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Employment (2)

Associazione OASI Maria SS: Troina, Sicilia, IT

2018-03-02 to present | Associate Researcher (Department of Laboratories)
Employment
Source: Self-asserted source
Santina Chiechio

Università degli Studi di Catania: Catania, Sicilia, IT

2007-10-01 to present | Professore Associato (Dipartimento di Scienze del Farmaco)
Employment
Source: Self-asserted source
Santina Chiechio

Works (50 of 68)

Items per page:
Page 1 of 2

Memantine and amantadine KLVFF peptide conjugates: Synthesis, structure determination, amyloid-β interaction and effects on recognition memory in mice

European Journal of Pharmacology
2025-03 | Journal article
Contributors: Eleonora Bocchieri; Stefania Zimbone; Maria Laura Giuffrida; Giuseppe Di Natale; Giuseppina Sabatino; Graziella Vecchio; Giuseppe Pappalardo; Santina Chiechio
Source: check_circle
Crossref

Exploring the Role of Hsp60 in Alzheimer’s Disease and Type 2 Diabetes: Suggestion for Common Drug Targeting

International Journal of Molecular Sciences
2023 | Journal article
EID:

2-s2.0-85167881675

Part of ISSN: 14220067 16616596
Contributors: Zimbone, S.; Di Rosa, M.C.; Chiechio, S.; Giuffrida, M.L.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier
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Increased Heat Pain Tolerance but Hyperalgesia to Tonic Inflammatory Pain in the CRND8 Mouse Model of Alzheimer's Disease

Journal of Alzheimer's Disease
2023 | Journal article
EID:

2-s2.0-85175496145

Part of ISSN: 18758908 13872877
Contributors: Merlo, S.; Costa, L.; Chiechio, S.; Busceti, C.L.; Ciranna, L.; Santangelo, R.; Sortino, M.A.; Fornai, F.; Nicoletti, F.; Copani, A.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Mu and Delta Opioid Receptor Targeting Reduces Connexin 43-Based Heterocellular Coupling during Neuropathic Pain

International Journal of Molecular Sciences
2022 | Journal article
EID:

2-s2.0-85130821297

Part of ISSN: 14220067 16616596
Contributors: Vicario, N.; Denaro, S.; Turnaturi, R.; Longhitano, L.; Spitale, F.M.; Spoto, S.; Marrazzo, A.; Zappalà, A.; Tibullo, D.; Volti, G.L. et al.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier
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Novel N-normetazocine Derivatives with Opioid Agonist/Sigma-1 Receptor Antagonist Profile as Potential Analgesics in Inflammatory Pain

Molecules
2022 | Journal article
EID:

2-s2.0-85137483599

Part of ISSN: 14203049
Contributors: Turnaturi, R.; Chiechio, S.; Pasquinucci, L.; Spoto, S.; Costanzo, G.; Dichiara, M.; Piana, S.; Grasso, M.; Amata, E.; Marrazzo, A. et al.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier
grade
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A standardized extract prepared from red orange and lemon wastes blocks high-fat diet-induced hyperglycemia and hyperlipidemia in mice

Molecules
2021 | Journal article
EID:

2-s2.0-85111159322

Part of ISSN: 14203049
Contributors: Chiechio, S.; Zammataro, M.; Barresi, M.; Amenta, M.; Ballistreri, G.; Fabroni, S.; Rapisarda, P.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier
grade
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The Multimodal MOPr/DOPr Agonist LP2 Reduces Allodynia in Chronic Constriction Injured Rats by Rescue of TGF-β1 Signalling

Frontiers in Pharmacology
2021 | Journal article
EID:

2-s2.0-85117467487

Part of ISSN: 16639812
Contributors: Fidilio, A.; Grasso, M.; Turnaturi, R.; Caruso, G.; Spitale, F.M.; Vicario, N.; Parenti, R.; Spoto, S.; Musso, N.; Marrazzo, A. et al.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Exploiting the power of stereochemistry in drug action: 3-[(2S,6S,11S)-8-Hydroxy-6,11-dimethyl-1,4,5,6-tetrahydro-2,6-methano-3-benzazocin-3(2H)-yl]-N-phenylpropanamide as potent sigma-1 receptor antagonist

ACS Chemical Neuroscience
2020 | Journal article
EID:

2-s2.0-85082779746

Part of ISBN:

19487193

Contributors: Turnaturi, R.; Pasquinucci, L.; Chiechio, S.; Grasso, M.; Marrazzo, A.; Amata, E.; Dichiara, M.; Prezzavento, O.; Parenti, C.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Intercellular communication and ion channels in neuropathic pain chronicization

Inflammation Research
2020 | Journal article
EID:

2-s2.0-85086332695

Part of ISBN:

1420908X 10233830

Contributors: Vicario, N.; Turnaturi, R.; Spitale, F.M.; Torrisi, F.; Zappalà, A.; Gulino, R.; Pasquinucci, L.; Chiechio, S.; Parenti, C.; Parenti, R.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Lipid Nanoparticle Inclusion Prevents Capsaicin-Induced TRPV1 Defunctionalization

Pharmaceutics
2020-04-10 | Journal article
Contributors: Carmelo Puglia; Debora Santonocito; Angela Bonaccorso; Teresa Musumeci; Barbara Ruozi; Rosario Pignatello; Claudia Carbone; Carmela Parenti; Santina Chiechio
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Crossref
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(2S)-N-2-methoxy-2-phenylethyl-6,7-benzomorphan compound (2S-LP2): Discovery of a biased mu/delta opioid receptor agonist

European Journal of Medicinal Chemistry
2019 | Journal article
EID:

2-s2.0-85061983229

Contributors: Pasquinucci, L.; Turnaturi, R.; Calò, G.; Pappalardo, F.; Ferrari, F.; Russo, G.; Arena, E.; Montenegro, L.; Chiechio, S.; Prezzavento, O. et al.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Progress in the development of more effective and safer analgesics for pain management

European Journal of Medicinal Chemistry
2019 | Journal article
EID:

2-s2.0-85072333329

Contributors: Turnaturi, R.; Chiechio, S.; Salerno, L.; Rescifina, A.; Pittalà, V.; Cantarella, G.; Tomarchio, E.; Parenti, C.; Pasquinucci, L.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Simultaneous Activation of Mu and Delta Opioid Receptors Reduces Allodynia and Astrocytic Connexin 43 in an Animal Model of Neuropathic Pain

Molecular Neurobiology
2019 | Journal article
EID:

2-s2.0-85064921554

Contributors: Vicario, N.; Pasquinucci, L.; Spitale, F.M.; Chiechio, S.; Turnaturi, R.; Caraci, F.; Tibullo, D.; Avola, R.; Gulino, R.; Parenti, R. et al.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Simultaneous targeting of MOR/DOR: A useful strategy for inflammatory pain modulation

European Journal of Pharmacology
2019 | Journal article
EID:

2-s2.0-85060755463

Contributors: Pasquinucci, L.; Turnaturi, R.; Montenegro, L.; Caraci, F.; Chiechio, S.; Parenti, C.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Synthesis, in vitro and in vivo characterization of new benzoxazole and benzothiazole-based sigma receptor ligands

European Journal of Medicinal Chemistry
2019 | Journal article
EID:

2-s2.0-85064736232

Contributors: Romeo, G.; Prezzavento, O.; Intagliata, S.; Pittalà, V.; Modica, M.N.; Marrazzo, A.; Turnaturi, R.; Parenti, C.; Chiechio, S.; Arena, E. et al.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Preclinical evidence of enhanced analgesic activity of duloxetine complexed with succinyl-β-cyclodextrin: A comparative study with cyclodextrin complexes

International Journal of Pharmaceutics
2019-07 | Journal article
Contributors: Mimimorena Seggio; Annalinda Contino; Giuseppe Maccarrone; Carmela Parenti; Sara Merlo; Giuseppe Pappalardo; Alessandro Giuffrida; Santina Chiechio
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Crossref
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L-acetylcarnitine: A mechanistically distinctive and potentially rapid-acting antidepressant drug

International Journal of Molecular Sciences
2018 | Journal article
EID:

2-s2.0-85039701502

Contributors: Chiechio, S.; Canonico, P.L.; Grilli, M.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier
grade
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Chronic treatment with fluoxetine induces sex-dependent analgesic effects and modulates HDAC2 and mGlu2 expression in female mice

Frontiers in Pharmacology
2017 | Journal article
EID:

2-s2.0-85031797543

Contributors: Zammataro, M.; Merlo, S.; Barresi, M.; Parenti, C.; Hu, H.; Sortino, M.A.; Chiechio, S.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Rosemary Essential Oil-Loaded Lipid Nanoparticles: In Vivo Topical Activity from Gel Vehicles

Pharmaceutics
2017-10 | Journal article
Source: check_circle
Multidisciplinary Digital Publishing Institute
grade
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Modulation of Chronic Pain by Metabotropic Glutamate Receptors

Advances in Pharmacology
2016 | Book chapter
EID:

2-s2.0-84954286987

Part of ISSN: 15578925 10543589
Contributors: Chiechio, S.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier
grade
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Repeated activation of delta opioid receptors counteracts nerve injury-induced TNF-α up-regulation in the sciatic nerve of rats with neuropathic pain: A possible correlation with delta opioid receptors-mediated antiallodinic effect

Molecular Pain
2016 | Journal article
EID:

2-s2.0-84995562578

Contributors: Vicario, N.; Parenti, R.; Aricò, G.; Turnaturi, R.; Scoto, G.M.; Chiechio, S.; Parenti, C.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Involvement of the heme-oxygenase pathway in the antiallodynic and antihyperalgesic activity of Harpagophytum procumbens in rats

Molecules
2015 | Journal article
EID:

2-s2.0-84947982588

Contributors: Parenti, C.; Aricò, G.; Chiechio, S.; Di Benedetto, G.; Parenti, R.; Scoto, G.M.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier
grade
Preferred source (of 2)‎

Monomeric ß-amyloid interacts with type-1 insulin-like growth factor receptors to provide energy supply to neurons

Frontiers in Cellular Neuroscience
2015 | Journal article
EID:

2-s2.0-84940192193

Contributors: Giuffrida, M.L.; Tomasello, M.F.; Pandini, G.; Caraci, F.; Battaglia, G.; Busceti, C.; Di Pietro, P.; Pappalardo, G.; Attanasio, F.; Chiechio, S. et al.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

HDAC and HAT inhibitors differently affect analgesia mediated by group II metabotropic glutamate receptors

Molecular Pain
2014 | Journal article
EID:

2-s2.0-84944037585

Contributors: Zammataro, M.; Sortino, M.A.; Parenti, C.; Gereau, R.W.; Chiechio, S.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Acetyl-L-carnitine: From a biological curiosity to a drug for the peripheral nervous system and beyond

Expert Review of Neurotherapeutics
2013 | Journal article
EID:

2-s2.0-84882785708

Contributors: Onofrj, M.; Ciccocioppo, F.; Varanese, S.; Di Muzio, A.; Calvani, M.; Chiechio, S.; Osio, M.; Thomas, A.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Beta-Amyloid monomer and insulin/IGF-1 signaling in Alzheimer's disease

Molecular Neurobiology
2012 | Journal article
EID:

2-s2.0-84880726942

Contributors: Giuffrida, M.L.; Tomasello, F.; Caraci, F.; Chiechio, S.; Nicoletti, F.; Copani, A.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Curcumin loaded NLC induces histone hypoacetylation in the CNS after intraperitoneal administration in mice

European Journal of Pharmaceutics and Biopharmaceutics
2012 | Journal article
EID:

2-s2.0-84861634891

Contributors: Puglia, C.; Frasca, G.; Musumeci, T.; Rizza, L.; Puglisi, G.; Bonina, F.; Chiechio, S.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Metabotropic glutamate receptors and the control of chronic pain

Current Opinion in Pharmacology
2012 | Journal article
EID:

2-s2.0-84857238962

Contributors: Chiechio, S.; Nicoletti, F.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Development, characterization, and in vitro and in vivo evaluation of benzocaine- and lidocaine-loaded nanostructrured lipid carriers

Journal of Pharmaceutical Sciences
2011 | Journal article
EID:

2-s2.0-79952234981

Contributors: Puglia, C.; Sarpietro, M.G.; Bonina, F.; Castelli, F.; Zammataro, M.; Chiechio, S.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Hyperalgesic activity of kisspeptin in mice

Molecular Pain
2011 | Journal article
EID:

2-s2.0-81555230341

Contributors: Spampinato, S.; Trabucco, A.; Biasiotta, A.; Biagioni, F.; Cruccu, G.; Copani, A.; Colledge, W.H.; Sortino, M.A.; Nicoletti, F.; Chiechio, S.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

MGlu2 metabotropic glutamate receptors restrain inflammatory pain and mediate the analgesic activity of dual mGlu2/mGlu3 receptor agonists

Molecular Pain
2011 | Journal article
EID:

2-s2.0-78651367251

Contributors: Zammataro, M.; Chiechio, S.; Montana, M.C.; Traficante, A.; Copani, A.; Nicoletti, F.; Gereau IV, R.W.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

The mGluR2 Activation Machinery and Treatment of Chronic Pain: from L-acetyl Carnitine to N-Acetyl Cysteine

Current Neuropharmacology
2011 | Journal article
Contributors: Notartomaso, Serena; Bernabucci, Matteo; Zappulla, Cristina; Fazio, Francesco; Cannella, Milena; Motolese, Marta; Zammataro, M.; Trabucco, A.; Copani, Agata; Gradini, Roberto et al.
Source: check_circle
Web of Science Researcher Profile Sync

Transcriptional regulation of type-2 metabotropic glutamate receptors: An epigenetic path to novel treatments for chronic pain

Trends in Pharmacological Sciences
2010 | Journal article
EID:

2-s2.0-77950537328

Contributors: Chiechio, S.; Copani, A.; Zammataro, M.; Battaglia, G.; IV, R.W.G.; Nicoletti, F.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Epigenetic modulation of mGlu2 receptors by histone deacetylase inhibitors in the treatment of inflammatory pain

Molecular Pharmacology
2009 | Journal article
EID:

2-s2.0-66049148780

Contributors: Chiechio, S.; Zammataro, M.; Morales, M.E.; Busceti, C.L.; Drago, F.; Gereau IV, R.W.; Copani, A.; Nicoletti, F.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Pregabalin in the treatment of chronic pain: An overview

Clinical Drug Investigation
2009 | Journal article
EID:

2-s2.0-61349198712

Contributors: Chiechio, S.; Zammataro, M.; Caraci, F.; Rampello, L.; Copani, A.; Sabato, A.F.; Nicoletti, F.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Targeting chronic pain with epigenetic drugs: Focus on mGlu2 receptors

Molecular and Cellular Pharmacology
2009 | Journal article
EID:

2-s2.0-77953376316

Contributors: Chiechio, S.; Zammataro, M.; Gereau IV, R.W.; Copani, A.; Nicoletti, F.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Acetyl-L-Carnitine in Neuropathic Pain: Experimental Data

CNS Drugs
2007 | Journal article
EID:

2-s2.0-35348878570

Contributors: Chiechio, S.; Copani, A.; Gereau, R.W.; Nicoletti, F.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Bone morphogenetic protein-7 delays podocyte injury due to high glucose

Nephrology Dialysis Transplantation
2007 | Journal article
EID:

2-s2.0-36749101547

Contributors: De Petris, L.; Hruska, K.A.; Chiechio, S.; Liapis, H.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Mice lacking central serotonergic neurons show enhanced inflammatory pain and an impaired analgesic response to antidepressant drugs

Journal of Neuroscience
2007 | Journal article
EID:

2-s2.0-34249815184

Contributors: Zhao, Z.-Q.; Chiechio, S.; Sun, Y.-G.; Zhang, K.-H.; Zhao, C.-S.; Scott, M.; Johnson, R.L.; Deneris, E.S.; Renner, K.J.; Gereau IV, R.W. et al.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

L-Acetylcarnitine: A proposed therapeutic agent for painful peripheral neuropathies

Current Neuropharmacology
2006 | Journal article
EID:

2-s2.0-33747270685

Contributors: Chiechio, S.; Copani, A.; Nicoletti, F.; Gereau IV, R.W.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Lmx1b is required for maintenance of central serotonergic neurons and mice lacking central serotonergic system exhibit normal locomotor activity

Journal of Neuroscience
2006 | Journal article
EID:

2-s2.0-33845423914

Contributors: Zhao, Z.-Q.; Scott, M.; Chiechio, S.; Wang, J.-S.; Renner, K.J.; Gereau IV, R.W.; Johnson, R.L.; Deneris, E.S.; Chen, Z.-F.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Transcriptional regulation of metabotropic glutamate receptor 2/3 expression by the NF-κB pathway in primary dorsal root ganglia neurons: A possible mechanism for the analgesic effect of L-acetylcarnitine

Molecular Pain
2006 | Journal article
EID:

2-s2.0-33747611426

Contributors: Chiechio, S.; Copani, A.; De Petris, L.; Morales, M.E.P.; Nicoletti, F.; Gereau IV, R.W.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

An evaluation of efficacy and safety of reboxetine in elderly patients affected by "retarded" post-stroke depression: A random, placebo-controlled study

Archives of Gerontology and Geriatrics
2005 | Journal article
EID:

2-s2.0-16244407729

Contributors: Rampello, L.; Alvano, A.; Chiechio, S.; Raffaele, R.; Vecchio, I.; Malaguarnera, M.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Evaluation of the prophylactic efficacy of amitriptyline and citalopram, alone or in combination, in patients with comorbidity of depression, migraine, and tension-type headache

Neuropsychobiology
2004 | Journal article
EID:

2-s2.0-8344281496

Contributors: Rampello, L.; Alvano, A.; Chiechio, S.; Malaguarnera, M.; Raffaele, R.; Vecchio, I.; Nicoletti, F.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Metabotropic receptors as targets for drugs of potential use in the treatment of neuropathic pain.

Journal of endocrinological investigation
2004 | Journal article
EID:

2-s2.0-16544374841

Contributors: Chiechio, S.; Copani, A.; Melchiorri, D.; Canudas, A.M.; Storto, M.; Calvani, M.; Nicolai, R.; Nicoletti, F.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Novel neuronal targets for the acetylcholinesterase inhibitor donepezil

Neuropharmacology
2004 | Journal article
EID:

2-s2.0-9644301088

Contributors: Sortino, M.A.; Frasca, G.; Chisari, M.; Platania, P.; Chiechio, S.; Vancheri, C.; Copani, A.; Canonico, P.L.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

Prediction of the response to citalopram and reboxetine in post-stroke depressed patients

Psychopharmacology
2004 | Journal article
EID:

2-s2.0-2342510868

Contributors: Rampello, L.; Chiechio, S.; Nicoletti, G.; Alvano, A.; Vecchio, I.; Raffaele, R.; Malaguarnera, M.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

β-amyloid-activated cell cycle in SH-SY5Y neuroblastoma cells: Correlation with the MAP kinase pathway

Journal of Molecular Neuroscience
2004 | Journal article
EID:

2-s2.0-2942572699

Contributors: Frasca, G.; Chiechio, S.; Vancheri, C.; Nicoletti, F.; Copani, A.; Sortino, M.A.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier

An increased expression of the mGlu5 receptor protein following LTP induction at the perforant path-dentate gyrus synapse in freely moving rats

Neuropharmacology
2003 | Journal article
EID:

2-s2.0-12244297768

Contributors: Manahan-Vaughan, D.; Ngomba, R.T.; Storto, M.; Kulla, A.; Catania, M.V.; Chiechio, S.; Rampello, L.; Passarelli, F.; Capece, A.; Reymann, K.G. et al.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier
grade
Preferred source (of 2)‎

Effects of phenformin on the proliferation of human tumor cell lines

Life Sciences
2003 | Journal article
EID:

2-s2.0-0242459925

Contributors: Caraci, F.; Chisari, M.; Frasca, G.; Chiechio, S.; Salomone, S.; Pinto, A.; Sortino, M.A.; Bianchi, A.
Source: Self-asserted source
Santina Chiechio via Scopus - Elsevier
Items per page:
Page 1 of 2

Peer review (10 reviews for 7 publications/grants)

Review activity for Healthcare. (1)
Review activity for International journal of molecular sciences. (1)
Review activity for Life. (1)
Review activity for Medical sciences. (1)
Review activity for Nutrients. (2)
Review activity for Pharmaceuticals. (3)
Review activity for Pharmaceutics. (1)