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Faculty of Pharmacy Cairo University: Cairo, Egypt, EG

Professor (Pharmaceutical Organic Chemistry)
Employment
Source: Self-asserted source
Asmaa Kassab

Works (50 of 51)

Items per page:
Page 1 of 2

New thienopyrimidine-based derivatives: Design, synthesis, and biological evaluation as potent anticancer agents and VEGFR-2 inhibitors

Journal of Molecular Structure
2025-07 | Journal article
Contributors: Myrna A. Farag; Manal M. Kandeel; Asmaa E. Kassab; Samar I. Faggal
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Crossref

Novel Ag(I)‐based 1,2,4‐Oxadiazole Complexes: Synthesis, X‐Ray Crystal Structure, and Biological Evaluation as Anticancer Candidates

Applied Organometallic Chemistry
2025-02 | Journal article
Contributors: Mohammed Salah Ayoup; Rabia E. Alashhab; Saied M. Soliman; Hamida Abdel‐Hamid; David B. Cordes; Aidan P. McKay; Doaa A. Ghareeb; Aliaa Masoud; Asmaa E. Kassab; Mohamed N. Abd Al Moaty
Source: check_circle
Crossref

Design, synthesis, and biological evaluation of 1,2,4-oxadiazole-based derivatives as multitarget anti-Alzheimer agents

RSC Medicinal Chemistry
2024 | Journal article
EID:

2-s2.0-85192483402

Part of ISSN: 26328682
Contributors: Ayoup, M.S.; Barakat, M.R.; Abdel-Hamid, H.; Emam, E.; Al-Faiyz, Y.S.; Masoud, A.A.; Ghareeb, D.A.; Sonousi, A.; Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
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Drug repurposing of fluoroquinolones as anticancer agents in 2023

RSC Advances
2024 | Journal article
Contributors: Asmaa E. Kassab; Rania M. Gomaa; Ehab M. Gedawy
Source: check_circle
Crossref

Fused thiophene as a privileged scaffold: A review on anti-Alzheimer's disease potentials via targeting cholinesterases, monoamine oxidases, glycogen synthase kinase-3, and Aβ aggregation

International Journal of Biological Macromolecules
2024 | Journal article
EID:

2-s2.0-85188718223

Part of ISSN: 18790003 01418130
Contributors: Kassab, A.E.; Gedawy, E.M.; Sayed, A.S.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Medicinal attributes of thienopyrimidine scaffolds incorporating the aryl urea motif as potential anticancer candidates via VEGFR inhibition

Archiv der Pharmazie
2024 | Journal article
EID:

2-s2.0-85192848279

Part of ISSN: 15214184 03656233
Contributors: Farag, M.A.; Kandeel, M.M.; Kassab, A.E.; Faggal, S.I.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
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N-Acylhydrazone Pharmacophore's Analgesic and Anti-inflammatory Profile: Recent Advancements during the Past Ten Years

Current Pharmaceutical Design
2024 | Journal article
EID:

2-s2.0-85185931305

Part of ISSN: 18734286 13816128
Contributors: Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

New 1,2,4-oxadiazole derivatives as potential multifunctional agents for the treatment of Alzheimer’s disease: design, synthesis, and biological evaluation

BMC Chemistry
2024 | Journal article
EID:

2-s2.0-85198413894

Part of ISSN: 2661801X
Contributors: Ayoup, M.S.; Ghanem, M.; Abdel-Hamid, H.; Abu-Serie, M.M.; Masoud, A.; Ghareeb, D.A.; Hawsawi, M.B.; Sonousi, A.; Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

New pyranopyrazole based derivatives: Design, synthesis, and biological evaluation as potential topoisomerase II inhibitors, apoptotic inducers, and antiproliferative agents

Bioorganic Chemistry
2024 | Journal article
EID:

2-s2.0-85184013430

Part of ISSN: 10902120 00452068
Contributors: Sobh, E.A.; Kassab, A.E.; El-Khouly, E.A.; S. A. Hassan, M.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Novel sulfonamide derivatives as multitarget antidiabetic agents: design, synthesis, and biological evaluation

RSC Advances
2024 | Journal article
EID:

2-s2.0-85186711886

Part of ISSN: 20462069
Contributors: Ayoup, M.S.; Khaled, N.; Abdel-Hamid, H.; Ghareeb, D.A.; Nasr, S.A.; Omer, A.; Sonousi, A.; Kassab, A.E.; Eltaweil, A.S.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
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Recent Advancements in Refashioning of NSAIDs and their Derivatives as Anticancer Candidates

Current Pharmaceutical Design
2024 | Journal article
EID:

2-s2.0-85193736438

Part of ISSN: 18734286 13816128
Contributors: Kassab, A.E.; Gedawy, E.M.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Repurposing of Indomethacin and Naproxen as anticancer agents: progress from 2017 to present

RSC Advances
2024 | Journal article
Contributors: Asmaa E. Kassab; Ehab M. Gedawy
Source: check_circle
Crossref

Anticancer agents incorporating the N-acylhydrazone scaffold: Progress from 2017 to present

Archiv der Pharmazie
2023 | Journal article
EID:

2-s2.0-85146328750

Part of ISSN: 15214184 03656233
Contributors: Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
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Benzotriazole scaffold: An overview of antiproliferative potential, mechanisms of action, and structure–activity relationships

Archiv der Pharmazie
2023 | Journal article
EID:

2-s2.0-85161577599

Part of ISSN: 15214184 03656233
Contributors: Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
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Design, synthesis, and biological evaluation of novel ciprofloxacin derivatives as potential anticancer agents targeting topoisomerase II enzyme

Journal of Enzyme Inhibition and Medicinal Chemistry
2023 | Journal article
EID:

2-s2.0-85140857461

Part of ISSN: 14756374 14756366
Contributors: Swedan, H.K.; Kassab, A.E.; Gedawy, E.M.; Elmeligie, S.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Design, synthesis, and biological evaluation of thienopyrimidine derivatives as multifunctional agents against Alzheimer's disease

Drug Development Research
2023 | Journal article
EID:

2-s2.0-85153293384

Part of ISSN: 10982299 02724391
Contributors: Eissa, K.I.; Kamel, M.M.; Mohamed, L.W.; Doghish, A.S.; Alnajjar, R.; Al-Karmalawy, A.A.; Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
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Development of new Alzheimer's disease drug candidates using donepezil as a key model

Archiv der Pharmazie
2023 | Journal article
EID:

2-s2.0-85138601116

Part of ISSN: 15214184 03656233
Contributors: Eissa, K.I.; Kamel, M.M.; Mohamed, L.W.; Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
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New Phenylthiazoles: Design, Synthesis, and Biological Evaluation as Antibacterial, Antifungal, and Anti-COVID-19 Candidates

Chemistry and Biodiversity
2023 | Journal article
EID:

2-s2.0-85174267780

Part of ISSN: 16121880 16121872
Contributors: Shahin, I.G.; Mohamed, K.O.; Taher, A.T.; Elsebaei, M.M.; Mayhoub, A.S.; Kassab, A.E.; Elshewy, A.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
Preferred source (of 2)‎

Pyrazolo[3,4-d]pyrimidine scaffold: A review on synthetic approaches and EGFR and VEGFR inhibitory activities

Archiv der Pharmazie
2023 | Journal article
EID:

2-s2.0-85139223382

Part of ISSN: 15214184 03656233
Contributors: Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
Preferred source (of 2)‎

Recent Advances in the Synthesis of Thiazole Ring: Mini Review

Mini-Reviews in Organic Chemistry
2023 | Journal article
EID:

2-s2.0-85146226269

Part of ISSN: 18756298 1570193X
Contributors: Shahin, I.G.; Mohamed, K.O.; Taher, A.T.; Mayhoub, A.S.; Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Topoisomerase II inhibitors design: Early studies and new perspectives

Bioorganic Chemistry
2023 | Journal article
EID:

2-s2.0-85153105404

Part of ISSN: 10902120 00452068
Contributors: Swedan, H.K.; Kassab, A.E.; Gedawy, E.M.; Elmeligie, S.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Anti-inflammatory activity of pyridazinones: A review

Archiv der Pharmazie
2022 | Journal article
EID:

2-s2.0-85129503849

Part of ISSN: 15214184 03656233
Contributors: Hassan, M.S.A.; Ahmed, E.M.; El-Malah, A.A.; Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
Preferred source (of 2)‎

Design and Synthesis of Novel Celecoxib Analogues with Potential Cytotoxic and Pro-apoptotic Activity against Breast Cancer Cell Line MCF-7

Medicinal Chemistry
2022 | Journal article
EID:

2-s2.0-85132453033

Part of ISSN: 18756638 15734064
Contributors: Abdelhaleem, E.F.; Kassab, A.E.; El-Nassan, H.B.; Khalil, O.M.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Design, synthesis, and biological evaluation of new celecoxib analogs as apoptosis inducers and cyclooxygenase-2 inhibitors

Archiv der Pharmazie
2022 | Journal article
EID:

2-s2.0-85135914610

Part of ISSN: 15214184 03656233
Contributors: Abdelhaleem, E.F.; Kassab, A.E.; El-Nassan, H.B.; Khalil, O.M.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
Preferred source (of 2)‎

Design, synthesis, and biological evaluation of thienopyrimidine and thienotriazine derivatives as multitarget anti-Alzheimer agents

Drug Development Research
2022 | Journal article
EID:

2-s2.0-85132585813

Part of ISSN: 10982299 02724391
Contributors: Eissa, K.I.; Kamel, M.M.; Mohamed, L.W.; Galal, M.A.; Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
Preferred source (of 2)‎

Recent advances in the development of celecoxib analogs as anticancer agents: A review

Archiv der Pharmazie
2022 | Journal article
EID:

2-s2.0-85136510409

Part of ISSN: 15214184 03656233
Contributors: Abdelhaleem, E.F.; Kassab, A.E.; El-Nassan, H.B.; Khalil, O.M.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
Preferred source (of 2)‎

Recent green approaches for the synthesis of pyrazolo[3,4-d]pyrimidines: A mini review

Archiv der Pharmazie
2022 | Journal article
EID:

2-s2.0-85125591996

Part of ISSN: 15214184 03656233
Contributors: Maher, M.; Zaher, A.F.; Mahmoud, Z.; Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
grade
Preferred source (of 2)‎

The Anti-MRSA Activity of Phenylthiazoles: A Comprehensive Review

Current Pharmaceutical Design
2022 | Journal article
EID:

2-s2.0-85144834113

Part of ISSN: 18734286 13816128
Contributors: Shahin, I.G.; Mohamed, K.O.; Taher, A.T.; Mayhoub, A.S.; Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Design, synthesis, anticancer evaluation, and molecular modelling studies of novel tolmetin derivatives as potential VEGFR-2 inhibitors and apoptosis inducers

Journal of Enzyme Inhibition and Medicinal Chemistry
2021 | Journal article
EID:

2-s2.0-85105083820

Part of ISSN: 14756374 14756366
Contributors: Kassab, A.E.; Gedawy, E.M.; Hamed, M.I.A.; Doghish, A.S.; Hassan, R.A.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Design, synthesis and biological evaluation of novel pyrazole sulfonamide derivatives as dual COX-2/5-LOX inhibitors

European Journal of Medicinal Chemistry
2020 | Journal article
EID:

2-s2.0-85078168035

Part of ISSN: 17683254 02235234
Contributors: Gedawy, E.M.; Kassab, A.E.; El Kerdawy, A.M.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Evaluation of N-phenyl-2-aminothiazoles for treatment of multi-drug resistant and intracellular Staphylococcus aureus infections

European Journal of Medicinal Chemistry
2020 | Journal article
EID:

2-s2.0-85088106132

Part of ISSN: 17683254 02235234
Contributors: Shahin, I.G.; Abutaleb, N.S.; Alhashimi, M.; Kassab, A.E.; Mohamed, K.O.; Taher, A.T.; Seleem, M.N.; Mayhoub, A.S.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

New pyridazine derivatives as selective COX-2 inhibitors and potential anti-inflammatory agents; design, synthesis and biological evaluation

Bioorganic Chemistry
2020 | Journal article
EID:

2-s2.0-85076159020

Part of ISSN: 10902120 00452068
Contributors: Ahmed, E.M.; Hassan, M.S.A.; El-Malah, A.A.; Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Novel pyrazolopyrimidine urea derivatives: Synthesis, antiproliferative activity, VEGFR-2 inhibition, and effects on the cell cycle profile

Archiv der Pharmazie
2020 | Journal article
EID:

2-s2.0-85082298628

Part of ISSN: 15214184 03656233
Contributors: Kassab, A.E.; El-Dash, Y.; Gedawy, E.M.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Novel pyrazolo[3,4-d]pyrimidines as potential cytotoxic agents: Design, synthesis, molecular docking and CDK2 inhibition

Anti-Cancer Agents in Medicinal Chemistry
2019 | Journal article
EID:

2-s2.0-85072582649

Part of ISSN: 18755992 18715206
Contributors: Maher, M.; Kassab, A.E.; Zaher, A.F.; Mahmoud, Z.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Novel pyrazolo[3,4-d]pyrimidines: design, synthesis, anticancer activity, dual EGFR/ErbB2 receptor tyrosine kinases inhibitory activity, effects on cell cycle profile and caspase-3-mediated apoptosis

Journal of Enzyme Inhibition and Medicinal Chemistry
2019 | Journal article
EID:

2-s2.0-85060617531

Part of ISSN: 14756374 14756366
Contributors: Maher, M.; Kassab, A.E.; Zaher, A.F.; Mahmoud, Z.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Synthesis and biological evaluation of pyridazinone derivatives as selective COX-2 inhibitors and potential anti-inflammatory agents

European Journal of Medicinal Chemistry
2019 | Journal article
EID:

2-s2.0-85063052475

Part of ISSN: 17683254 02235234
Contributors: Ahmed, E.M.; Kassab, A.E.; El-Malah, A.A.; Hassan, M.S.A.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Design and synthesis of thienopyrimidine urea derivatives with potential cytotoxic and pro-apoptotic activity against breast cancer cell line MCF-7

European Journal of Medicinal Chemistry
2018 | Journal article
EID:

2-s2.0-85033568440

Part of ISSN: 17683254 02235234
Contributors: Abdelhaleem, E.F.; Abdelhameid, M.K.; Kassab, A.E.; Kandeel, M.M.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Design, synthesis and biological evaluation of chromenopyrimidines as potential cytotoxic agents

Future Medicinal Chemistry
2018 | Journal article
EID:

2-s2.0-85048641375

Part of ISSN: 17568927 17568919
Contributors: El-Bakhshawangy, N.M.; El-Nassan, H.B.; Kassab, A.E.; Taher, A.T.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Novel benzotriazole N-acylarylhydrazone hybrids: Design, synthesis, anticancer activity, effects on cell cycle profile, caspase-3 mediated apoptosis and FAK inhibition

Bioorganic Chemistry
2018 | Journal article
EID:

2-s2.0-85049743434

Part of ISSN: 10902120 00452068
Contributors: Kassab, A.E.; Hassan, R.A.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Novel ciprofloxacin hybrids using biology oriented drug synthesis (BIODS) approach: Anticancer activity, effects on cell cycle profile, caspase-3 mediated apoptosis, topoisomerase II inhibition, and antibacterial activity

European Journal of Medicinal Chemistry
2018 | Journal article
EID:

2-s2.0-85043458226

Part of ISSN: 17683254 02235234
Contributors: Kassab, A.E.; Gedawy, E.M.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Synthesis of 4-Heteroaryl–Quinazoline Derivatives as Potential Anti-breast Cancer Agents

Journal of Heterocyclic Chemistry
2017 | Journal article
EID:

2-s2.0-84963829050

Part of ISSN: 19435193 0022152X
Contributors: Kassab, A.E.; Gedawy, E.M.; El-Nassan, H.B.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Design, synthesis, antitumor and antimicrobial activity of novel 6,7-dimethoxyquinazoline derivatives

Heterocycles
2016 | Journal article
EID:

2-s2.0-84962614534

Part of ISSN: 18810942 03855414
Contributors: Kassab, A.E.; Gedawy, E.M.; Mahmoud, Z.; Khattab, R.A.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Synthesis, anticancer activity, effect on cell cycle profile, and apoptosis-inducing ability of novel hexahydrocyclooctathieno[2,3-d]-pyrimidine derivatives

Chemical and Pharmaceutical Bulletin
2016 | Journal article
EID:

2-s2.0-84969555967

Part of ISSN: 13475223 00092363
Contributors: Kassab, A.E.; Gedawy, E.M.; El-Malah, A.A.; Abdelghany, T.M.; Abdel-Bakky, M.S.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Design, synthesis and biological evaluation of new thieno[2,3-d]pyrimidines as anti-inflammatory agents

Anti-Inflammatory and Anti-Allergy Agents in Medicinal Chemistry
2015 | Journal article
EID:

2-s2.0-84958966166

Part of ISSN: 1875614X 18715230
Contributors: El-Malah, A.A.; Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Synthesis and anticancer activity of novel tetrahydroquinoline and tetrahydropyrimidoquinoline derivatives

Medicinal Chemistry Research
2015 | Journal article
EID:

2-s2.0-84937967187

Part of ISSN: 15548120 10542523
Contributors: Gedawy, E.M.; Kassab, A.E.; El-Malah, A.A.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Synthesis, anticancer activity and effects on cell cycle profile and apoptosis of novel thieno[2,3-d]pyrimidine and thieno[3,2-e] triazolo[4,3-c]pyrimidine derivatives

European Journal of Medicinal Chemistry
2015 | Journal article
EID:

2-s2.0-84918589758

Part of ISSN: 17683254 02235234
Contributors: Kandeel, M.M.; Refaat, H.M.; Kassab, A.E.; Shahin, I.G.; Abdelghany, T.M.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Novel tacrine analogs as potential cholinesterase inhibitors in Alzheimer's disease

Archiv der Pharmazie
2014 | Journal article
EID:

2-s2.0-84893767216

Part of ISSN: 03656233 15214184
Contributors: El-Malah, A.; Gedawy, E.M.; Kassab, A.E.; Salam, R.M.A.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Synthesis and anticancer activity of novel 2-pyridyl hexahyrocyclooctathieno[2,3-d]pyrimidine derivatives

European Journal of Medicinal Chemistry
2013 | Journal article
EID:

2-s2.0-84874601067

Part of ISSN: 02235234 17683254
Contributors: Kassab, A.E.; Gedawy, E.M.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Synthesis of effective anticancer thieno [2,3-d] pyrimidine-4-ones and thieno [3,2-e]triazolo[4,3-c]pyrimidines

International Journal of Pharmacy and Pharmaceutical Sciences
2012 | Journal article
EID:

2-s2.0-84862615677

Part of ISSN: 09751491
Contributors: Kandeel, M.M.; Mounir, A.A.; Refaat, H.M.; Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier

Synthesis of potent anticancer thieno[2,3-d]pyrimidine derivatives

Journal of Chemical Research
2012 | Journal article
EID:

2-s2.0-84864592339

Part of ISSN: 17475198
Contributors: Kandeel, M.M.; Mounir, A.A.; Refaat, H.M.; Kassab, A.E.
Source: Self-asserted source
Asmaa Kassab via Scopus - Elsevier
Items per page:
Page 1 of 2

Peer review (14 reviews for 5 publications/grants)

Review activity for ACS omega. (1)
Review activity for Bioorganic chemistry. (7)
Review activity for Chemistry & biodiversity. (1)
Review activity for European journal of medicinal chemistry. (4)
Review activity for International journal of biological macromolecules. (1)