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Works (8)

Chlorinated Enyne Fatty Acid Amides from a Marine Cyanobacterium: Discovery of Taveuniamides L-M and Pharmacological Characterization of Taveuniamide F as a GPCR Antagonist with CNR1 Selectivity

Marine Drugs
2023-12 | Journal article | Author
Contributors: Lobna A. Elsadek; Emma Ellis; Gustavo Seabra; Valerie Paul; Hendrik Luesch
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Multidisciplinary Digital Publishing Institute

Discovery and Anti-Inflammatory Activity of a Cyanobacterial Fatty Acid Targeting the Keap1/Nrf2 Pathway

Marine Drugs
2023-10 | Journal article | Author
Contributors: Fatma H. Al-Awadhi; Emily F. Simon; Na Liu; ranjala ratnayake; Valerie Paul; Hendrik Luesch
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Multidisciplinary Digital Publishing Institute

Isolation and Biological Activity of Iezoside and Iezoside B, SERCA Inhibitors from Floridian Marine Cyanobacteria

Marine Drugs
2023-06 | Journal article | Author
Contributors: Sofia Kokkaliari; Danmeng Luo; Valerie Paul; Hendrik Luesch
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Multidisciplinary Digital Publishing Institute

Anti-Inflammatory Dysidazirine Carboxylic Acid from the Marine Cyanobacterium <i>Caldora</i> sp. Collected from the Reefs of Fort Lauderdale, Florida

Molecules
2022-03 | Journal article | Author
Contributors: Sarath P. Gunasekera; Sofia Kokkaliari; ranjala ratnayake; Thomas Sauvage; Larissa A. H. dos Santos; Hendrik Luesch; Valerie Paul
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Multidisciplinary Digital Publishing Institute

GPCR Pharmacological Profiling of Aaptamine from the Philippine Sponge <i>Stylissa</i> sp. Extends Its Therapeutic Potential for Noncommunicable Diseases

Molecules
2021-09 | Journal article | Author
Contributors: Harmie Luyao; Hendrik Luesch; Mylene Uy
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Multidisciplinary Digital Publishing Institute

Largazole Inhibits Ocular Angiogenesis by Modulating the Expression of VEGFR2 and p21

Marine Drugs
2021-08 | Journal article | Author
Contributors: Beiying Qiu; Alison Tan; Tan Zhi; Qi-Yin Chen; Hendrik Luesch; Xiaomeng Wang
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Multidisciplinary Digital Publishing Institute

Isolation, Structure Elucidation and Biological Evaluation of Lagunamide D: A New Cytotoxic Macrocyclic Depsipeptide from Marine Cyanobacteria

Marine Drugs
2019-02 | Journal article | Author
Contributors: Danmeng Luo; Masteria Yunovilsa Putra; Tao Ye; Valerie Paul; Hendrik Luesch
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Multidisciplinary Digital Publishing Institute

Kempopeptin C, a Novel Marine-Derived Serine Protease Inhibitor Targeting Invasive Breast Cancer

Marine Drugs
2017-09 | Journal article
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Multidisciplinary Digital Publishing Institute

Peer review (33 reviews for 8 publications/grants)

Review activity for ACS chemical biology. (2)
Review activity for ACS medicinal chemistry letters. (2)
Review activity for ACS omega. (1)
Review activity for ACS synthetic biology. (1)
Review activity for Journal of medicinal chemistry. (5)
Review activity for Journal of natural products. (7)
Review activity for Journal of the American Chemical Society. (4)
Review activity for Organic letters. (11)