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Works (10)

Novel HDAC6 Inhibitors Increase Tubulin Acetylation and Rescue Axonal Transport of Mitochondria in a Model of Charcot-Marie-Tooth Type 2F

ACS Chemical Neuroscience
2020 | Journal article
EID:

2-s2.0-85078440885

Part of ISBN:

19487193

Contributors: Adalbert, R.; Kaieda, A.; Antoniou, C.; Loreto, A.; Yang, X.; Gilley, J.; Hoshino, T.; Uga, K.; Makhija, M.T.; Coleman, M.P.
Source: Self-asserted source
Akira Kaieda via Scopus - Elsevier

Identification of 2,6-Disubstituted 3 H-Imidazo[4,5- b]pyridines as Therapeutic Agents for Dysferlinopathies through Phenotypic Screening on Patient-Derived Induced Pluripotent Stem Cells

Journal of Medicinal Chemistry
2019 | Journal article
EID:

2-s2.0-85073264096

Part of ISBN:

15204804 00222623

Contributors: Takada, H.; Kaieda, A.; Tawada, M.; Nagino, T.; Sasa, K.; Oikawa, T.; Oki, A.; Sameshima, T.; Miyamoto, K.; Miyamoto, M. et al.
Source: Self-asserted source
Akira Kaieda via Scopus - Elsevier

Structure-Based Design, Synthesis, and Biological Evaluation of Imidazo[4,5-b]pyridin-2-one-Based p38 MAP Kinase Inhibitors: Part 1

ChemMedChem
2019 | Journal article
EID:

2-s2.0-85064710591

Part of ISBN:

18607187 18607179

Contributors: Kaieda, A.; Takahashi, M.; Fukuda, H.; Okamoto, R.; Morimoto, S.; Gotoh, M.; Miyazaki, T.; Hori, Y.; Unno, S.; Kawamoto, T. et al.
Source: Self-asserted source
Akira Kaieda via Scopus - Elsevier

Structure-Based Design, Synthesis, and Biological Evaluation of Imidazo[4,5-b]Pyridin-2-one-Based p38 MAP Kinase Inhibitors: Part 2

ChemMedChem
2019 | Journal article
EID:

2-s2.0-85074871445

Part of ISBN:

18607187 18607179

Contributors: Kaieda, A.; Takahashi, M.; Fukuda, H.; Okamoto, R.; Morimoto, S.; Gotoh, M.; Miyazaki, T.; Hori, Y.; Unno, S.; Kawamoto, T. et al.
Source: Self-asserted source
Akira Kaieda via Scopus - Elsevier

Structure-based design, synthesis, and biological evaluation of imidazo[1,2-b]pyridazine-based p38 MAP kinase inhibitors

Bioorganic and Medicinal Chemistry
2018 | Journal article
EID:

2-s2.0-85039557829

Part of ISBN:

14643391 09680896

Contributors: Kaieda, A.; Takahashi, M.; Takai, T.; Goto, M.; Miyazaki, T.; Hori, Y.; Unno, S.; Kawamoto, T.; Tanaka, T.; Itono, S. et al.
Source: Self-asserted source
Akira Kaieda via Scopus - Elsevier

Discovery of novel, highly potent, and selective matrix metalloproteinase (MMP)-13 inhibitors with a 1,2,4-triazol-3-yl moiety as a zinc binding group using a structure-based design approach

Journal of Medicinal Chemistry
2017 | Journal article
EID:

2-s2.0-85010782797

Part of ISBN:

15204804 00222623

Contributors: Nara, H.; Kaieda, A.; Sato, K.; Naito, T.; Mototani, H.; Oki, H.; Yamamoto, Y.; Kuno, H.; Santou, T.; Kanzaki, N. et al.
Source: Self-asserted source
Akira Kaieda via Scopus - Elsevier

Design, synthesis, and biological activity of novel, potent, and highly selective fused pyrimidine-2-carboxamide-4-one-based matrix metalloproteinase (MMP)-13 zinc-binding inhibitors

Bioorganic and Medicinal Chemistry
2016 | Journal article
EID:

2-s2.0-84999025978

Part of ISBN:

14643391 09680896

Contributors: Nara, H.; Sato, K.; Kaieda, A.; Oki, H.; Kuno, H.; Santou, T.; Kanzaki, N.; Terauchi, J.; Uchikawa, O.; Kori, M.
Source: Self-asserted source
Akira Kaieda via Scopus - Elsevier

New utilizations of optically active homoallylamines: Highly stereoselective synthesis of cyclic guanidine and thiourea

Heterocycles
2005 | Journal article
EID:

2-s2.0-33646868802

Part of ISBN:

03855414

Contributors: Yanada, R.; Kaieda, A.; Yanada, K.; Takemoto, Y.
Source: Self-asserted source
Akira Kaieda via Scopus - Elsevier

Aluminum-controlled reactivity and diastereoselectivity toward radical reactions of optically active aldimines with metallic samarium

Journal of Organic Chemistry
2001 | Journal article
EID:

2-s2.0-0035936779

Part of ISBN:

00223263

Contributors: Yanada, R.; Okaniwa, M.; Kaieda, A.; Ibuka, T.; Takemoto, Y.
Source: Self-asserted source
Akira Kaieda via Scopus - Elsevier

Diastereoselective Barbier-type and palladium-mediated allylation of optically active aldimine with allylindium reagents

Journal of Organic Chemistry
2001 | Journal article
EID:

2-s2.0-0035798191

Part of ISBN:

00223263

Contributors: Yanada, R.; Kaieda, A.; Takemoto, Y.
Source: Self-asserted source
Akira Kaieda via Scopus - Elsevier