Personal information

United States

Activities

Employment (3)

Vanderbilt University School of Medicine: Nashville, TN, US

2023-06-01 to present | Drug Discovery Scientist (Biochemistry)
Employment
Source: Self-asserted source
Kangsa Amporndanai

Vanderbilt University: Nashville, Tennessee, US

2021-06-14 to 2023-05-31 | Postdoctoral Scholar (Biochemistry)
Employment
Source: Self-asserted source
Kangsa Amporndanai

University of Liverpool: Liverpool, Merseyside, GB

2019-04-01 to 2021-03-31 | Postdoctoral Research Associate (Biochemistry & Systems Biology)
Employment
Source: Self-asserted source
Kangsa Amporndanai

Education and qualifications (1)

University of Liverpool: Liverpool, Merseyside, GB

2014-12-01 to 2018-11-30 | Doctor of Philosophy (Biochemistry)
Education
Source: Self-asserted source
Kangsa Amporndanai

Works (12)

Fragment-Based Screen of SARS-CoV-2 Papain-like Protease (PLpro)

ACS Medicinal Chemistry Letters
2024-08-08 | Journal article
Contributors: Ashley J. Taylor; Kangsa Amporndanai; Tyson A. Rietz; Bin Zhao; Anusha Thiruvaipati; Qiangqiang Wei; Taylor M. South; Mackenzie M. Crow; Chideraa Apakama; John L. Sensintaffar et al.
Source: check_circle
Crossref
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Preferred source (of 2)‎

Ebselen analogues delay disease onset and its course in fALS by on-target SOD-1 engagement

Scientific Reports
2024-05-27 | Journal article
Part of ISSN: 2045-2322
Contributors: Seiji Watanabe; Kangsa Amporndanai; Raheela Awais; Caroline Latham; Muhammad Awais; Paul M. O’Neill; Koji Yamanaka; S. Samar Hasnain
Source: Self-asserted source
Kangsa Amporndanai

Structure-Based Discovery of Potent, Orally Bioavailable Benzoxazepinone-Based WD Repeat Domain 5 Inhibitors

Journal of Medicinal Chemistry
2023-12-28 | Journal article | Author
Part of ISSN: 0022-2623
Part of ISSN: 1520-4804
Contributors: Kevin B. Teuscher; Jonathan Mills; Jianhua Tian; Changho Han; Kenneth M. Meyers; Jiqing Sai; Taylor M. South; Mackenzie M. Crow; Mayme Van Meveren; John L. Sensintaffar et al.
Source: Self-asserted source
Kangsa Amporndanai

Targeting the Ubiquinol-Reduction (Qi) Site of the Mitochondrial Cytochrome bc1 Complex for the Development of Next Generation Quinolone Antimalarials

Biology
2022-07-25 | Journal article
Part of ISSN: 2079-7737
Source: Self-asserted source
Kangsa Amporndanai

Parasitological profiling shows 4(1H)-quinolone derivatives as new lead candidates for malaria

European Journal of Medicinal Chemistry Reports
2021-10-23 | Journal article
Part of ISSN: 2772-4174
Source: Self-asserted source
Kangsa Amporndanai

Inhibition mechanism of SARS-CoV-2 main protease by ebselen and its derivatives

Nature Communications
2021-05-24 | Journal article
Part of ISSN: 2041-1723
Source: Self-asserted source
Kangsa Amporndanai

Ebselen as template for stabilization of A4V mutant dimer for motor neuron disease therapy

Communications Biology
2020 | Journal article
EID:

2-s2.0-85081386331

Part of ISSN: 23993642
Contributors: Chantadul, V.; Wright, G.S.A.; Amporndanai, K.; Shahid, M.; Antonyuk, S.V.; Washbourn, G.; Rogers, M.; Roberts, N.; Pye, M.; O’Neill, P.M. et al.
Source: Self-asserted source
Kangsa Amporndanai via Scopus - Elsevier

Novel Selenium-based compounds with therapeutic potential for SOD1-linked amyotrophic lateral sclerosis

EBioMedicine
2020 | Journal article
EID:

2-s2.0-85089837737

Part of ISSN: 23523964
Contributors: Amporndanai, K.; Rogers, M.; Watanabe, S.; Yamanaka, K.; O'Neill, P.M.; Hasnain, S.S.
Source: Self-asserted source
Kangsa Amporndanai via Scopus - Elsevier

Potent Tetrahydroquinolone Eliminates Apicomplexan Parasites

Frontiers in Cellular and Infection Microbiology
2020 | Journal article
EID:

2-s2.0-85087309623

Part of ISSN: 22352988
Contributors: McPhillie, M.J.; Zhou, Y.; Hickman, M.R.; Gordon, J.A.; Weber, C.R.; Li, Q.; Lee, P.J.; Amporndanai, K.; Johnson, R.M.; Darby, H. et al.
Source: Self-asserted source
Kangsa Amporndanai via Scopus - Elsevier

Purification and Structural Characterization of Aggregation-Prone Human TDP-43 Involved in Neurodegenerative Diseases

iScience
2020 | Journal article
EID:

2-s2.0-85085285767

Part of ISSN: 25890042
Contributors: Wright, G.S.A.; Watanabe, T.F.; Amporndanai, K.; Plotkin, S.S.; Cashman, N.R.; Antonyuk, S.V.; Hasnain, S.S.
Source: Self-asserted source
Kangsa Amporndanai via Scopus - Elsevier

Potent Antimalarial 2-Pyrazolyl Quinolone bc<inf>1</inf> (Q<inf>i</inf>) Inhibitors with Improved Drug-like Properties

ACS Medicinal Chemistry Letters
2018 | Journal article
EID:

2-s2.0-85056458774

Part of ISSN: 19485875
Contributors: David Hong, W.; Leung, S.C.; Amporndanai, K.; Davies, J.; Priestley, R.S.; Nixon, G.L.; Berry, N.G.; Samar Hasnain, S.; Antonyuk, S.; Ward, S.A. et al.
Source: Self-asserted source
Kangsa Amporndanai via Scopus - Elsevier

X-ray and cryo-EM structures of inhibitor-bound cytochrome bc 1 complexes for structure-based drug discovery

IUCrJ
2018 | Journal article
EID:

2-s2.0-85043248409

Part of ISSN: 20522525
Contributors: Amporndanai, K.; Johnson, R.M.; O'Neill, P.M.; Fishwick, C.W.G.; Jamson, A.H.; Rawson, S.; Muench, S.P.; Samar Hasnain, S.; Antonyuk, S.V.
Source: Self-asserted source
Kangsa Amporndanai via Scopus - Elsevier