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Works (9)

Novel D2/5-HT receptor modulators related to cariprazine with potential implication to schizophrenia treatment

European Journal of Medicinal Chemistry
2022-03 | Journal article
Contributors: Radomir Juza; Iveta Vojtechova; Kristyna Stefkova-Mazochova; Wim Dehaen; Tomas Petrasek; Lukas Prchal; Tereza Kobrlova; Jiri Janousek; Premysl Vlcek; Eva Mezeiova et al.
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Pharmacokinetic, pharmacodynamic, and behavioural studies of deschloroketamine in Wistar rats

British Journal of Pharmacology
2022-01 | Journal article
Contributors: Kristýna Štefková‐Mazochová; Hynek Danda; Wim Dehaen; Bronislav Jurásek; Klára Šíchová; Nikola Pinterová‐Leca; Vladimír Mazoch; Barbora Hrčka Krausová; Bohdan Kysilov; Tereza Smejkalová et al.
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How to Reward Your Drug Agent?

NeurIPS 2021 Workshop on Deep Generative Models and Downstream Applications
2021 | Conference paper
URI:

https://openreview.net/forum?id=aJt1LUxUIqB

Contributors: Andrea Karlova; Wim Dehaen; Andrei Penciu
Source: Self-asserted source
Wim Dehaen

Molecular Fingerprint VAE

ICML Workshop on Computational Biology 2021
2021 | Conference paper
URI:

https://icml-compbio.github.io/icml-website-2021/2021/papers/WCBICML2021_paper_49.pdf

Contributors: Karlova, Andrea; Dehaen, Wim,; Svozil, Daniel
Source: Self-asserted source
Wim Dehaen

Heterocyclic Cathinones as Inhibitors of Kynurenine Aminotransferase II—Design, Synthesis, and Evaluation

Pharmaceuticals
2021-12-10 | Journal article
Contributors: Michal Maryška; Lucie Svobodová; Wim Dehaen; Martina Hrabinová; Michaela Rumlová; Ondřej Soukup; Martin Kuchař
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Synthesis and In Vitro Evaluation of Novel Dopamine Receptor D2 3,4-dihydroquinolin-2(1H)-one Derivatives Related to Aripiprazole

Biomolecules
2021-08-24 | Journal article
Part of ISSN: 2218-273X
Contributors: Wim Dehaen; Radomir Juza; Kristyna Stefkova; Wim Dehaen; Alena Randakova; Tomas Petrasek; Iveta Vojtechova; Tereza Kobrlova; Lenka Pulkrabkova; Lubica Muckova et al.
Source: Self-asserted source
Wim Dehaen

QSAR-derived affinity fingerprints (part 1): fingerprint construction and modeling performance for similarity searching, bioactivity classification and scaffold hopping

Journal of Cheminformatics
2020-12 | Journal article
Part of ISSN: 1758-2946
Contributors: Wim Dehaen; Ctibor Škuta; Isidro Cortes-Ciriano; Wim Dehaen; Pavel Kříž; Gerard JP van Westen; Igor V. Tetko; Andreas Bender; Daniel Svozil
Source: Self-asserted source
Wim Dehaen

Can X-Ray Powder Diffraction Be a Suitable Forensic Method for Illicit Drug Identification?

Frontiers in Chemistry
2020-06-23 | Journal article
Part of ISSN: 2296-2646
Contributors: Wim Dehaen; Bronislav Jurásek; Vilém Bartůněk; Štěpán Huber; Patrik Fagan; Vladimír Setnička; František Králík; Wim Dehaen; Daniel Svozil; Martin Kuchař
Source: Self-asserted source
Wim Dehaen

Systematic study of interaction of the neutral form of anilines with undecylcalix[4]resorcinarene derivatives by means of potentiometry

Supramolecular Chemistry
2010-07 | Journal article
Part of ISSN: 1061-0278
Part of ISSN: 1029-0478
Contributors: Wim Dehaen; R. Poduval; K. Kurzątkowska; M. Stobiecka; W.F.A. Dehaen; W. Dehaen; H. Radecka; J. Radecki
Source: Self-asserted source
Wim Dehaen

Peer review (3 reviews for 2 publications/grants)

Review activity for Chemické zvesti. (2)
Review activity for Journal of chemical information and modeling. (1)