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Synthesis and antiproliferative activity of 3-(2-chloroethyl)-5-methyl-6-phenyl-8-(trifluoromethyl)-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4-(3H)-one

European Journal of Medicinal Chemistry
2015 | Journal article
EID:

2-s2.0-84927130269

Contributors: Maggio, B.; Raimondi, M.V.; Raffa, D.; Plescia, F.; Cascioferro, S.; Cancemi, G.; Tolomeo, M.; Grimaudo, S.; Daidone, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis, antiproliferative activity and possible mechanism of action of novel 2-acetamidobenzamides bearing the 2-phenoxy functionality

Bioorganic and Medicinal Chemistry
2015 | Journal article
EID:

2-s2.0-84940761444

Contributors: Raffa, D.; Maggio, B.; Plescia, F.; Cascioferro, S.; Raimondi, M.V.; Cancemi, G.; D'Anneo, A.; Lauricella, M.; Cusimano, M.G.; Bai, R. et al.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Radical cyclization and 1,5-hydrogen transfer in selected aromatic diazonium salts

Heterocycles
2014 | Journal article
EID:

2-s2.0-84892735193

Contributors: Maggio, B.; Fontana, G.; Raffa, D.; Ferrante, F.; Daidone, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and antiproliferative activity of new derivatives containing the polycyclic system 5,7:7,13-dimethanopyrazolo[3,4-b]pyrazolo[3′,4′:2, 3]azepino[4,5-f]azocine

European Journal of Medicinal Chemistry
2014 | Journal article
EID:

2-s2.0-84889593319

Contributors: Maggio, B.; Raffa, D.; Raimondi, M.V.; Cusimano, M.G.; Plescia, F.; Cascioferro, S.; Cancemi, G.; Lauricella, M.; Carlisi, D.; Daidone, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Unexpected synthesis of 3,5-dimethyl-1-phenyl-1,5-dihydro-4Hpyrazolo[ 4,3-c]quinolin-4-one by non-classical Pschorr reaction, endowed with binding affinity for the central benzodiazepine receptor

Arkivoc
2014 | Journal article
EID:

2-s2.0-84896982905

Contributors: Daidone, G.; Maggio, B.; Raffa, D.; Meneghetti, F.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

2-Cinnamamido, 2-(3-phenylpropiolamido), and 2-(3-phenylpropanamido) benzamides: Synthesis, antiproliferativeactivity, and mechanism of action

European Journal of Medicinal Chemistry
2013 | Journal article
EID:

2-s2.0-84878725211

Contributors: Raffa, D.; Maggio, B.; Raimondi, M.V.; Cusimano, M.G.; Amico, G.; Carollo, A.; Conaldi, P.G.; Bai, R.; Hamel, E.; Daidone, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Non-classical transformation of benzendiazonium hydrogen sulfates. access to 1,3-dimethylisochromeno[4,3-c]pyrazol-5(1h)-one, a potential benzodiazepine receptor ligand

Molecules
2013 | Journal article
EID:

2-s2.0-84886611776

Contributors: Maggio, B.; Raffa, D.; Raimondi, M.V.; Daidone, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and anti-staphylococcal activity of new 4-diazopyrazole derivatives

European Journal of Medicinal Chemistry
2012 | Journal article
EID:

2-s2.0-84867620523

Contributors: Raimondi, M.V.; Maggio, B.; Raffa, D.; Plescia, F.; Cascioferro, S.; Cancemi, G.; Schillaci, D.; Cusimano, M.G.; Vitale, M.; Daidone, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis, benzodiazepine receptor binding and molecular modelling of isochromeno[4,3-c]pyrazol-5(1H)-one derivatives

European Journal of Medicinal Chemistry
2012 | Journal article
EID:

2-s2.0-84864417084

Contributors: Maggio, B.; Raffa, D.; Raimondi, M.V.; Plescia, F.; Trincavelli, M.L.; Martini, C.; Meneghetti, F.; Basile, L.; Guccione, S.; Daidone, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis of substituted 3-amino-N-phenyl-1H-indazole-1-carboxamides endowed with antiproliferative activity

European Journal of Medicinal Chemistry
2011 | Journal article
EID:

2-s2.0-78650512829

Contributors: Maggio, B.; Raimondi, M.V.; Raffa, D.; Plescia, F.; Cascioferro, S.; Plescia, S.; Tolomeo, M.; Di Cristina, A.; Pipitone, R.M.; Grimaudo, S. et al.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis, antiproliferative activity, and mechanism of action of a series of 2-{[(2E)-3-phenylprop-2-enoyl]amino}benzamides

European Journal of Medicinal Chemistry
2011 | Journal article
EID:

2-s2.0-79957501021

Contributors: Raffa, D.; Maggio, B.; Plescia, F.; Cascioferro, S.; Plescia, S.; Raimondi, M.V.; Daidone, G.; Tolomeo, M.; Grimaudo, S.; Di Cristina, A. et al.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and biological evaluation of new indazole derivatives

Arkivoc
2010 | Journal article
EID:

2-s2.0-77958507459

Contributors: Plescia, S.; Raffa, D.; Plescia, F.; Casula, G.; Maggio, B.; Daidone, G.; Raimondi, M.V.; Cusimano, M.G.; Bombieri, G.; Meneghetti, F.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

5-Amino-1-phenyl-3-trifluoromethyl-1H-pyrazole-4-carboxylic acid

Acta Crystallographica Section E: Structure Reports Online
2009 | Journal article
EID:

2-s2.0-70249099199

Contributors: Caruso, F.; Raimondi, M.V.; Daidone, G.; Pettinari, C.; Rossi, M.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

N-(indazolyl)benzamido derivatives as CDK1 inhibitors: Design, synthesis, biological activity, and molecular docking studies

Archiv der Pharmazie
2009 | Journal article
EID:

2-s2.0-66349085643

Contributors: Raffa, D.; Maggio, B.; Cascioferro, S.; Raimondi, M.V.; Daidone, G.; Plescia, S.; Schillaci, D.; Cusimano, M.G.; Titone, L.; Colomba, C. et al.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and antiproliferative activity of 3-amino-N-phenyl-1H-indazole-1-carboxamides

European Journal of Medicinal Chemistry
2009 | Journal article
EID:

2-s2.0-57949110737

Contributors: Raffa, D.; Maggio, B.; Cascioferro, S.; Raimondi, M.V.; Schillaci, D.; Gallo, G.; Daidone, G.; Plescia, S.; Meneghetti, F.; Bombieri, G. et al.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

1,4-Dimethyl-3-phenyl-3H-pyrazolo[3,4-c]isoquinolin-5(4H)-one

Acta Crystallographica Section E: Structure Reports Online
2008 | Journal article
EID:

2-s2.0-43149101312

Contributors: Meneghetti, F.; Bombieri, G.; Maggio, B.; Daidone, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

4-Diazopyrazole derivatives as potential new antibiofilm agents

Chemotherapy
2008 | Journal article
EID:

2-s2.0-52849135125

Contributors: Schillaci, D.; Maggio, B.; Raffa, D.; Daidone, G.; Cascioferro, S.; Cusimano, M.G.; Raimondi, M.V.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Comparative studies of the Pschorr reaction in the pyrazole series. Access to the new dibenzo[e,g]pyrazolo[1,5-a][1,3]diazocine system of pharmaceutical interest

Arkivoc
2008 | Journal article
EID:

2-s2.0-79961238195

Contributors: Maggio, B.; Raffa, D.; Raimondi, M.V.; Cascioferro, S.; Plescia, S.; Sabatino, M.A.; Bombieri, G.; Meneghetti, F.; Daidone, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and induction of G0-G1 phase arrest with apoptosis of 3,5-dimethyl-6-phenyl-8-(trifluoromethyl)-5,6-dihydropyrazolo[3,4-f][1,2,3,5]tetrazepin-4(3H)-one

European Journal of Medicinal Chemistry
2008 | Journal article
EID:

2-s2.0-54049095595

Contributors: Maggio, B.; Raffa, D.; Raimondi, M.V.; Cascioferro, S.; Plescia, F.; Tolomeo, M.; Barbusca, E.; Cannizzo, G.; Mancuso, S.; Daidone, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and biological activity of new anti-inflammatory compounds containing the 1,4-benzodioxine and/or pyrrole system

Bioorganic and Medicinal Chemistry
2007 | Journal article
EID:

2-s2.0-34249650109

Contributors: Harrak, Y.; Rosell, G.; Daidone, G.; Plescia, S.; Schillaci, D.; Pujol, M.D.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis of alkyl-5,8-dimethyl-6-phenyl-5,6-dihydropyrazolo[3,4-f] [1,2,3,5]tetrazepin-4(3H)-ones of pharmaceutical interest

Arkivoc
2006 | Journal article
EID:

2-s2.0-33845693550

Contributors: Maggio, B.; Raffa, D.; Raimondi, M.V.; Plescia, F.; Cascioferro, S.; Daidone, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Comparative structural studies of4-diazopyrazole derivatives by X-ray diffraction and theoretical investigation

Heterocycles
2005 | Journal article
EID:

2-s2.0-33646878312

Contributors: Daidone, G.; Maggio, B.; Raimondi, M.V.; Bombieri, G.; Marchini, N.; Artali, R.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Nonclassical Pschorr and Sandmeyer reactions in pyrazole series

Helvetica Chimica Acta
2005 | Journal article
EID:

2-s2.0-24144479382

Contributors: Maggio, B.; Daidone, G.; Raffa, D.; Plescia, S.; Bombieri, G.; Meneghetti, F.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Erratum: Synthesis, cytotoxicity, and inhibitory effects on tubulin polymerization of a new 3-heterocyclo substituted 2-styrylquinazolinones (European Journal of Medicinal Chemistry (2004) 39 (299-304) DOI: 10.1016/j.ejmech.2003.12.009.)

European Journal of Medicinal Chemistry
2004 | Journal article
EID:

2-s2.0-3242716034

Contributors: Raffa, D.; Edler, M.C.; Daidone, G.; Maggio, B.; Merikech, M.; Plescia, S.; Schillaci, D.; Bai, R.; Hamel, E.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and antileukemic activity of new 3-(1-phenyl-3-methylpyrazol-5- yl)-2-styrylquinazolin-4(3H)-ones

Farmaco
2004 | Journal article
EID:

2-s2.0-1342300596

Contributors: Raffa, D.; Daidone, G.; Maggio, B.; Cascioferro, S.; Plescia, F.; Schillaci, D.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and antileukemic activity of new 3-(5-methylisoxazol-3-yl) and 3-(pyrimidin-2-yl)-2-styrylquinazolin-4(3H)-ones

Farmaco
2004 | Journal article
EID:

2-s2.0-2642523539

Contributors: Raffa, D.; Daidone, G.; Maggio, B.; Cascioferro, S.; Plescia, F.; Schillaci, D.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and antiproliferative activity of triazenoindazoles and triazenopyrazoles: A comparative study

European Journal of Medicinal Chemistry
2004 | Journal article
EID:

2-s2.0-1642346523

Contributors: Daidone, G.; Raffa, D.; Maggio, B.; Raimondi, M.V.; Plescia, F.; Schillaci, D.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and in vitro antileukemic activity of new 4-triazenopyrazole derivatives

Farmaco
2004 | Journal article
EID:

2-s2.0-2142781641

Contributors: Daidone, G.; Maggio, B.; Raffa, D.; Plescia, S.; Schillaci, D.; Raimondi, M.V.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis, cytotoxicity, and inhibitory effects on tubulin polymerization of a new 3-heterocyclo substituted 2-styrylquinazolinones

European Journal of Medicinal Chemistry
2004 | Journal article
EID:

2-s2.0-1842557498

Contributors: Raffa, D.; Edler, M.C.; Daidone, G.; Maggio, B.; Merickech, M.; Plescia, S.; Schillaci, D.; Bai, R.; Hamel, E.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and antifungal activity of new N-(1-phenyl-4-carbetoxypyrazol-5- yl)-, N-(indazol-3-yl)- and N-(indazol-5-yl)-2-iodobenzamides

Farmaco
2002 | Journal article
EID:

2-s2.0-0036516935

Contributors: Raffa, D.; Daidone, G.; Plescia, F.; Schillaci, D.; Maggio, B.; Torta, L.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and antimicrobial evaluation of new phenoxyacetamide derivatives

Bollettino Chimico Farmaceutico
2002 | Journal article
EID:

2-s2.0-0036269808

Contributors: Raffa, D.; Migliara, O.; Daidone, G.; Maggio, B.; Schiilaci, D.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis of pyrazole-4-carbohydrazide derivatives of pharmaceuticalinterest

Arkivoc
2002 | Journal article
EID:

2-s2.0-3242742838

Contributors: Daidone, G.; Raffa, D.; Plescia, F.; Maggio, B.; Roccaro, A.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Phenylamides of 1-phenyl (or methyl)-5-benzamidopyrazole-4-carboxylic acid as vratizolin analogs with analgesic and antiinflammatory activities

Archiv der Pharmazie
2001 | Journal article
EID:

2-s2.0-0035014618

Contributors: Daidone, G.; Plescia, F.; Maggio, B.; Raffa, D.; Cutuli, V.M.C.; Mangano, N.G.; Caruso, A.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and pharmacological study of ethyl 1-methyl-5-(substituted 3,4-dihydro-4-oxoquinazolin-3-yl)-1H-pyrazole-4-acetates

European Journal of Medicinal Chemistry
2001 | Journal article
EID:

2-s2.0-0035441090

Contributors: Maggio, B.; Daidone, G.; Raffa, D.; Plescia, S.; Mantione, L.; Cutuli, V.M.C.; Mangano, N.G.; Caruso, A.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and antifungal activity of new N-isoxazolyl-2-iodobenzamides

Farmaco
1999 | Journal article
EID:

2-s2.0-0032946049

Contributors: Raffa, D.; Daidone, G.; Maggio, B.; Schillaci, D.; Plescia, F.; Torta, L.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and antiproliferative activity of novel 3-(indazol-3-yl)- quinazolin-4(3H)-one and 3-(indazol-3-yl)-benzotriazin-4(3H)-one derivatives

Archiv der Pharmazie
1999 | Journal article
EID:

2-s2.0-0032830929

Contributors: Raffa, D.; Daidone, G.; Maggio, B.; Schillaci, D.; Plescia, F.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and pharmacological activities of novel 3-(isoxazol-3-yl)- quinazolin-4(3H)-one derivatives

Archiv der Pharmazie
1999 | Journal article
EID:

2-s2.0-0033030420

Contributors: Daidone, G.; Raffa, D.; Maggio, B.; Plescia, F.; Cutuli, V.M.C.; Mangano, N.G.; Caruso, A.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis of new 3-(3-phenyl-isoxazol-5-yl) or 3-[(3-phenyl-isoxazol-5- yl)amino] substituted 4(3H)-quinazolinone derivatives with antineoplastic activity

Pharmazie
1999 | Journal article
EID:

2-s2.0-0033029184

Contributors: Raffa, D.; Daidone, G.; Schillaci, D.; Maggio, B.; Plescia, F.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Antimicrobial and antineoplastic activities of new 4-diazopyrazole derivatives

European Journal of Medicinal Chemistry
1998 | Journal article
EID:

2-s2.0-0032104228

Contributors: Daidone, G.; Maggio, B.; Plescia, S.; Raffa, D.; Musiu, C.; Milia, C.; Perra, G.; Marongiu, M.E.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Consecutive Pschorr-Sandmeyer reactions in a pyrazole series. Part 2. Access to the [2]benzopyrano[4,3-c]pyrazole system of pharmaceutical interest

Journal of the Chemical Society - Perkin Transactions 1
1998 | Journal article
EID:

2-s2.0-33748654451

Contributors: Daidone, G.; Maggio, B.; Raffa, D.; Plescia, S.; Benetollo, F.; Bombieri, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and pharmacological evaluation of 1-methyl-5-[substituted-4 (3H)-oxo- 1,2,3-benzotriazin-3-yl] 1H-pyrazole-4-acetic acid derivatives

Farmaco
1998 | Journal article
EID:

2-s2.0-0032580694

Contributors: Daidone, G.; Maggio, B.; Plescia, S.; Raffa, D.; Schillaci, D.; Migliara, O.; Caruso, A.; Cutuli, V.M.C.; Amico-Roxas, M.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis of novel pyrazole derivatives of pharmaceutical interest

Pharmazie
1998 | Journal article
EID:

2-s2.0-0031808650

Contributors: Migliara, O.; Daidone, G.; Plescia, S.; Schillaci, D.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and antineoplastic activity of new 4-diazopyrazole derivatives

Farmaco
1997 | Journal article
EID:

2-s2.0-0031425631

Contributors: Daidone, G.; Maggio, B.; Raffa, D.; Schillaci, D.; Plescia, S.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

One-step synthesis, crystallographic studies and antimicrobial activity of new 4-diazopyrazole derivatives

European Journal of Medicinal Chemistry
1996 | Journal article
EID:

2-s2.0-0029950195

Contributors: Daidone, G.; Bajardi, M.L.; Plescia, S.; Raffa, D.; Schillaci, D.; Maggio, B.; Benetollo, F.; Bombieri, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis, crystallographic studies and biological evaluation of some 2-substituted 3-indazolyl-4(3H)-quinazolinones and 3-indazolyl-4(3H)-benzotriazinones

Heterocycles
1996 | Journal article
EID:

2-s2.0-0001459587

Contributors: Daidone, G.; Plescia, S.; Raffa, D.; Schillaci, D.; Maggio, B.; Benetollo, F.; Bombieri, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Facile synthesis of 5-benzamido-4-diazopyrazole derivatives, a class of biologically active agents and key intermediates

Synthetic Communications
1995 | Journal article
EID:

2-s2.0-0028957070

Contributors: Daidone, G.; Bajardi, M.L.; Raffa, D.; Maggio, B.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis of new 2-{[(phenoxy or phenyl)acetyl]amino}benzoic acid derivatives as 3α-hydroxysteroid dehydrogenase inhibitors and potential antiinflammatory agents

Archiv der Pharmazie
1995 | Journal article
EID:

2-s2.0-0028805553

Contributors: Daidone, G.; Plescia, S.; Bajardi, M.L.; Schillaci, D.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

3α-Hydroxysteroid dehydrogenase inhibitory activity of some N(3)-(1-R-4-carboxypyrazol-5-yl)-1,2,3-benzotriazin-4(3H)-one and quinazolin-4(3H)-one acids

Farmaco
1994 | Journal article
EID:

2-s2.0-0027999028

Contributors: Plescia, S.; Raffa, D.; Daidone, G.; Schillaci, D.; Maggio, B.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Synthesis and pharmacological study of ethyl 1-methyl-5-[2-substituted-4-oxo-3(4H)-quinazolinyl]-1H-pyrazole-4-acetates

European Journal of Medicinal Chemistry
1994 | Journal article
EID:

2-s2.0-0028046743

Contributors: Daidone, G.; Maggio, B.; Raffa, D.; Plescia, S.; Bajardi, M.; Caruso, A.; Cutuli, V.; Amico-Roxas, M.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier

Modifications and extensions of the Pschorr reaction in pyrazole series. Access to the [2]benzopyrano[4,3-c]pyrazole system of pharmaceutical interest

Journal of the Chemical Society, Perkin Transactions 1
1993 | Journal article
EID:

2-s2.0-37049071378

Contributors: Daidone, G.; Plescia, S.; Maggio, B.; Sprio, V.; Benetollo, F.; Bombieri, G.
Source: Self-asserted source
Giuseppe Daidone via Scopus - Elsevier
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