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Works (29)

Pitfalls of NMDA Receptor Modulation by Neuroactive Steroids. The Effect of Positive and Negative Modulation of NMDA Receptors in an Animal Model of Schizophrenia

Biomolecules
2021-07-14 | Journal article
Part of ISSN: 2218-273X
Source: Self-asserted source
Vojtech Vyklicky

Conformational rearrangement of the NMDA receptor amino-terminal domain during activation and allosteric modulation

Nature Communications
2021-05-11 | Journal article
Contributors: Vojtech Vyklicky; Cherise Stanley; Chris Habrian; Ehud Y. Isacoff
Source: check_circle
Crossref

Palmitoylation Controls NMDA Receptor Function and Steroid Sensitivity

The Journal of Neuroscience
2021-03-10 | Journal article
Contributors: Pavla Hubalkova; Marek Ladislav; Vojtech Vyklicky; Tereza Smejkalova; Barbora Hrcka Krausova; Bohdan Kysilov; Jan Krusek; Zaneta Naimová; Miloslav Korinek; Hana Chodounska et al.
Source: check_circle
Crossref

Site of Action of Brain Neurosteroid Pregnenolone Sulfate at the N-Methyl-D-Aspartate Receptor

The Journal of Neuroscience
2020-07-29 | Journal article
Contributors: Barbora Hrcka Krausova; Bohdan Kysilov; Jiri Cerny; Vojtech Vyklicky; Tereza Smejkalova; Marek Ladislav; Ales Balik; Miloslav Korinek; Hana Chodounska; Eva Kudova et al.
Source: check_circle
Crossref

Conformational pathway provides unique sensitivity to a synaptic mGluR

Nature Communications
2019-12 | Journal article
Part of ISSN: 2041-1723
Source: Self-asserted source
Vojtech Vyklicky
grade
Preferred source (of 2)‎

Genetically Targeted Optical Control of an Endogenous G Protein-Coupled Receptor

Journal of the American Chemical Society
2019-07-24 | Journal article
Part of ISSN: 0002-7863
Part of ISSN: 1520-5126
Source: Self-asserted source
Vojtech Vyklicky

Strong Inhibitory Effect, Low Cytotoxicity and High Plasma Stability of Steroidal Inhibitors of N-Methyl-D-Aspartate Receptors With C-3 Amide Structural Motif

Frontiers in Pharmacology
2018-11-12 | Journal article
Part of ISSN: 1663-9812
Source: Self-asserted source
Vojtech Vyklicky

Positive Modulators of the N-Methyl-d-aspartate Receptor: Structure–Activity Relationship Study of Steroidal 3-Hemiesters

Journal of Medicinal Chemistry
2018-05-24 | Journal article
Part of ISSN: 0022-2623
Part of ISSN: 1520-4804
Source: Self-asserted source
Vojtech Vyklicky

Surface Expression, Function, and Pharmacology of Disease-Associated Mutations in the Membrane Domain of the Human GluN2B Subunit

Frontiers in Molecular Neuroscience
2018-04-06 | Journal article
Part of ISSN: 1662-5099
Source: Self-asserted source
Vojtech Vyklicky

Total Synthesis of ent-Pregnanolone Sulfate and Its Biological Investigation at the NMDA Receptor

Organic Letters
2018-02-16 | Journal article
Part of ISSN: 1523-7060
Part of ISSN: 1523-7052
Source: Self-asserted source
Vojtech Vyklicky

Physicochemical and biological properties of novel amide-based steroidal inhibitors of NMDA receptors

Steroids
2017 | Journal article
Source: Self-asserted source
Vojtech Vyklicky

Analysis of whole-cell NMDA receptor currents

Neuromethods
2016 | Book
EID:

2-s2.0-84942626778

Contributors: Vyklicky, V.; Korinek, M.; Balik, A.; Smejkalova, T.; Krausova, B.; Vyklicky, L.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier
grade
Preferred source (of 2)‎

Neurosteroid-like Inhibitors of N-Methyl-d-aspartate Receptor: Substituted 2-Sulfates and 2-Hemisuccinates of Perhydrophenanthrene

Journal of medicinal chemistry
2016 | Journal article
Source: Self-asserted source
Vojtech Vyklicky

Preferential Inhibition of Tonically over Phasically Activated NMDA Receptors by Pregnane Derivatives.

2016-02 | Journal article
Contributors: Vyklicky V; Smejkalova T; Krausova B; Balik A; Korinek M; Borovska J; Horak M; Chvojkova M; Kleteckova L; Vales K et al.
Source: Self-asserted source
Vojtech Vyklicky via Europe PubMed Central
grade
Preferred source (of 2)‎

A New Class of Potent N-Methyl- d -Aspartate Receptor Inhibitors: Sulfated Neuroactive Steroids with Lipophilic D-Ring Modifications

Journal of Medicinal Chemistry
2015 | Journal article
EID:

2-s2.0-84939159901

Contributors: Kudova, E.; Chodounska, H.; Slavikova, B.; Budesinsky, M.; Nekardova, M.; Vyklicky, V.; Krausova, B.; Svehla, P.; Vyklicky, L.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier

Block of NMDA receptor channels by endogenous neurosteroids: Implications for the agonist induced conformational states of the channel vestibule

Scientific Reports
2015 | Journal article
EID:

2-s2.0-84934990481

Contributors: Vyklicky, V.; Krausova, B.; Cerny, J.; Balik, A.; Zapotocky, M.; Novotny, M.; Lichnerova, K.; Smejkalova, T.; Kaniakova, M.; Korinek, M. et al.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier

Cholesterol modulates open probability and desensitization of NMDA receptors

Journal of Physiology
2015 | Journal article
EID:

2-s2.0-84929502927

Contributors: Korinek, M.; Vyklicky, V.; Borovska, J.; Lichnerova, K.; Kaniakova, M.; Krausova, B.; Krusek, J.; Balik, A.; Smejkalova, T.; Horak, M. et al.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier

Parallel fluorescence and phosphorescence monitoring of singlet oxygen photosensitization in rats

Journal of Innovative Optical Health Sciences
2015 | Journal article
EID:

2-s2.0-84946471407

Contributors: Dědic, R.; Stíbal, A.; Vyklický, V.; Franěk, M.; Svoboda, A.; Hála, J.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier

Structure, function, and pharmacology of NMDA receptor channels

Physiological Research
2014 | Journal article
EID:

2-s2.0-84897608820

Contributors: Vyklicky, V.; Korinek, M.; Smejkalova, T.; Balik, A.; Krausova, B.; Kaniakova, M.; Lichnerova, K.; Cerny, J.; Krusek, J.; Dittert, I. et al.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier

Pregnenolone sulfate activates NMDA receptor channels

Physiological Research
2013 | Journal article
EID:

2-s2.0-84891649635

Contributors: Adamusová, E.; Cais, O.; Vyklický, V.; Kudová, E.; Chodounská, H.; Horák, M.; Vyklický, L.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier

Spectral- and time-resolved phosphorescence of photosensitizers and singlet oxygen: From in vitro towards in vivo

Journal of Luminescence
2013 | Journal article
EID:

2-s2.0-84884682230

Contributors: Vyklický, V.; Dědic, R.; Curkaniuk, N.; Hála, J.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier

Access of inhibitory neurosteroids to the NMDA receptor

British Journal of Pharmacology
2012 | Journal article
EID:

2-s2.0-84860879085

Contributors: Borovska, J.; Vyklicky, V.; Stastna, E.; Kapras, V.; Slavikova, B.; Horak, M.; Chodounska, H.; Vyklicky Jr., L.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier

Key amino acid residues within the third membrane domains of NR1 and NR2 subunits contribute to the regulation of the surface delivery of N-methyl-D-aspartate receptors

Journal of Biological Chemistry
2012 | Journal article
EID:

2-s2.0-84864377667

Contributors: Kaniakova, M.; Krausova, B.; Vyklicky, V.; Korinek, M.; Lichnerova, K.; Vyklicky, L.; Horak, M.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier

Neuroactive steroids with perfluorobenzoyl group

Steroids
2012 | Journal article
EID:

2-s2.0-84865562988

Contributors: Černý, I.; Buděšínský, M.; Pouzar, V.; Vyklický, V.; Krausová, B.; Vyklický Jr., L.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier

Pregnanolone derivatives substituted in 3alpha-position with the cationic group, method of their production, usage and pharmaceutical preparation involving them

2012-02 | Other
Source: Self-asserted source
Vojtech Vyklicky

Azido analogs of neuroactive steroids

Steroids
2011 | Journal article
EID:

2-s2.0-79960440314

Contributors: Vidrna, L.; Černý, I.; Pouzar, V.; Borovská, J.; Vyklický, V.; Vyklický Jr., L.; Chodounská, H.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier

Neurosteroid modulation of N-methyl-d-aspartate receptors: Molecular mechanism and behavioral effects

Steroids
2011 | Journal article
EID:

2-s2.0-80053576102

Contributors: Korinek, M.; Kapras, V.; Vyklicky, V.; Adamusova, E.; Borovska, J.; Vales, K.; Stuchlik, A.; Horak, M.; Chodounska, H.; Vyklicky Jr., L.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier

Singlet oxygen lifetime dependence on photosensitizer concentration in lipid films

Journal of Luminescence
2011 | Journal article
EID:

2-s2.0-79952190297

Contributors: Dědic, R.; Vyklický, V.; Svoboda, A.; Hála, J.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier

Phosphorescence of singlet oxygen and 5,10,15,20-tetrakis(1-methyl-4-pyridinio)porphine: Time and spectral-resolved study

Journal of Molecular Structure
2009 | Journal article
EID:

2-s2.0-65049090653

Contributors: Dědic, R.; Vyklický, V.; Svoboda, A.; Hála, J.
Source: Self-asserted source
Vojtech Vyklicky via Scopus - Elsevier