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King's College London: London, GB

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King's College London

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Development of small-molecule fluorescent probes targeting neutrophils via N-formyl peptide receptors

RSC Medicinal Chemistry
2025 | Journal article
Contributors: Qi Xu; Kalwant S. Authi; Liliya N. Kirpotina; Igor A. Schepetkin; Mark T. Quinn; Agostino Cilibrizzi
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Crossref

Beyond transition block metals: exploring the reactivity of phosphine PTA and its oxide [PTA(O)] towards gallium(iii)

RSC Advances
2024 | Journal article
Contributors: Antonella Guerriero; Andrea Ienco; Thomas Hicks; Agostino Cilibrizzi
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‘Main Mechanical Forces-Chemical Interactions’ Interplay as a Tool to Elucidate Folding Mechanisms

Peptide Science
2024-09 | Journal article | Author
SOURCE-WORK-ID:

086d2df0-f7a4-4571-afc7-69d7764b66a2

EID:

2-s2.0-85194840754

Contributors: Michele Larocca; Giuseppe Floresta; Daniele Verderese; agostino cilibrizzi
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King's College London

Dominant Chemical Interactions Governing the Folding Mechanism of Oligopeptides

International Journal of Molecular Sciences
2024-09-04 | Journal article
Contributors: Michele Larocca; Giuseppe Floresta; Daniele Verderese; Agostino Cilibrizzi
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[68Ga]Ga-Schizokinen, a Potential Radiotracer for Selective Bacterial Infection Imaging

ACS Infectious Diseases
2024-08-09 | Journal article
Contributors: Asma Akter; George Firth; Afnan M. F. Darwesh; Margaret S. Cooper; Hataichanok Chuljerm; Agostino Cilibrizzi; Philip J. Blower; Robert C. Hider; Oliver Lyons; Silke Schelenz et al.
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[68Ga]Ga-Schizokinen, a Potential Radiotracer for Selective Bacterial Infection Imaging

ACS Infectious Diseases
2024-07-16 | Journal article | Author
SOURCE-WORK-ID:

9773ddac-976a-4987-982b-a1adceb0e908

Contributors: ASMA AKTER; George Firth; Afnan Darwesh; Maggie Cooper; Hataichanok Chuljerm; agostino cilibrizzi; Philip Blower; Robert Hider; Oliver Lyons; Silke Schelenz et al.
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King's College London

New quinoline-based PDE4 inhibitors through GSK-256066 fragment-based elaboration

JOURNAL OF MOLECULAR STRUCTURE
2024-01-05 | Journal article | Author
SOURCE-WORK-ID:

c8b27f72-9c53-48c7-b8d2-5f085a5ddb8c

EID:

2-s2.0-85172664100

Contributors: Letizia Crocetti; Maria Paola Giovannoni; Claudia Vergelli; Gabriella Guerrini; Fabrizio Melani; agostino cilibrizzi
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King's College London
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Evaluating thermogravimetric analysis for the measurement of drug loading in mesoporous silica nanoparticles (MSNs)

THERMOCHIMICA ACTA
2023-12 | Journal article | Author
SOURCE-WORK-ID:

8422baac-5fb7-409a-a6ed-4f93527b44f6

EID:

2-s2.0-85175143723

Contributors: M. Almaghrabi; A. Alqurshi; S. A. Jadhav; F. Mazzacuva; agostino cilibrizzi; Bahijja Tolulope Abraham; Paul Royall
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King's College London

Optimization of 4-amino-pyridazin-3(2H)-one as a valid core scaffold for FABP4 inhibitors

Archiv Der Pharmazie
2023-10 | Journal article | Author
SOURCE-WORK-ID:

61fc823b-8cc5-4ecb-8ac2-7272e34a0b6e

EID:

2-s2.0-85166415318

Contributors: Giuseppe Floresta; Letizia Crocetti; Renan Rodrigues de Oliveira Silva; Vincenzo Patamia; Francesca Mazzacuva; Yu Chee Sonia Chen; Claudia Vergelli; agostino cilibrizzi
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King's College London
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Non-salt based co-amorphous formulation produced by freeze-drying

INTERNATIONAL JOURNAL OF PHARMACEUTICS
2023-10-15 | Journal article | Author
SOURCE-WORK-ID:

5a81a592-2785-475c-93ba-ac5cc690287d

EID:

2-s2.0-85171884163

Contributors: Mohammed Suleiman Alsalhi; Paul Royall; Hisham Al-Obaidi; Alyaa Alsalhi; agostino cilibrizzi; Ka Lung Andrew Chan
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King's College London
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Optical Imaging Opportunities to Inspect the Nature of Cytosolic Iron Pools

Molecules
2023-09-06 | Journal article | Author
SOURCE-WORK-ID:

a3262653-b9a2-45eb-a31b-02a6aee84a56

EID:

2-s2.0-85172775134

Contributors: Robert Charles Hider; Charareh Pourzand; Yongmin Ma; agostino cilibrizzi
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King's College London
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PDE4 Inhibitors

International Journal of Molecular Sciences
2023-07-15 | Journal article | Author
SOURCE-WORK-ID:

83abbbd4-c954-4348-b70e-042033a67efb

EID:

2-s2.0-85166029697

Contributors: Jian Jin; Francesca Mazzacuva; Letizia Crocetti; Maria Paola Giovannoni; agostino cilibrizzi
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King's College London
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Steered Molecular Dynamics Simulations Study on FABP4 Inhibitors

Molecules
2023-03-17 | Journal article | Author
SOURCE-WORK-ID:

2b9c789d-8c39-4743-b396-c067a734f0c6

EID:

2-s2.0-85151107971

Contributors: Rosario Tomarchio; Vincenzo Patamia; Chiara Zagni; Letizia Crocetti; agostino cilibrizzi; Giuseppe Floresta; Antonio Rescifina
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King's College London
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The Colorimetric Detection of the Hydroxyl Radical

International Journal of Molecular Sciences
2023-02-19 | Journal article | Author
SOURCE-WORK-ID:

50ee7b59-1ba7-4068-b76c-a570b9f0a0d4

EID:

2-s2.0-85148961031

Contributors: Yandong Ran; Mohammed Moursy; Robert C. Hider; agostino cilibrizzi
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King's College London
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Ligand Growing Experiments Suggested 4-amino and 4-ureido pyridazin-3(2H)-one as Novel Scaffold for FABP4 Inhibition

Pharmaceuticals
2022-11 | Journal article | Author
SOURCE-WORK-ID:

68f41e2d-4517-4ba4-8a3c-eb14f2443f99

EID:

2-s2.0-85141789524

Contributors: Letizia Crocetti; Giuseppe Floresta; Chiara Zagni; Divya Merugu; Francesca Mazzacuva; Renan Rodrigues de Oliveira Silva; Claudia Vergelli; Maria Paola Giovannoni; agostino cilibrizzi
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King's College London
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Pyridazin-3(2H)-one as New FABP4 Inhibitors Suggested by Molecular Growing Experiments

Medical Sciences Forum
2022-11 | Journal article | Author
Contributors: Giuseppe Floresta; LETIZIA CROCETTI; Chiara Zagni; agostino cilibrizzi
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Multidisciplinary Digital Publishing Institute
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PSMA-targeted NIR probes for image-guided detection of prostate cancer

Colloids and Surfaces B: Biointerfaces
2022-10 | Journal article | Author
SOURCE-WORK-ID:

048ffc52-1e4e-41ff-9a6c-f7cf7e7dee58

EID:

2-s2.0-85135711841

Contributors: agostino cilibrizzi; Julie Tzu Wen Wang; Siham Memdouh; Antonella Iacovone; Kate McElroy; Noor Jaffar; Jennifer D. Young; Robert C. Hider; Philip Blower; KHULOUD AL-JAMAL et al.
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King's College London

An Overview of PDE4 Inhibitors in Clinical Trials

Molecules
2022-08 | Journal article | Author
SOURCE-WORK-ID:

b37aea86-39f5-4589-b428-2be9d6e36ab2

EID:

2-s2.0-85136341858

Contributors: Letizia Crocetti; Giuseppe Floresta; agostino cilibrizzi; Maria Paola Giovannoni
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King's College London
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Targeting integrin αvβ6 with gallium-68 tris (hydroxypyridinone) based PET probes

Dalton Transactions
2022-08-11 | Journal article | Author
SOURCE-WORK-ID:

638e4467-0a16-4914-a105-505c89d9101f

EID:

2-s2.0-85136967858

Contributors: Giuseppe Floresta; Siham Memdouh; Truc Thuy Pham; Michelle Ma; Philip Blower; Robert C. Hider; Vincenzo Abbate; agostino cilibrizzi
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King's College London
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Editorial

Frontiers in Chemistry
2022-08-08 | Other | Author
SOURCE-WORK-ID:

5b734814-790a-446f-9685-0cb5d92504cf

EID:

2-s2.0-85136518792

Contributors: Letizia Crocetti; Mark T. Quinn; agostino cilibrizzi; Maria Paola Giovannoni
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King's College London

Synthesis and inverse virtual screening of new bi-cyclic structures towards cancer-relevant cellular targets

STRUCTURAL CHEMISTRY
2022-06 | Journal article | Author
SOURCE-WORK-ID:

113a6c05-83a2-4d00-bc16-45e6a22a0924

EID:

2-s2.0-85124730878

Contributors: Letizia Crocetti; Giuseppe Floresta; Shabnam Nazir; Claudia Vergelli; Amrit Bhogal; Claudio Biancalani; Nicoletta Cesari; Maria Paola Giovannoni; agostino cilibrizzi
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King's College London
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Synthesis, biological evaluation, molecular modeling, and structural analysis of new pyrazole and pyrazolone derivatives as N-formyl peptide receptors agonists

Chemical Biology and Drug Design
2021-10 | Journal article | Author
SOURCE-WORK-ID:

5caea3d5-4f40-4150-8399-f7aa431f923b

EID:

2-s2.0-85114847892

Contributors: Claudia Vergelli; Andrei I. Khlebnikov; Letizia Crocetti; Gabriella Guerrini; Niccolò Cantini; Liliya N. Kirpotina; Igor A. Schepetkin; agostino cilibrizzi; Mark T. Quinn; Patrizia Rossi et al.
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King's College London

Effect of iron chelation on anti-pseudomonal activity of doxycycline

INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS
2021-09-20 | Journal article | Author
SOURCE-WORK-ID:

db834dd5-266a-4ddb-b527-7a63d48247cd

EID:

2-s2.0-85118254429

Contributors: M.E. Faure; agostino cilibrizzi; Vincenzo Abbate; K.D. Bruce; R.C. Hider
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King's College London
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Dipeptide inhibitors of the prostate specific membrane antigen (PSMA): A comparison of urea and thiourea derivatives

Bioorganic & medicinal chemistry letters
2021-06-15 | Journal article | Author
SOURCE-WORK-ID:

7e4e296e-ed68-43d3-9c0b-f3f805c14791

EID:

2-s2.0-85104585948

Contributors: Jennifer D. Young; Michelle Ma; Thomas Eykyn; Andrew Atkinson; Vincenzo Abbate; agostino cilibrizzi; Robert Hider; Philip Blower
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King's College London
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Principles that rule the calculation of dihedral angles in secondary structures

JOURNAL OF MOLECULAR STRUCTURE
2021-04-05 | Journal article | Author
SOURCE-WORK-ID:

5f355a30-a241-4a5f-9e82-5cd4c8959e33

EID:

2-s2.0-85099265142

Contributors: Michele Larocca; Giuseppe Floresta; agostino cilibrizzi
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King's College London

Pharmacokinetics of Mephedrone Enantiomers in Whole Blood after a Controlled Intranasal Administration to Healthy Human Volunteers

Pharmaceuticals
2020-12-23 | Journal article | Author
SOURCE-WORK-ID:

2a14fd69-c5e6-4722-8831-e7e34192e799

EID:

2-s2.0-85098643732

Contributors: Joanna Czerwinska; Mark C. Parkin; agostino cilibrizzi; Claire George; Andrew T. Kicman; Paul I. Dargan; Vincenzo Abbate
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King's College London
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Glutathione and the intracellular labile heme pool

Biometals
2020-12-10 | Journal article | Author
SOURCE-WORK-ID:

062cb133-ed47-426a-804a-216d80f309ee

EID:

2-s2.0-85097539826

Contributors: Rosemary O’keeffe; Gladys Latunde-Dada; Yu-lin Chen; Xiaole L. Kong; agostino cilibrizzi; Robert C. Hider
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King's College London
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Characterization of two siderophores produced by Bacillus megaterium

Biochimica et Biophysica Acta - General Subjects
2020-10 | Journal article | Author
SOURCE-WORK-ID:

f1431c7b-2a79-4c12-a883-c34910af9708

EID:

2-s2.0-85086720736

Contributors: Hataichanok Chuljerm; Manu Deeudom; Suthat Fucharoen; Francesca Mazzacuva; Robert C. Hider; Somdet Srichairatanakool; agostino cilibrizzi
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King's College London

Illuminating the Path to Target GPCR Structures and Functions

Biochemistry
2020-10-13 | Journal article | Author
SOURCE-WORK-ID:

23aa5a81-979a-4a47-8182-74a5ddd9af2b

EID:

2-s2.0-85092944583

Contributors: Christian D.T. Nielsen; Divya Dhasmana; Giuseppe Floresta; Thorsten Wohland; agostino cilibrizzi
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King's College London
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Solid-Phase Synthesis and In-Silico Analysis of Iron-Binding Catecholato Chelators

International Journal of Molecular Sciences
2020-10-12 | Journal article | Author
SOURCE-WORK-ID:

f15fb71b-5167-4855-a02f-912a35f46410

EID:

2-s2.0-85092465378

Contributors: Ranko Gacesa; Andrea Tripodi; agostino cilibrizzi; Antonella Leggio; Robert Hider; Vincenzo Abbate
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King's College London
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Human telomere double G-quadruplex recognition by berberine-bisquinolinium imaging conjugates in vitro and in cells

International Journal of Biological Macromolecules
2020-09-01 | Journal article | Author
SOURCE-WORK-ID:

d6865644-7019-4e8c-b5f5-ffee84b85e44

EID:

2-s2.0-85084992927

Contributors: Ting Cong Liao; Tian Zhu Ma; Suo Bin Chen; agostino cilibrizzi; Meng Jia Zhang; Jun Hui Li; Chun Qiong Zhou
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King's College London

Synthetic Approaches for Piperidone-Based Templates as Scaffolds to Access Chirally Enriched Donepezil Analogues

ACS Omega
2020-02-11 | Journal article | Author
SOURCE-WORK-ID:

23db93de-e28e-4b9f-b374-ffc3a16345cf

EID:

2-s2.0-85080970864

Contributors: Anna Poeschl; David M. Mountford; Robert C. Hider; agostino cilibrizzi
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King's College London
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Repurposing strategies on pyridazinone-based series by pharmacophore- and structure-driven screening

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
2020-01-01 | Journal article | Author
SOURCE-WORK-ID:

9b1b0a06-2b35-49c7-920a-0595cbaa9fd8

EID:

2-s2.0-85084276957

Contributors: Giuseppe Floresta; Letizia Crocetti; Maria Paola Giovannoni; Pierfrancesco Biagini; agostino cilibrizzi
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King's College London
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iVS analysis to evaluate the impact of scaffold diversity in the binding to cellular targets relevant in cancer

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
2019 | Journal article | Author
SOURCE-WORK-ID:

4e7f42ac-e44d-4736-9de0-53eb1847d0d4

EID:

2-s2.0-85055447506

Contributors: agostino cilibrizzi; Giuseppe Floresta; Vincenzo Abbate; Maria Paola Giovannoni
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King's College London

3D-QSAR assisted identification of FABP4 inhibitors

BIOORGANIC CHEMISTRY
2019-03-01 | Journal article | Author
SOURCE-WORK-ID:

5c760840-8050-4504-9aad-9e6d88cd7f4f

EID:

2-s2.0-85057798313

Contributors: Giuseppe Floresta; agostino cilibrizzi; Vincenzo Abbate; Ambra Spampinato; Chiara Zagni; Antonio Rescifina
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King's College London
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The role of mitochondrial labile iron in Friedreich's ataxia skin fibroblasts sensitivity to ultraviolet A

Metallomics
2019-03-01 | Journal article | Author
SOURCE-WORK-ID:

c6d385ea-b8a5-4f35-9cf6-476bdc113783

EID:

2-s2.0-85063316356

Contributors: Olivier Reelfs; Vincenzo Abbate; agostino cilibrizzi; Mark A. Pook; Robert C. Hider; Charareh Pourzand
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King's College London
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Dihedral Angle Calculations to Elucidate the Folding of Peptides through Its Main Mechanical Forces

Biochemistry
2019-02-26 | Journal article | Author
SOURCE-WORK-ID:

194238f4-b15e-40bc-b5db-e23601dc32e2

EID:

2-s2.0-85062319998

Contributors: Michele Larocca; Fabrizia Foglia; agostino cilibrizzi
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King's College London
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Mass spectrometry measurement of albumin–alpha fetoprotein ratio as an indicator of iPSC-derived hepatocyte differentiation

Methods in Molecular Biology
2019-01-01 | Book chapter | Author
SOURCE-WORK-ID:

ac6f53bd-721c-41dc-8abf-c40f73453f04

EID:

2-s2.0-85066263897

Contributors: Francesca Mazzacuva; Maëlle Lorvellec; agostino cilibrizzi; Kevin Mills; Wendy E. Heywood; Peter Clayton; Paul Gissen
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King's College London

Measurement of bile acids as a marker of the functionality of iPSC-derived hepatocytes

Methods in Molecular Biology
2019-01-01 | Book chapter | Author
SOURCE-WORK-ID:

38b1ac55-d8e9-4490-b3ee-a6e105bc90f8

EID:

2-s2.0-85066258017

Contributors: Francesca Mazzacuva; Maëlle Lorvellec; agostino cilibrizzi; Kevin Mills; Peter Clayton; Paul Gissen
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King's College London

Synthesis and iron coordination properties of schizokinen and its imide derivative

Dalton Transactions
2019-01-01 | Journal article | Author
SOURCE-WORK-ID:

79bc733f-1b4e-4d15-90f6-b77be490f286

EID:

2-s2.0-85075692395

Contributors: Hataichanok Chuljerm; Yu Lin Chen; Somdet Srichairatanakool; Robert C. Hider; agostino cilibrizzi
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King's College London
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A case of extensive protein platination: the reaction of lysozyme with a Pt(ii)–terpyridine complex

Dalton Transactions
2018 | Journal article
Contributors: Giarita Ferraro; Tiziano Marzo; Teresa Infrasca; Agostino Cilibrizzi; Ramon Vilar; Luigi Messori; Antonello Merlino
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Crossref

FABP4 inhibitors 3D-QSAR model and isosteric replacement of BMS309403 datasets

Data in Brief
2018-12-19 | Journal article | Author
SOURCE-WORK-ID:

7dc3efb9-39ac-4e3f-8d62-fedca862f97f

EID:

2-s2.0-85059158868

Contributors: Giuseppe Floresta; agostino cilibrizzi; Vincenzo Abbate; Ambra Spampinato; Chiara Zagni; Antonio Rescifina
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King's College London
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Preparation, structure, cytotoxicity and mechanism of action of ferritin-Pt(II) terpyridine compound nanocomposites

Nanomedicine
2018-12-03 | Journal article | Author
SOURCE-WORK-ID:

e22660fb-5f29-47b6-9f7d-f0380d02293b

EID:

2-s2.0-85058086378

Contributors: Giarita Ferraro; Andrea Pica; Ganna Petruk; Francesca Pane; Angela Amoresano; agostino cilibrizzi; Ramon Vilar; Daria Maria Monti; Antonello Merlino
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King's College London

Hydroxypyridinone Journey into Metal Chelation

Chemical Reviews
2018-08-22 | Journal article
Contributors: Agostino Cilibrizzi; Vincenzo Abbate; Yu-Lin Chen; Yongmin Ma; Tao Zhou; Robert C. Hider
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Crossref

Hydroxypyridinone Journey into Metal Chelation

Chemical Reviews
2018-07-23 | Journal article | Author
SOURCE-WORK-ID:

3206f39c-1249-4536-95ea-d5434eebd8ce

EID:

2-s2.0-85052104317

Contributors: agostino cilibrizzi; Vincenzo Abbate; Yu-Lin Chen; Yongmin Ma; Tao Zhou; Robert Charles Hider
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King's College London

Correspondence: Compound 17b and formyl peptide receptor biased agonism in relation to cardioprotective effects in ischaemia-reperfusion injury

Nature Communications
2018-02-07 | Journal article | Author
SOURCE-WORK-ID:

8a7c15be-e9f5-4b75-a933-50cf9d672b24

EID:

2-s2.0-85041862212

Contributors: agostino cilibrizzi
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King's College London
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Small-molecule optical probes for cell imaging of protein sulfenylation and their application to monitor cisplatin induced protein oxidation

Sensors And Actuators B-Chemical
2017-09 | Journal article | Author
SOURCE-WORK-ID:

5e2d935e-9aa4-4f08-b5ba-6101fc62f9b9

EID:

2-s2.0-85017311622

Contributors: agostino cilibrizzi; Mattia Terenghi; Marina Fedorova; Rudiger Woscholski; David Klug; Ramon Vilar
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King's College London

Analytical characterization of three cathinone derivatives, 4-MPD, 4 F-PHP and bk-EPDP, purchased as bulk powder from online vendors

Drug Testing And Analysis
2017-07-18 | Journal article | Author
SOURCE-WORK-ID:

c330ebc7-5c4e-434a-bf06-795fcbd68c09

EID:

2-s2.0-85025110197

Contributors: Orapan Apirakkan; Anca Frinculescu; Trevor Shine; Mark C. Parkin; agostino cilibrizzi; Nunzianda Frascione; Vincenzo Abbate
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King's College London

A tri-functional vanadium(IV) complex to detect cysteine oxidation

DALTON TRANSACTIONS (2003)
2017-05-08 | Journal article | Author
SOURCE-WORK-ID:

9d970b35-0798-4262-b3b4-926c889bf654

EID:

2-s2.0-85021716374

Contributors: agostino cilibrizzi; Marina Fedorova; Juliet Collins; Robin J. Leatherbarrow; Rudiger Woscholski; Ramon Vilar
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King's College London
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Synthesis and analytical characterization of new thiazol-2-(3H)-ones as human neutrophil elastase (HNE) inhibitors

Chemistry Central Journal
2017-01-01 | Journal article | Author
SOURCE-WORK-ID:

7bb9000b-0a87-469f-9720-da4aeeea2f13

EID:

2-s2.0-85047203044

Contributors: Letizia Crocetti; Gianluca Bartolucci; agostino cilibrizzi; Maria Paola Giovannoni; Gabriella Guerrini; Antonella Iacovone; Marta Menicatti; Igor A. Schepetkin; Andrei I. Khlebnikov; Mark T. Quinn et al.
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King's College London
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Peer review (1 review for 1 publication/grant)

Review activity for European journal of inorganic chemistry. (1)