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Scopus Author ID: 14069230200

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Works (11)

Structure-Based Discovery of Potent, Orally Bioavailable Benzoxazepinone-Based WD Repeat Domain 5 Inhibitors

Journal of Medicinal Chemistry
2023-12-28 | Journal article
DOI: 10.1021/acs.jmedchem.3c01529
Part of ISSN: 0022-2623
Part of ISSN: 1520-4804
Contributors: Kevin B. Teuscher; Jonathan Mills; Jianhua Tian; Changho Han; Kenneth M. Meyers; Jiqing Sai; Taylor M. South; Mackenzie M. Crow; Mayme Van Meveren; John L. Sensintaffar et al.
Source: Self-asserted source
Kenneth Meyers

Structure-based discovery of potent WD repeat domain 5 inhibitors that demonstrate efficacy and safety in preclinical animal models

Proceedings of the National Academy of Sciences
2023-01-03 | Journal article
DOI: 10.1073/pnas.2211297120
Contributors: Kevin B. Teuscher; Somenath Chowdhury; Kenneth M. Meyers; Jianhua Tian; Jiqing Sai; Mayme Van Meveren; Taylor M. South; John L. Sensintaffar; Tyson A. Rietz; Soumita Goswami et al.
Source: check_circle
Crossref

Discovery of Potent Orally Bioavailable WD Repeat Domain 5 (WDR5) Inhibitors Using a Pharmacophore-Based Optimization

Journal of Medicinal Chemistry
2022-04-28 | Journal article
DOI: 10.1021/acs.jmedchem.2c00195
Part of ISSN: 0022-2623
Part of ISSN: 1520-4804
Contributors: Kevin B. Teuscher; Kenneth M. Meyers; Qiangqiang Wei; Jonathan Mills; Jianhua Tian; Joseph Alvarado; Jiqing Sai; Mayme Van Meveren; Taylor M. South; Tyson A. Rietz et al.
Source: Self-asserted source
Kenneth Meyers

Discovery and Structure-Based Optimization of Potent and Selective WD Repeat Domain 5 (WDR5) Inhibitors Containing a Dihydroisoquinolinone Bicyclic Core

Journal of Medicinal Chemistry
2020-01-23 | Journal article
DOI: 10.1021/acs.jmedchem.9b01608
Part of ISSN: 0022-2623
Part of ISSN: 1520-4804
Contributors: Jianhua Tian; Kevin B. Teuscher; Erin R. Aho; Joseph R. Alvarado; Jonathan Mills; Kenneth M. Meyers; Rocco D. Gogliotti; Changho Han; Jonathan D. Macdonald; Jiqing Sai et al.
Source: Self-asserted source
Kenneth Meyers
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Preferred source (of 2)‎

Dihydrobenzisoxazole-4-one compounds are novel selective inhibitors of aldosterone synthase (CYP11B2) with in vivo activity

Bioorganic & Medicinal Chemistry Letters
2018-03 | Journal article
DOI: 10.1016/j.bmcl.2017.12.015
Part of ISSN: 0960-894X
Contributors: Kenneth Meyers; Derek A. Cogan; Jennifer Burke; Raquel Arenas; Michael Balestra; Nicholas F. Brown; Zhidong Chen; Matthew A. Cerny; Holly E. Clifford; Federico Colombo et al.
Source: Self-asserted source
Kenneth Meyers

Aminomethyl tetrahydronaphthalene biphenyl carboxamide MCH-R1 antagonists-Increasing selectivity over hERG

2007 | Journal article
DOI:

10.1016/j.bmcl.2006.10.053

EID:

2-s2.0-33846253270
Contributors: Meyers, K.M.; Kim, N.; Méndez-Andino, J.L.; Hu, X.E.; Mumin, R.N.; Klopfenstein, S.R.; Wos, J.A.; Mitchell, M.C.; Paris, J.L.; Ackley, D.C. et al.
Source: Self-asserted source
Kenneth Meyers via Scopus - Elsevier

Aminomethyl tetrahydronaphthalene ketopiperazine MCH-R1 antagonists-Increasing selectivity over hERG

2007 | Journal article
DOI:

10.1016/j.bmcl.2006.10.052

EID:

2-s2.0-33846262178
Contributors: Meyers, K.M.; Méndez-Andino, J.L.; Colson, A.-O.; Warshakoon, N.C.; Wos, J.A.; Mitchell, M.C.; Hodge, K.M.; Howard, J.M.; Ackley, D.C.; Holbert, J.K. et al.
Source: Self-asserted source
Kenneth Meyers via Scopus - Elsevier

Novel pyrazolopiperazinone- and pyrrolopiperazinone-based MCH-R1 antagonists

2007 | Journal article
DOI:

10.1016/j.bmcl.2006.10.096

EID:

2-s2.0-33846231078
Contributors: Meyers, K.M.; Méndez-Andino, J.; Colson, A.-O.; Hu, X.E.; Wos, J.A.; Mitchell, M.C.; Hodge, K.; Howard, J.; Paris, J.L.; Dowty, M.E. et al.
Source: Self-asserted source
Kenneth Meyers via Scopus - Elsevier

The efficacy and cardiac evaluation of aminomethyl tetrahydronaphthalene ketopiperazines: A novel class of potent MCH-R1 antagonists

2007 | Journal article
DOI:

10.1016/j.bmc.2006.12.028

EID:

2-s2.0-33846638308
Contributors: Méndez-Andino, J.L.; Colson, A.-O.; Meyers, K.M.; Mitchell, M.C.; Hodge, K.; Howard, J.M.; Kim, N.; Ackley, D.C.; Holbert, J.K.; Mittelstadt, S.W. et al.
Source: Self-asserted source
Kenneth Meyers via Scopus - Elsevier

Design and synthesis of substituted quinolines as novel and selective melanin concentrating hormone antagonists as anti-obesity agents

2006 | Journal article
DOI:

10.1016/j.bmcl.2006.07.006

EID:

2-s2.0-33747353075
Contributors: Warshakoon, N.C.; Sheville, J.; Bhatt, R.T.; Ji, W.; Mendez-Andino, J.L.; Meyers, K.M.; Kim, N.; Wos, J.A.; Mitchell, C.; Paris, J.L. et al.
Source: Self-asserted source
Kenneth Meyers via Scopus - Elsevier

Identification of substituted 4-aminopiperidines and 3-aminopyrrolidines as potent MCH-R1 antagonists for the treatment of obesity

2006 | Journal article
DOI:

10.1016/j.bmcl.2006.07.053

EID:

2-s2.0-33748333162
Contributors: Kim, N.; Meyers, K.M.; Mendez-Andino, J.L.; Warshakoon, N.C.; Ji, W.; Wos, J.A.; Colson, A.; Mitchell, M.C.; Davis, J.R.; Pinney, B.B. et al.
Source: Self-asserted source
Kenneth Meyers via Scopus - Elsevier
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