; Fujita, M.
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Mohamed via Scopus - Elsevier

A Dithiol Compound Binds to the Zinc Finger Protein TRAF6 and Suppresses Its Ubiquitination

ChemMedChem
2017 | Journal article
EID:

2-s2.0-85037681849

Contributors: Koga, R.; Radwan, M.O.; Ejima, T.; Kanemaru, Y.; Tateishi, H.; Ali, T.F.S.; Ciftci, H.I.; Shibata, Y.; Taguchi, Y.; Inoue, J.-I. et al.
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Mohamed via Scopus - Elsevier

A novel inhibitor of farnesyltransferase with a zinc site recognition moiety and a farnesyl group

Bioorganic & Medicinal Chemistry Letters
2017-08 | Journal article
Contributors: Ayumi Tanaka; Mohamed O. Radwan; Akiyuki Hamasaki; Asumi Ejima; Emiko Obata; Ryoko Koga; Hiroshi Tateishi; Yoshinari Okamoto; Mikako Fujita; Mitsuyoshi Nakao et al.
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Marine Inspired 2-(5-Halo-1H-indol-3-yl)-N,N-dimethylethanamines as Modulators of Serotonin Receptors: An Example Illustrating the Power of Bromine as Part of the Uniquely Marine Chemical Space

Marine Drugs
2017-08-09 | Journal article
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Mohamed
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Synthesis and biological activity of new 18β-glycyrrhetinic acid derivatives

Arabian Journal of Chemistry
2016 | Journal article
EID:

2-s2.0-84880343041

Contributors: Radwan, M.O.; Ismail, M.A.H.; El-Mekkawy, S.; Ismail, N.S.M.; Hanna, A.G.
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Mohamed via Scopus - Elsevier
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Peer review (84 reviews for 21 publications/grants)

Review activity for Antibiotics. (2)
Review activity for Arabian journal of chemistry. (4)
Review activity for Archiv der Pharmazie. (2)
Review activity for Biomedicines. (4)
Review activity for Biomolecules. (2)
Review activity for Evidence-based complementary and alternative medicine (1)
Review activity for Frontiers in chemistry. (1)
Review activity for International journal of molecular sciences. (10)
Review activity for Journal of biochemical and molecular toxicology. (1)
Review activity for Journal of marine science and engineering. (4)
Review activity for Letters in drug design & discovery. (2)
Review activity for Life. (2)
Review activity for Marine drugs. (2)
Review activity for Molecules. (26)
Review activity for Natural product research (1)
Review activity for Pharmaceuticals. (10)
Review activity for Pharmaceutics. (4)
Review activity for Scientia pharmaceutica. (3)
Review activity for Scientific reports. (1)
Review activity for Türk biyokimya dergisi. (1)
Review activity for Türk tarım ve doğa bilimleri dergisi. (1)