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Works (12)

Thermodynamics-Guided Design Reveals a Cooperative Hydrogen Bond in DC-SIGN-targeted Glycomimetics

Journal of Medicinal Chemistry
2024-08-22 | Journal article
Contributors: Dilara D. Nemli; Xiaohua Jiang; Roman P. Jakob; Laura Muñoz Gloder; Oliver Schwardt; Said Rabbani; Timm Maier; Beat Ernst; Jonathan Cramer
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Analogues of the pan-selectin antagonist rivipansel (GMI-1070)

European Journal of Medicinal Chemistry
2024-06 | Journal article
Contributors: Beatrice Wagner; Martin Smieško; Roman P. Jakob; Tobias Mühlethaler; Jonathan Cramer; Tim Maier; Said Rabbani; Oliver Schwardt; Beat Ernst
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Combating DC‐SIGN‐mediated SARS‐CoV‐2 dissemination by glycan‐mimicking polymers

Archiv der Pharmazie
2024-04 | Journal article
Contributors: Jonathan Cramer; Xiaohua Jiang; Butrint Aliu; Beat Ernst
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Prodrugs of E‐selectin Antagonists with Enhanced Pharmacokinetic Properties

ChemMedChem
2022-01-05 | Journal article
Contributors: Philipp Dätwyler; Xiaohua Jiang; Beatrice Wagner; Norbert Varga; Tobias Mühlethaler; Katja Hostettler; Said Rabbani; Oliver Schwardt; Beat Ernst
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Poly‐l‐lysine Glycoconjugates Inhibit DC‐SIGN‐mediated Attachment of Pandemic Viruses

ChemMedChem
2021-08-05 | Journal article
Contributors: Jonathan Cramer; Butrint Aliu; Xiaohua Jiang; Timothy Sharpe; Lijuan Pang; Adrian Hadorn; Said Rabbani; Beat Ernst
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Hydroxyl Groups in Synthetic and Natural-Product-Derived Therapeutics: A Perspective on a Common Functional Group

Journal of Medicinal Chemistry
2019-10-24 | Journal article
Contributors: Jonathan Cramer; Christoph P. Sager; Beat Ernst
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Binding of the Bacterial Adhesin FimH to Its Natural, Multivalent High-Mannose Type Glycan Targets

Journal of the American Chemical Society
2019-01-16 | Journal article
Contributors: Maximilian M. Sauer; Roman P. Jakob; Thomas Luber; Fabia Canonica; Giulio Navarra; Beat Ernst; Carlo Unverzagt; Timm Maier; Rudi Glockshuber
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Dynamic Combinatorial Chemistry: A New Methodology Comes of Age

Chemistry – A European Journal
2019-01-02 | Journal article
Contributors: Priska Frei; Rachel Hevey; Beat Ernst
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Selective Inhibitors of Human Neuraminidase 3

Journal of Medicinal Chemistry
2018-03-08 | Journal article
Contributors: Tianlin Guo; Philipp Dätwyler; Ekaterina Demina; Michele R. Richards; Peng Ge; Chunxia Zou; Ruixiang Zheng; Anne Fougerat; Alexey V. Pshezhetsky; Beat Ernst et al.
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What contributes to an effective mannose recognition domain?

Beilstein Journal of Organic Chemistry
2017-12-04 | Journal article
Contributors: Christoph P Sager; Deniz Eriş; Martin Smieško; Rachel Hevey; Beat Ernst
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A Secondary Structural Element in a Wide Range of Fucosylated Glycoepitopes

Chemistry – A European Journal
2017-08-25 | Journal article
Contributors: Thomas Aeschbacher; Mirko Zierke; Martin Smieško; Mayeul Collot; Jean‐Maurice Mallet; Beat Ernst; Frédéric H.‐T. Allain; Mario Schubert
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Urinary Tract Infection: Which Conformation of the Bacterial Lectin FimH Is Therapeutically Relevant?

Journal of Medicinal Chemistry
2017-07-13 | Journal article
Contributors: Katharina Mayer; Deniz Eris; Oliver Schwardt; Christoph P. Sager; Said Rabbani; Simon Kleeb; Beat Ernst
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Peer review (6 reviews for 4 publications/grants)

Review activity for ACS medicinal chemistry letters. (1)
Review activity for Chemistry. (1)
Review activity for ChemMedChem. (1)
Review activity for Journal of medicinal chemistry. (3)