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Picomolar FKBP inhibitors enabled by a single water-displacing methyl group in bicyclic [4.3.1] aza-amides

Chemical Science
2021 | Journal article
Contributors: Jürgen M. Kolos; Sebastian Pomplun; Sascha Jung; Benedikt Rieß; Patrick L. Purder; Andreas M. Voll; Stephanie Merz; Monika Gnatzy; Thomas M. Geiger; Ingrid Quist-Løkken et al.
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