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Works (10)

The effect of gem-difluorination on the conformation and properties of a model macrocyclic system

Chemical Science
2024 | Journal article
Contributors: T. J. Cogswell; R. J. Lewis; C. Sköld; A. Nordqvist; M. Ahlqvist; L. Knerr
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Incorporation of Intracellular NanoSIMS Tracers to Oligonucleotide Conjugates via Strain Promoted Sydnone–Alkyne Cycloaddition

Bioconjugate Chemistry
2024-07-17 | Journal article
Contributors: Loujahine Lincy-Bianchi; Maximilian Häfner; Cécile Becquart; Carolina Tängemo; Michael E. Kurczy; Claire C. Munier; Laurent Knerr
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Late-Stage Functionalization with Cysteine Staples Generates Potent and Selective Melanocortin Receptor-1 Agonists

Journal of Medicinal Chemistry
2022-10-13 | Journal article
Contributors: Andrew M. White; Anita Dellsén; Niklas Larsson; Quentin Kaas; Frank Jansen; Alleyn T. Plowright; Laurent Knerr; Thomas Durek; David J. Craik
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Glucagon Like Peptide 1 Receptor Agonists for Targeted Delivery of Antisense Oligonucleotides to Pancreatic Beta Cell

Journal of the American Chemical Society
2021-03-10 | Journal article
Contributors: Laurent Knerr; Thazha P. Prakash; Richard Lee; William J. Drury III; Mehran Nikan; Wuxia Fu; Elaine Pirie; Leonardo De Maria; Eric Valeur; Ahlke Hayen et al.
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Stereocontrolled Synthesis of Tetrafluoropentanols: Multivicinal Fluorinated Alkane Units for Drug Discovery

Organic Letters
2019-10-04 | Journal article
Contributors: Patrick Bentler; Nathalie Erdeljac; Kathrin Bussmann; Marie Ahlqvist; Laurent Knerr; Klaus Bergander; Constantin G. Daniliuc; Ryan Gilmour
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Synthesis of Diverse α‐Fluoroalkoxyaryl Derivatives and Their Use for the Generation of Fluorinated Macrocycles

Chemistry – A European Journal
2019-01-24 | Journal article
Contributors: Thomas J. Cogswell; Anders Dahlén; Laurent Knerr
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Targeted delivery of antisense oligonucleotides to pancreatic β-cells

Science Advances
2018-10-05 | Journal article
Contributors: C. Ämmälä; W. J. Drury, III; L. Knerr; I. Ahlstedt; P. Stillemark-Billton; C. Wennberg-Huldt; E.-M. Andersson; E. Valeur; R. Jansson-Löfmark; D. Janzén et al.
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Design of Selective sPLA2-X Inhibitor (−)-2-{2-[Carbamoyl-6-(trifluoromethoxy)-1H-indol-1-yl]pyridine-2-yl}propanoic Acid

ACS Medicinal Chemistry Letters
2018-07-12 | Journal article
Contributors: Fabrizio Giordanetto; Laurent Knerr; Peter Nordberg; Daniel Pettersen; Nidhal Selmi; Hans-Georg Beisel; Hannah de la Motte; Åsa Månsson; Mikael Dahlström; Johan Broddefalk et al.
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Discovery of a Series of Indole-2 Carboxamides as Selective Secreted Phospholipase A2 Type X (sPLA2-X) Inhibitors

ACS Medicinal Chemistry Letters
2018-07-12 | Journal article
Contributors: Laurent Knerr; Fabrizio Giordanetto; Peter Nordberg; Daniel Pettersen; Nidhal Selmi; Hans-Georg Beisel; Hannah de la Motte; Thomas Olsson; Tim D. J. Perkins; Margareta Herslöf et al.
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Direct Synthesis of N-Alkyl Arylglycines by Organocatalytic Asymmetric Transfer Hydrogenation of N-Alkyl Aryl Imino Esters

Organic Letters
2017-10-20 | Journal article
Contributors: Javier Mazuela; Thomas Antonsson; Magnus J. Johansson; Laurent Knerr; Stephen P. Marsden
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Peer review (2 reviews for 2 publications/grants)

Review activity for Israel journal of chemistry. (1)
Review activity for Organic letters. (1)