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Chromosome-specific retention of cancer-associated DNA hypermethylation following pharmacological inhibition of DNMT1

Communications Biology
2022-06-02 | Journal article
Contributors: Ashley K. Wiseman; Rochelle L. Tiedemann; Huihui Fan; Hui Shen; Zachary Madaj; Michael T. McCabe; Melissa B. Pappalardi; Peter A. Jones
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Discovery of a first-in-class reversible DNMT1-selective inhibitor with improved tolerability and efficacy in acute myeloid leukemia

Nature Cancer
2021-09-27 | Journal article
Contributors: Melissa B. Pappalardi; Kathryn Keenan; Mark Cockerill; Wendy A. Kellner; Alexandra Stowell; Christian Sherk; Kristen Wong; Sarath Pathuri; Jacques Briand; Michael Steidel et al.
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