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Scopus Author ID: 57184348500

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Leiden University: Leiden, NL

Employment
Source: Self-asserted source
Daan van der Es

Works (26)

Stereochemical optimization of N,2-substituted cycloalkylamines as norepinephrine reuptake inhibitors

RSC Medicinal Chemistry
2024-09-12 | Journal article
DOI: 10.1039/d4md00521j
OTHER-ID:

7ae66f2f-0600-476a-8902-b39660e67df0
Contributors: Dilweg; M.A.; Mocking,T.A.M.; Maragkoudakis; P.; Westen; G.J.P. van; Heitman; L.H.; IJzerman; A.P.; Jespers; W.; Es; D. van der
Source: check_circle
Leiden University

Inducing Receptor Degradation as a Novel Approach to Target CC Chemokine Receptor 2 (CCR2)

International Journal of Molecular Sciences
2024-08 | Journal article | Author
DOI: 10.3390/ijms25168984
Contributors: Natalia V. Ortiz Zacarías; Sascha Röth; Jeremy D. Broekhuis; Daan van der Es; Kevin Moreau; Laura Heitman
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Multidisciplinary Digital Publishing Institute
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Preferred source (of 2)‎

Labeling of CC chemokine receptor 2 with a versatile intracellular allosteric probe

ACS Chemical Biology
2024-08-26 | Journal article
DOI: 10.1021/acschembio.4c00439
OTHER-ID:

b5a4e0cb-b6d3-4b0c-bede-96f2f2ec15ed
Contributors: Hollander; L.S. den; Beerkens; B.L.H.; Dekkers; S.; Veldhoven; J.P.D. van; Ortiz Zacarías; N.V.; Horst; C. van der; Sieders; E.G.; Valk; B. de; Wang; J.; IJzerman et al.
Source: check_circle
Leiden University

N-Acyl-N-alkyl sulfonamide probes for ligand-directed covalent labeling of GPCRs

ACS Chemical Biology
2024-06-26 | Journal article
DOI: 10.1021/acschembio.4c00210
OTHER-ID:

56e0155e-0a07-4590-abf6-7612f5ca5461
Contributors: Beerkens; B.L.H.; Andrianopoulou; V.; Wang; X.; Liu; R.; Westen; G.J. P. van; Jespers; W.; IJzerman; A.P.; Heitman; L.H.; Es; D. van der
Source: check_circle
Leiden University

Exploring novel dilazep derivatives as hENT1 inhibitors and potentially covalent molecular tools

Purinergic Signalling
2024-06-15 | Journal article
DOI: 10.1007/s11302-024-10026-x
OTHER-ID:

c04e5daf-2b53-4c95-bf2b-7340dbad4768
Contributors: Dilweg; M.A.; Gorostiola González; M.; Ruiter; M.D. de; Meijboom; N.J.; Veldhoven; J.P.D. van; Liu; R.; Jespers; W.; Westen; G.J.P. van; Heitman; L.H.; IJzerman et al.
Source: check_circle
Leiden University

Development of an affinity-based probe to profile endogenous human adenosine A3 receptor expression

Journal of Medicinal Chemistry
2023-08-02 | Journal article
DOI: 10.1021/acs.jmedchem.3c00854
OTHER-ID:

1b2a7dc6-5e8a-416c-ab0d-541574a0e961
Contributors: Beerkens; B.L.H.; Snijders; I.M.; Snoeck; J.; Liu; R.; Tool; A.T.J.; Le Dévédec; S.E.; Jespers; W.; Kuijpers; T.W.; Westen; G.J.P. van; Heitman et al.
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Leiden University

A chemical biological approach to study G protein-coupled receptors

ACS Chemical Biology
2022-10-24 | Journal article
DOI: 10.1021/acschembio.2c00589
OTHER-ID:

7b596c01-045b-4c6c-bf98-42dfd7909f78

WOSUID:

000877139300001
Contributors: Beerkens; B.L.H.; Koc; C.; Liu; R.; Florea; B.I.; Le Dévédec; S.E.; Heitman; L.H.; IJzerman; A.P.; Es; D. van der
Source: check_circle
Leiden University

Crystal Structure and Subsequent Ligand Design of a Nonriboside Partial Agonist Bound to the Adenosine A<sub>2A</sub>Receptor

Journal of Medicinal Chemistry
2021 | Journal article
DOI: 10.1021/acs.jmedchem.0c01856
EID:

2-s2.0-85104048175

Part of ISSN: 15204804 00222623
Contributors: Amelia, T.; Van Veldhoven, J.P.D.; Falsini, M.; Liu, R.; Heitman, L.H.; Van Westen, G.J.P.; Segala, E.; Verdon, G.; Cheng, R.K.Y.; Cooke, R.M. et al.
Source: Self-asserted source
Daan van der Es via Scopus - Elsevier
grade
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Design and Characterization of an Intracellular Covalent Ligand for CC Chemokine Receptor 2

Journal of Medicinal Chemistry
2021 | Journal article
DOI: 10.1021/acs.jmedchem.0c01137
EID:

2-s2.0-85102906861

Part of ISSN: 15204804 00222623
Contributors: Ortiz Zacarías, N.V.; Chahal, K.K.; Šimková, T.; Van Der Horst, C.; Zheng, Y.; Inoue, A.; Theunissen, E.; Mallee, L.; Van Der Es, D.; Louvel, J. et al.
Source: Self-asserted source
Daan van der Es via Scopus - Elsevier
grade
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Epitope Recognition of a Monoclonal Antibody Raised against a Synthetic Glycerol Phosphate Based Teichoic Acid

ACS Chemical Biology
2021 | Journal article
DOI: 10.1021/acschembio.1c00422
EID:

2-s2.0-85111235949

Part of ISSN: 15548937 15548929
Contributors: Berni, F.; Kalfopoulou, E.; Gimeno Cardells, A.M.; Carboni, F.; Van Der Es, D.; Romero-Saavedra, F.; Laverde, D.; Miklic, K.; Malic, S.; Rovis, T.L. et al.
Source: Self-asserted source
Daan van der Es via Scopus - Elsevier
grade
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Generation of glucosylated: Sn -1-glycerolphosphate teichoic acids: Glycerol stereochemistry affects synthesis and antibody interaction

RSC Chemical Biology
2021 | Journal article
DOI: 10.1039/d0cb00206b
EID:

2-s2.0-85106171016

Part of ISSN: 26330679
Contributors: Berni, F.; Wang, L.; Kalfopoulou, E.; Nguyen, D.L.; Van Der Es, D.; Huebner, J.; Overkleeft, H.S.; Hokke, C.H.; Van Der Marel, G.A.; Van Diepen, A. et al.
Source: Self-asserted source
Daan van der Es via Scopus - Elsevier

Molecular probes for the human adenosine receptors

Purinergic Signalling
2021 | Journal article
DOI: 10.1007/s11302-020-09753-8
EID:

2-s2.0-85097508526

Part of ISSN: 15739546 15739538
Contributors: Yang, X.; Heitman, L.H.; IJzerman, A.P.; van der Es, D.
Source: Self-asserted source
Daan van der Es via Scopus - Elsevier
grade
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Profiling acidic metabolites by capillary electrophoresis‐mass spectrometry in low numbers of mammalian cells using a novel chemical derivatization approach

Analytical Science Advances
2021-12-14 | Journal article
DOI: 10.1002/ansa.202100054
OTHER-ID:

1dbfd4f7-0e6e-43ed-8ee7-3bd20813709a
Contributors: Mever; M. van; Willacey; C.C.W.; Zhang; W.; Drouin; N.F.P.; Christina; A.E.; Lindenburg; P.W.; Veldhoven; J.P. D. van; Es; D. van der; Harms; A.C.; Hankemeier et al.
Source: check_circle
Leiden University

A stabilized glycomimetic conjugate vaccine inducing protective antibodies against Neisseria meningitidis serogroup A

Nature Communications
2020 | Journal article
DOI: 10.1038/s41467-020-18279-x
EID:

2-s2.0-85090321242

Part of ISSN: 20411723
Contributors: Enotarpi, J.; Tontini, M.; Balocchi, C.; van der Es, D.; Auberger, L.; Balducci, E.; Carboni, F.; Proietti, D.; Casini, D.; Filippov, D.V. et al.
Source: Self-asserted source
Daan van der Es via Scopus - Elsevier
grade
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Design and pharmacological profile of a novel covalent partial agonist for the adenosine A<sub>1</sub> receptor

Biochemical Pharmacology
2020 | Journal article
DOI: 10.1016/j.bcp.2020.114144
EID:

2-s2.0-85088027705

Part of ISSN: 18732968 00062952
Contributors: Yang, X.; Dilweg, M.A.; Osemwengie, D.; Burggraaff, L.; van der Es, D.; Heitman, L.H.; IJzerman, A.P.
Source: Self-asserted source
Daan van der Es via Scopus - Elsevier
grade
Preferred source (of 2)‎

Design, Synthesis and Pharmacological Profiles of LUF7746, a Novel Covalent Partial Agonist for the Adenosine A1 Receptor

ChemRxiv
2020 | Other
DOI: 10.26434/chemrxiv.11903286.v1
EID:

2-s2.0-85095658419

Part of ISSN: 25732293
Contributors: Yang, X.; Dilweg, M.A.; Osemwengie, D.; Burggraaff, L.; van der Es, D.; Heitman, L.H.; IJzerman, A.P.
Source: Self-asserted source
Daan van der Es via Scopus - Elsevier

Development of Covalent Ligands for G Protein-Coupled Receptors: A Case for the Human Adenosine A<sub>3</sub> Receptor

Journal of Medicinal Chemistry
2019 | Journal article
DOI: 10.1021/acs.jmedchem.8b02026
EID:

2-s2.0-85064126878

Part of ISSN: 15204804 00222623
Contributors: Yang, X.; Van Veldhoven, J.P.D.; Offringa, J.; Kuiper, B.J.; Lenselink, E.B.; Heitman, L.H.; Van Der Es, D.; Ijzerman, A.P.
Source: Self-asserted source
Daan van der Es via Scopus - Elsevier
grade
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LC–MS/MS analysis of the central energy and carbon metabolites in biological samples following derivatization by dimethylaminophenacyl bromide

Journal of Chromatography A
2019 | Journal article
DOI: 10.1016/j.chroma.2019.460413
EID:

2-s2.0-85070108865

Part of ISSN: 18733778 00219673
Contributors: Willacey, C.C.W.; Naaktgeboren, M.; Lucumi Moreno, E.; Wegrzyn, A.B.; van der Es, D.; Karu, N.; Fleming, R.M.T.; Harms, A.C.; Hankemeier, T.
Source: Self-asserted source
Daan van der Es via Scopus - Elsevier
grade
Preferred source (of 2)‎

An Affinity-Based Probe for the Human Adenosine A<sub>2A</sub> Receptor

Journal of Medicinal Chemistry
2018 | Journal article
DOI: 10.1021/acs.jmedchem.8b00860
EID:

2-s2.0-85052326052

Part of ISSN: 15204804 00222623
Contributors: Yang, X.; Michiels, T.J.M.; De Jong, C.; Soethoudt, M.; Dekker, N.; Gordon, E.; Van Der Stelt, M.; Heitman, L.H.; Van Der Es, D.; Ijzerman, A.P.
Source: Self-asserted source
Daan van der Es via Scopus - Elsevier
grade
Preferred source (of 2)‎

Streamlined Synthesis and Evaluation of Teichoic Acid Fragments

Chemistry - A European Journal
2018-02 | Journal article
DOI: 10.1002/chem.201800153
Part of ISSN: 0947-6539
Contributors: Daan van der Es; Francesca Berni; Wouter F. J. Hogendorf; Nico Meeuwenoord; Diana Laverde; Angela van Diepen; Herman S. Overkleeft; Dmitri V. Filippov; Cornelis H. Hokke; Johannes Huebner et al.
Source: Self-asserted source
Daan van der Es via Crossref Metadata Search
grade
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Teichoic acids: synthesis and applications

Chemical Society Reviews
2017 | Journal article
DOI: 10.1039/c6cs00270f
Part of ISSN: 0306-0012
Contributors: Daan van der Es; Wouter F. J. Hogendorf; Herman S. Overkleeft; Gijsbert A. van der Marel; Jeroen D. C. Codée
Source: Self-asserted source
Daan van der Es via Crossref Metadata Search
grade
Preferred source (of 3)‎

Kinetics of human cannabinoid 1 (CB1) receptor antagonists: Structure-kinetics relationships (SKR) and implications for insurmountable antagonism

Biochemical Pharmacology
2017-11 | Journal article
DOI: 10.1016/j.bcp.2017.10.014
Part of ISSN: 0006-2952
Contributors: Lizi Xia; Henk de Vries; Xue Yang; Eelke B. Lenselink; Athina Kyrizaki; Francis Barth; Julien Louvel; Matthias K. Dreyer; Daan van der Es; Adriaan P. IJzerman et al.
Source: Self-asserted source
Daan van der Es via Crossref Metadata Search
grade
Preferred source (of 3)‎

Synthesis of phosphodiester-containing bacterial cell wall components : teichoic acids, capsular polysaccharides and phosphatidyl glycerol analogues

2016-10-04 | Dissertation or Thesis
OTHER-ID:

26d788f9-423c-4d20-8682-e688ca21ee41
Contributors: Es; D. van der
Source: check_circle
Leiden University

Synthesis of E. faecium wall teichoic acid fragments.

2016-09 | Journal article
DOI: 10.1016/j.bmc.2016.03.019
PMID: 26993744
Contributors: van der Es D; Groenia NA; Laverde D; Overkleeft HS; Huebner J; van der Marel GA; Codée JD
Source: Self-asserted source
Daan van der Es via Europe PubMed Central
grade
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β-Rhamnosides from 6-thio mannosides

Chem. Commun.
2012 | Journal article
DOI: 10.1039/c2cc17623h
Contributors: Alphert E. Christina; Daan van der Es; Jasper Dinkelaar; Hermen S. Overkleeft; Gijsbert A. van der Marel; Jeroen D. C. Codée
Source: Self-asserted source
Daan van der Es via Crossref Metadata Search
grade
Preferred source (of 2)‎

Development of subtype-selective covalent ligands for the adenosine A2B receptor by tuning the reactive group

RSC Medicinal Chemistry
Journal article
DOI: 10.1039/D2MD00132B
OTHER-ID:

1765d86e-3796-48fa-a922-1acbe9484ad3
Contributors: Beerkens; B.L.H.; Wang; X.; Avgeropoulou; M.; Adistia; L.N.; Veldhoven; J.P.D. van; Jespers; W.; Liu; R.; Heitman; L.H.; IJzerman; A.P.; Es et al.
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Leiden University
grade
Preferred source (of 2)‎

Peer review (7 reviews for 7 publications/grants)

Review activity for ACS medicinal chemistry letters. (1)
Review activity for ACS omega. (1)
Review activity for Analytical chemistry. (1)
Review activity for Communications chemistry. (1)
Review activity for Journal of medicinal chemistry. (1)
Review activity for Nature communications (1)
Review activity for The journal of physical chemistry. (1)
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