Personal information

Activities

Employment (4)

University of Leicester: Leicester, Leicester, GB

2010-08-01 to 2016-06-30 | Lecturer of Chemical Biology (Chemistry)
Employment
Source: Self-asserted source
Andrew Jamieson

University of Oxford: Oxford, Oxfordshire, GB

2009-07-01 to 2010-07-30 | Postdoctoral Research Associate (Chemistry)
Employment
Source: Self-asserted source
Andrew Jamieson

Yale University: New Haven, CT, US

2008-07-01 to 2009-06-30 | Postdoctoral Research Fellow (Chemistry)
Employment
Source: Self-asserted source
Andrew Jamieson

University of Montreal: Montreal, Quebec, CA

2007-01-01 to 2008-06-30 | Postdoctoral Research Fellow (Chemistry)
Employment
Source: Self-asserted source
Andrew Jamieson

Education and qualifications (2)

University of Glasgow: Glasgow, Scotland, GB

2003-10-01 to 2006-12-15 | PhD Organic Chemistry (Chemistry)
Education
Source: Self-asserted source
Andrew Jamieson

University of Glasgow: Glasgow, Scotland, GB

1998-10-01 to 2003-06-30 | BSc (Hons) Chemistry with Medicinal Chemistry (Chemistry)
Education
Source: Self-asserted source
Andrew Jamieson

Funding (2)

DNA Templated Synthesis of De Novo Protein β-Motifs

2015-03 to 2017-02 | Grant
Leverhulme Trust (London, GB)
GRANT_NUMBER:

RPG-2014-372

Source: Self-asserted source
Andrew Jamieson

1,3-Diyne Constrained alpha-Helix Peptides: New tools for Interrogating Protein-Protein Interactions

Source: Self-asserted source
Andrew Jamieson via DimensionsWizard

Works (37)

Raman active diyne-girder conformationally constrained p53 stapled peptides bind to MDM2 for visualisation without fluorophores

RSC Chemical Biology
2025 | Journal article
Contributors: Danielle C. Morgan; Laura McDougall; Astrid Knuhtsen; Lori Buetow; Craig F. Steven; Oscar A. Shepperson; Danny T. Huang; Alison N. Hulme; Andrew G. Jamieson
Source: check_circle
Crossref

Targeting PfCLK3 with Covalent Inhibitors: A Novel Strategy for Malaria Treatment

2024-05-21 | Preprint
Contributors: Andrew Jamieson; Skye Brettell; Omar Jahna; Abbey Begen; Gillian Cann; Niniola Olaniyan; Saumya Sharma; Tamas Yelland; Alison Hole; Benazir Alam et al.
Source: check_circle
Crossref

Rotamer-Controlled Dual Emissive α-Amino Acids

Organic Letters
2023-08-11 | Journal article
Contributors: Rochelle McGrory; Danielle C. Morgan; Andrew G. Jamieson; Andrew Sutherland
Source: check_circle
Crossref

Development of Bifunctional, Raman Active Diyne‐Girder Stapled α‐Helical Peptides**

Chemistry – A European Journal
2023-07-20 | Journal article
Contributors: Danielle C. Morgan; Laura McDougall; Astrid Knuhtsen; Andrew G. Jamieson
Source: check_circle
Crossref

Development of bifunctional, Raman active diyne-girder stapled alpha-helical peptides

2023-02-23 | Preprint
Contributors: Andrew Jamieson; Danielle Morgan; Laura McDougall; Astrid Knuhtsen
Source: check_circle
Crossref

Hydroxamic Acid-Modified Peptide Library Provides Insights into the Molecular Basis for the Substrate Selectivity of HDAC Corepressor Complexes

ACS Chemical Biology
2022-09-16 | Journal article
Contributors: Lewis J. Archibald; Edward A. Brown; Christopher J. Millard; Peter J. Watson; Naomi S. Robertson; Siyu Wang; John W. R. Schwabe; Andrew G. Jamieson
Source: check_circle
Crossref

μ‐Conotoxin KIIIA peptidomimetics that block human voltage‐gated sodium channels

Peptide Science
2021-01 | Journal article
Contributors: Astrid Knuhtsen; Rachel Whiting; Fergus S. McWhinnie; Charlotte Whitmore; Brian O. Smith; A. Christopher Green; Christopher M. Timperley; Kenneth I. Kinnear; Andrew G. Jamieson
Source: check_circle
Crossref

A short peptide that preferentially binds c-MYC G-quadruplex DNA

Chemical Communications
2020 | Journal article
Contributors: Aisling Minard; Danielle Morgan; Federica Raguseo; Anna Di Porzio; Denise Liano; Andrew G. Jamieson; Marco Di Antonio
Source: check_circle
Crossref

Conformationally rigid pyrazoloquinazoline α-amino acids: one- and two-photon induced fluorescence

Chemical Communications
2020 | Journal article
Contributors: Jonathan D. Bell; Alexander H. Harkiss; David Nobis; Eilidh Malcolm; Astrid Knuhtsen; Christopher R. Wellaway; Andrew G. Jamieson; Steven W. Magennis; Andrew Sutherland
Source: check_circle
Crossref

Development of Potent PfCLK3 Inhibitors Based on TCMDC-135051 as a New Class of Antimalarials

Journal of Medicinal Chemistry
2020-09-10 | Journal article
Contributors: Amit Mahindra; Omar Janha; Kopano Mapesa; Ana Sanchez-Azqueta; Mahmood M. Alam; Alfred Amambua-Ngwa; Davis C. Nwakanma; Andrew B. Tobin; Andrew G. Jamieson
Source: check_circle
Crossref

α-Conotoxin GI triazole-peptidomimetics: potent and stable blockers of a human acetylcholine receptor

Chemical Science
2019 | Journal article
Contributors: Astrid Knuhtsen; Charlotte Whitmore; Fergus S. McWhinnie; Laura McDougall; Rachel Whiting; Brian O. Smith; Christopher M. Timperley; A. Christopher Green; Kenneth I. Kinnear; Andrew G. Jamieson
Source: check_circle
Crossref

Development of Potent and Selective PfCLK3 Inhibitors Based on GSK-TCMDC151 as a New Class of Antimalarials

2019-09-13 | Other
Contributors: Amit Mahindra; Omar Janha; Kopano Mapesa; Ana Sanchez-Azqueta; Mahmood M. Alam; Andrew Tobin; Andrew Jamieson
Source: check_circle
Crossref

Synthesis of HDAC Substrate Peptidomimetic Inhibitors Using Fmoc Amino Acids Incorporating Zinc-Binding Groups

Organic Letters
2019-05-03 | Journal article
Contributors: Amit Mahindra; Christopher J. Millard; Iona Black; Lewis J. Archibald; John W. R. Schwabe; Andrew G. Jamieson
Source: check_circle
Crossref

Synthesis and Fluorescent Properties of β-Pyridyl α-Amino Acids

The Journal of Organic Chemistry
2019-03-01 | Journal article
Contributors: Alexander H. Harkiss; Jonathan D. Bell; Astrid Knuhtsen; Andrew G. Jamieson; Andrew Sutherland
Source: check_circle
Crossref

Enzymatically-stable oxetane-based dipeptide hydrogels

Chemical Communications
2018 | Journal article
Contributors: Laura McDougall; Emily R. Draper; Jonathan D. Beadle; Michael Shipman; Piotr Raubo; Andrew G. Jamieson; Dave J. Adams
Source: check_circle
Crossref

Lipopeptidomimetics derived from teixobactin have potent antibacterial activity against Staphylococcus aureus

Chemical Communications
2018 | Journal article
Contributors: Georgina C. Girt; Amit Mahindra; Zaaima J. H. Al Jabri; Megan De Ste Croix; Marco R. Oggioni; Andrew G. Jamieson
Source: check_circle
Crossref

Urotensin-II peptidomimetic incorporating a non-reducible 1,5-triazole disulfide bond reveals a pseudo-irreversible covalent binding mechanism to the urotensin G-protein coupled receptor

Organic & Biomolecular Chemistry
2017 | Journal article
Contributors: Salvatore Pacifico; Aidan Kerckhoffs; Andrew J. Fallow; Rachel E. Foreman; Remo Guerrini; John McDonald; David G. Lambert; Andrew G. Jamieson
Source: check_circle
Crossref

Solid-Phase Synthesis of Oxetane Modified Peptides

Organic Letters
2017-06-16 | Journal article
Contributors: Jonathan D. Beadle; Astrid Knuhtsen; Alex Hoose; Piotr Raubo; Andrew G. Jamieson; Michael Shipman
Source: check_circle
Crossref

Insights into the recruitment of class IIa histone deacetylases (HDACs) to the SMRT/NCoR transcriptional repression complex

Journal of Biological Chemistry
2015 | Journal article
EID:

2-s2.0-84937510624

Contributors: Hudson, G.M.; Watson, P.J.; Fairall, L.; Jamieson, A.G.; Schwabe, J.W.R.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

Robust asymmetric synthesis of unnatural alkenyl amino acids for conformationally constrained α-helix peptides

Organic and Biomolecular Chemistry
2014 | Journal article
EID:

2-s2.0-84908073010

Contributors: Aillard, B.; Robertson, N.S.; Baldwin, A.R.; Robins, S.; Jamieson, A.G.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

The ansamycin antibiotic, rifamycin SV, inhibits BCL6 transcriptional repression and forms a complex with the BCL6-BTB/POZ domain

PLoS ONE
2014 | Journal article
EID:

2-s2.0-84897056484

Contributors: Evans, S.E.; Goult, B.T.; Fairall, L.; Jamieson, A.G.; Ko Ferrigno, P.; Ford, R.; Schwabe, J.W.R.; Wagner, S.D.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

Peptide Scanning for Studying Structure-Activity Relationships in Drug Discovery

Chemical Biology and Drug Design
2013 | Journal article
EID:

2-s2.0-84871395889

Contributors: Jamieson, A.G.; Boutard, N.; Sabatino, D.; Lubell, W.D.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

A 1,3-phenyl-linked hydantoin oligomer scaffold as a β-strand mimetic

Chemical Communications
2012 | Journal article
EID:

2-s2.0-84860127595

Contributors: Jamieson, A.G.; Russell, D.; Hamilton, A.D.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

A novel dihydro-pyrazolo(3,4d)(1,2,4)triazolo(1,5a)pyrimidin-4-one (AJ23) is an antagonist at adenosine A1 receptors and enhances consolidation of step-down avoidance

Behavioural Brain Research
2012 | Journal article
EID:

2-s2.0-84864042714

Contributors: Harvey, A.L.; Young, L.C.; Kornisiuk, E.; Snitcofsky, M.; Colettis, N.; Blanco, C.; Jerusalinsky, D.; Jamieson, A.G.; Hartley, R.C.; Stone, T.W.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

Hydrogen-bonded synthetic mimics of protein secondary structure as disruptors of protein-protein interactions.

Current topics in microbiology and immunology
2011 | Journal article
EID:

2-s2.0-79957512405

Contributors: Adler, M.J.; Jamieson, A.G.; Hamilton, A.D.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

Insertion of multiple alpha-amino gamma-lactam (Agl) residues into a peptide sequence by solid-phase synthesis on synphase lanterns.

Biopolymers
2010 | Journal article
EID:

2-s2.0-77951927012

Contributors: Ronga, L.; Jamieson, A.G.; Beauregard, K.; Quiniou, C.; Chemtob, S.; Lubell, W.D.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

Structure-activity analysis of the growth hormone secretagogue GHRP-6 by α- And β-Amino γ-lactam positional scanning

Chemical Biology and Drug Design
2010 | Journal article
EID:

2-s2.0-71449093017

Contributors: Boutard, N.; Jamieson, A.G.; Ong, H.; Lubell, W.D.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

α-Amino-β-hydroxy-γ-lactam for constraining peptide Ser and Tnr residue conformation

Organic Letters
2010 | Journal article
EID:

2-s2.0-77951182664

Contributors: St-Cyr, D.J.; Jamieson, A.G.; Lubell, W.D.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

Portraits of the pioneers of the American Peptide Society.

Advances in experimental medicine and biology
2009 | Journal article
EID:

2-s2.0-66349135131

Contributors: Bourguet, C.B.; Dörr, A.; Godina, T.; Proulx, C.; Fridkin, G.; Jamieson, A.; Sabatino, D.; Kassem, T.; Boutard, N.; Arsenault, J. et al.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

Positional scanning for peptide secondary structure by systematic solid-phase synthesis of amino lactam peptides

Journal of the American Chemical Society
2009 | Journal article
EID:

2-s2.0-67650549812

Contributors: Jamieson, A.G.; Boutard, N.; Beauregard, K.; Bodas, M.S.; Ong, H.; Quiniou, C.; Chemtob, S.; Lubell, W.D.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

Ether-directed palladium(II)-catalysed aza-Claisen rearrangements: studies on the origin of the directing effect

Tetrahedron
2007 | Journal article
EID:

2-s2.0-33846627635

Contributors: Jamieson, A.G.; Sutherland, A.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

Ether-directed, stereoselective aza-claisen rearrangements: Synthesis of the piperidine alkaloid, α-conhydrine

Organic Letters
2007 | Journal article
EID:

2-s2.0-34247466568

Contributors: Jamieson, A.G.; Sutherland, A.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

Palladium(II)-catalysed rearrangement reactions

Current Organic Chemistry
2006 | Journal article
EID:

2-s2.0-33744750539

Contributors: Fanning, K.N.; Jamieson, A.G.; Sutherland, A.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

Scope and limitations of ether-directed, metal-catalysed aza-Claisen rearrangements; Improved stereoselectivity using non-coordinating solvents

Organic and Biomolecular Chemistry
2006 | Journal article
EID:

2-s2.0-33746254995

Contributors: Jamieson, A.G.; Sutherland, A.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

A highly stereoselective ether directed palladium catalysed aza-Claisen rearrangement

Organic and Biomolecular Chemistry
2005 | Journal article
EID:

2-s2.0-15244358225

Contributors: Jamieson, A.G.; Sutherland, A.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

Stereoselective β-hydroxy-α-amino acid synthesis via an ether-directed, palladium-catalysed aza-Claisen rearrangement

Organic and Biomolecular Chemistry
2005 | Journal article
EID:

2-s2.0-27744556864

Contributors: Fanning, K.N.; Jamieson, A.G.; Sutherland, A.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

The first enantioselective synthesis of the amino acid, (2S,3S,4R)-γ-hydroxyisoleucine using a palladium(ii) catalysed 3,3-sigmatropic rearrangement

Organic and Biomolecular Chemistry
2004 | Journal article
EID:

2-s2.0-1842534456

Contributors: Jamieson, A.G.; Sutherland, A.; Willis, C.L.
Source: Self-asserted source
Andrew Jamieson via Scopus - Elsevier

Peer review (32 reviews for 12 publications/grants)

Review activity for Accounts of chemical research. (1)
Review activity for ACS chemical biology. (1)
Review activity for ACS infectious diseases. (1)
Review activity for ACS medicinal chemistry letters. (2)
Review activity for ChemBioChem. (1)
Review activity for Chemistry. (4)
Review activity for ChemMedChem. (2)
Review activity for Current opinion in chemical biology. (1)
Review activity for Journal of medicinal chemistry. (10)
Review activity for Journal of the American Chemical Society. (1)
Review activity for Nature (1)
Review activity for Organic letters. (7)