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Works (24)

Anti-Diabetic Activity of Glycyrrhetinic Acid Derivatives FC-114 and FC-122: Scale-Up, In Silico, In Vitro, and In Vivo Studies

International Journal of Molecular Sciences
2023-08 | Journal article | Author
Contributors: Samuel Álvarez-Almazán; Luz Cassandra Solís-Domínguez; Paulina Duperou-Luna; Teresa Fuerte-Gómez; Martin González-Andrade; María E. Aranda-Barradas; Juan Francisco Palacios Espinosa; Jaime Pérez-Villanueva; Félix Matadamas-Martínez; SUSANA PATRICIA MIRANDA CASTRO et al.
Source: check_circle
Multidisciplinary Digital Publishing Institute

Casiopeinas of Third Generations: Synthesis, Characterization, Cytotoxic Activity and Structure–Activity Relationships of Mixed Chelate Compounds with Bioactive Secondary Ligands

Molecules
2022-05 | Journal article | Author
Contributors: Yeshenia Figueroa-DePaz; Jaime Pérez-Villanueva; Olivia Soria-Arteche; Diego Martínez-Otero; Virginia Gómez-Vidales; Luis Ortiz-Frade; Lena Ruiz-Azuara
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Multidisciplinary Digital Publishing Institute

Synthesis and Cytotoxic Activity of Combretastatin A-4 and 2,3-Diphenyl-2<i>H</i>-indazole Hybrids

Pharmaceuticals
2021-08 | Journal article | Author
Contributors: Jaime Pérez-Villanueva; Félix Matadamas-Martínez; Lilián Yépez-Mulia; Vadim Pérez Koldenkova; Martha Leyte-Lugo; Karen Rodríguez-Villar; Francisco Cortés-Benítez; Ana Perla Macías-Jiménez; Ignacio González-Sánchez; Ariana Romero-Velásquez et al.
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Multidisciplinary Digital Publishing Institute

Indole- and Pyrazole-Glycyrrhetinic Acid Derivatives as PTP1B Inhibitors: Synthesis, In Vitro and In Silico Studies

Molecules
2021-07 | Journal article | Author
Contributors: Ledy De-la-Cruz-Martínez; Constanza Duran-Becerra; Martin González-Andrade; José C. Páez-Franco; Juan Manuel Germán-Acacio; Julio Espinosa-Chávez; J. Martin Torres-Valencia; Jaime Pérez-Villanueva; Juan Francisco Palacios Espinosa; Olivia Soria-Arteche et al.
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Multidisciplinary Digital Publishing Institute

Synthesis, Antiprotozoal Activity, and Cheminformatic Analysis of 2-Phenyl-2<i>H</i>-Indazole Derivatives

Molecules
2021-04 | Journal article | Author
Contributors: Karen Rodríguez-Villar; Lilián Yépez-Mulia; Miguel Cortés-Gines; Jacobo David Aguilera-Perdomo; Edgar A. Quintana-Salazar; Kevin Samael Olascoaga Del Angel; Francisco Cortés-Benítez; Juan Francisco Palacios-Espinosa; Olivia Soria-Arteche; Jaime Pérez-Villanueva
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Multidisciplinary Digital Publishing Institute

Design, Synthesis and Anticandidal Evaluation of Indazole and Pyrazole Derivatives

Pharmaceuticals
2021-02 | Journal article | Author
Contributors: Karen Rodríguez-Villar; Alicia Hernández-Campos; Lilián Yépez-Mulia; Teresita del Rosario Sainz-Espuñes; Olivia Soria-Arteche; Juan Francisco Palacios-Espinosa; Francisco Cortés-Benítez; Martha Leyte-Lugo; Bárbara Varela-Petrissans; Edgar A. Quintana-Salazar et al.
Source: check_circle
Multidisciplinary Digital Publishing Institute

Benzoic acid derivatives with trypanocidal activity: Enzymatic analysis and molecular docking studies toward trans-sialidase

Molecules
2017 | Journal article
EID:

2-s2.0-85033782334

Part of ISBN:

14203049

Contributors: Kashif, M.; Moreno-Herrera, A.; Villalobos-Rocha, J.C.; Nogueda-Torres, B.; Pérez-Villanueva, J.; Rodríguez-Villar, K.; Medina-Franco, J.L.; De Andrade, P.; Carvalho, I.; Rivera, G.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Synthesis and biological evaluation of 2H-indazole derivatives: Towards antimicrobial and anti-inflammatory dual agents

Molecules
2017 | Journal article
EID:

2-s2.0-85033779771

Part of ISBN:

14203049

Contributors: Pérez-Villanueva, J.; Yépez-Mulia, L.; González-Sánchez, I.; Palacios-Espinosa, J.F.; Soria-Arteche, O.; Del Rosario Sainz-Espuñes, T.; Cerbón, M.A.; Rodríguez-Villar, K.; Rodríguez-Vicente, A.K.; Cortés-Gines, M. et al.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Synthesis of curcuminoids and evaluation of their cytotoxic and antioxidant properties

Molecules
2017 | Journal article
EID:

2-s2.0-85020231748

Part of ISBN:

14203049

Contributors: Lozada-García, M.C.; Enríquez, R.G.; Ramírez-Apán, T.O.; Nieto-Camacho, A.; Palacios-Espinosa, J.F.; Custodio-Galván, Z.; Soria-Arteche, O.; Pérez-Villanueva, J.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Activity cliffs and activity cliff generators based on chemotype-related activity landscapes

Molecular Diversity
2015 | Journal article
EID:

2-s2.0-84942981512

Part of ISBN:

1573501X 13811991

Contributors: Pérez-Villanueva, J.; Méndez-Lucio, O.; Soria-Arteche, O.; Medina-Franco, J.L.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Chemoinformatic characterization of activity and selectivity switches of antiprotozoal compounds

Future Medicinal Chemistry
2014 | Journal article
EID:

2-s2.0-84893109925

Part of ISBN:

17568927 17568919

Contributors: Aguayo-Ortiz, R.; Pérez-Villanueva, J.; Hernández-Campos, A.; Castillo, R.; Meurice, N.; Medina-Franco, J.L.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Cyclic systems distribution along similarity measures: Insights for an application to activity landscape modeling

Molecular Informatics
2013 | Journal article
EID:

2-s2.0-84874037909

Part of ISBN:

18681743 18681751

Contributors: Pérez-Villanueva, J.; Méndez-Lucio, O.; Soria-Arteche, O.; Izquierdo, T.; Concepciõn Lozada, M.; Gloria-Greimel, W.A.; Medina-Franco, J.L.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Synthesis and antiprotozoal activity of novel 2-{[2-(1H-imidazol-1-yl) ethyl]sulfanyl}-1H-benzimidazole derivatives

Bioorganic and Medicinal Chemistry Letters
2013 | Journal article
EID:

2-s2.0-84879417008

Part of ISBN:

0960894X 14643405

Contributors: Pérez-Villanueva, J.; Hernández-Campos, A.; Yépez-Mulia, L.; Méndez-Cuesta, C.; Méndez-Lucio, O.; Hernández-Luis, F.; Castillo, R.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Activity landscape modeling of PPAR ligands with dual-activity difference maps

Bioorganic and Medicinal Chemistry
2012 | Journal article
EID:

2-s2.0-84861193545

Part of ISBN:

09680896 14643391

Contributors: Méndez-Lucio, O.; Pérez-Villanueva, J.; Castillo, R.; Medina-Franco, J.L.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

CASE Plots for the Chemotype-Based Activity and Selectivity Analysis: A CASE Study of Cyclooxygenase Inhibitors

Chemical Biology and Drug Design
2012 | Journal article
EID:

2-s2.0-84867231295

Part of ISBN:

17470277 17470285

Contributors: Pérez-Villanueva, J.; Medina-Franco, J.L.; Méndez-Lucio, O.; Yoo, J.; Soria-Arteche, O.; Izquierdo, T.; Lozada, M.C.; Castillo, R.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Identifying activity cliff generators of PPAR ligands using SAS maps

Molecular Informatics
2012 | Journal article
EID:

2-s2.0-84872826468

Part of ISBN:

18681743 18681751

Contributors: Méndez-Lucio, O.; Pérez-Villanueva, J.; Castillo, R.; Medina-Franco, J.L.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

In vitro and in vivo trypanocidal activity of some benzimidazole derivatives against two strains of Trypanosoma cruzi

Acta Tropica
2012 | Journal article
EID:

2-s2.0-84857115113

Part of ISBN:

0001706X 18736254

Contributors: Díaz-Chiguer, D.L.; Márquez-Navarro, A.; Nogueda-Torres, B.; de la Luz León-ávila, G.; Pérez-Villanueva, J.; Hernández-Campos, A.; Castillo, R.; Ambrosio, J.R.; Nieto-Meneses, R.; Yépez-Mulia, L. et al.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

3D-QSAR studies on purine-carbonitriles as cruzain inhibitors: Comparative molecular field analysis (CoMFA) and comparative molecular similarity indices analysis (CoMSIA)

MedChemComm
2011 | Journal article
EID:

2-s2.0-80455163178

Part of ISBN:

20402503 20402511

Contributors: Méndez-Lucio, O.; Pérez-Villanueva, J.; Romo-Mancillas, A.; Castillo, R.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Antiprotozoal activity of proton-pump inhibitors

Bioorganic and Medicinal Chemistry Letters
2011 | Journal article
EID:

2-s2.0-81255199185

Part of ISBN:

0960894X 14643405

Contributors: Pérez-Villanueva, J.; Romo-Mancillas, A.; Hernández-Campos, A.; Yépez-Mulia, L.; Hernández-Luis, F.; Castillo, R.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Comparative molecular field analysis (CoMFA) and comparative molecular similarity indices analysis (CoMSIA) of some benzimidazole derivatives with trichomonicidal activity

European Journal of Medicinal Chemistry
2011 | Journal article
EID:

2-s2.0-79958252481

Part of ISBN:

02235234 17683254

Contributors: Pérez-Villanueva, J.; Medina-Franco, J.L.; Caulfield, T.R.; Hernández-Campos, A.; Hernández-Luis, F.; Yépez-Mulia, L.; Castillo, R.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Multitarget structure-activity relationships characterized by activity-difference maps and consensus similarity measure

Journal of Chemical Information and Modeling
2011 | Journal article
EID:

2-s2.0-80053327464

Part of ISBN:

15499596 15205142

Contributors: Medina-Franco, J.L.; Yongye, A.B.; Pérez-Villanueva, J.; Houghten, R.A.; Martínez-Mayorga, K.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Structure-activity relationships of benzimidazole derivatives as antiparasitic agents: Dual activity-difference (DAD) maps

MedChemComm
2011 | Journal article
EID:

2-s2.0-79952451546

Part of ISBN:

20402503 20402511

Contributors: Pérez-Villanueva, J.; Santos, R.; Hernández-Campos, A.; Giulianotti, M.A.; Castillo, R.; Medina-Franco, J.L.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Towards a systematic characterization of the antiprotozoal activity landscape of benzimidazole derivatives

Bioorganic and Medicinal Chemistry
2010 | Journal article
EID:

2-s2.0-77957991633

Part of ISBN:

09680896

Contributors: Pérez-Villanueva, J.; Santos, R.; Hernández-Campos, A.; Giulianotti, M.A.; Castillo, R.; Medina-Franco, J.L.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Synthesis and in vitro cysticidal activity of new benzimidazole derivatives

European Journal of Medicinal Chemistry
2009 | Journal article
EID:

2-s2.0-61349184552

Part of ISBN:

02235234 17683254

Contributors: Palomares-Alonso, F.; Jung-Cook, H.; Pérez-Villanueva, J.; Piliado, J.C.; Rodríguez-Morales, S.; Palencia-Hernández, G.; López-Balbiaux, N.; Hernández-Campos, A.; Castillo, R.; Hernández-Luis, F.
Source: Self-asserted source
Jaime Pérez-Villanueva via Scopus - Elsevier

Peer review (2 reviews for 2 publications/grants)

Review activity for Computation. (1)
Review activity for Molecules. (1)