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Data from STimulator of INterferon Genes Agonism Accelerates Antitumor Activity in Poorly Immunogenic Tumors

2023-04-03 | Preprint
Contributors: Samanthi A. Perera; Johnny E. Kopinja; Yanhong Ma; Eric S. Muise; Jason Laskey; Kalyan Chakravarthy; Yiping Chen; Long Cui; Jeremy Presland; Manjiri Sathe et al.
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Data from STimulator of INterferon Genes Agonism Accelerates Antitumor Activity in Poorly Immunogenic Tumors

2023-04-03 | Preprint
Contributors: Samanthi A. Perera; Johnny E. Kopinja; Yanhong Ma; Eric S. Muise; Jason Laskey; Kalyan Chakravarthy; Yiping Chen; Long Cui; Jeremy Presland; Manjiri Sathe et al.
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Figure S1 from STimulator of INterferon Genes Agonism Accelerates Antitumor Activity in Poorly Immunogenic Tumors

2023-04-03 | Preprint
Contributors: Samanthi A. Perera; Johnny E. Kopinja; Yanhong Ma; Eric S. Muise; Jason Laskey; Kalyan Chakravarthy; Yiping Chen; Long Cui; Jeremy Presland; Manjiri Sathe et al.
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Figure S1 from STimulator of INterferon Genes Agonism Accelerates Antitumor Activity in Poorly Immunogenic Tumors

2023-04-03 | Preprint
Contributors: Samanthi A. Perera; Johnny E. Kopinja; Yanhong Ma; Eric S. Muise; Jason Laskey; Kalyan Chakravarthy; Yiping Chen; Long Cui; Jeremy Presland; Manjiri Sathe et al.
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Crossref

Figure S2 from STimulator of INterferon Genes Agonism Accelerates Antitumor Activity in Poorly Immunogenic Tumors

2023-04-03 | Preprint
Contributors: Samanthi A. Perera; Johnny E. Kopinja; Yanhong Ma; Eric S. Muise; Jason Laskey; Kalyan Chakravarthy; Yiping Chen; Long Cui; Jeremy Presland; Manjiri Sathe et al.
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Figure S2 from STimulator of INterferon Genes Agonism Accelerates Antitumor Activity in Poorly Immunogenic Tumors

2023-04-03 | Preprint
Contributors: Samanthi A. Perera; Johnny E. Kopinja; Yanhong Ma; Eric S. Muise; Jason Laskey; Kalyan Chakravarthy; Yiping Chen; Long Cui; Jeremy Presland; Manjiri Sathe et al.
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Figure S3 from STimulator of INterferon Genes Agonism Accelerates Antitumor Activity in Poorly Immunogenic Tumors

2023-04-03 | Preprint
Contributors: Samanthi A. Perera; Johnny E. Kopinja; Yanhong Ma; Eric S. Muise; Jason Laskey; Kalyan Chakravarthy; Yiping Chen; Long Cui; Jeremy Presland; Manjiri Sathe et al.
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Crossref

Figure S3 from STimulator of INterferon Genes Agonism Accelerates Antitumor Activity in Poorly Immunogenic Tumors

2023-04-03 | Preprint
Contributors: Samanthi A. Perera; Johnny E. Kopinja; Yanhong Ma; Eric S. Muise; Jason Laskey; Kalyan Chakravarthy; Yiping Chen; Long Cui; Jeremy Presland; Manjiri Sathe et al.
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Crossref

Supplementary Data from STimulator of INterferon Genes Agonism Accelerates Antitumor Activity in Poorly Immunogenic Tumors

2023-04-03 | Preprint
Contributors: Samanthi A. Perera; Johnny E. Kopinja; Yanhong Ma; Eric S. Muise; Jason Laskey; Kalyan Chakravarthy; Yiping Chen; Long Cui; Jeremy Presland; Manjiri Sathe et al.
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Crossref

Supplementary Data from STimulator of INterferon Genes Agonism Accelerates Antitumor Activity in Poorly Immunogenic Tumors

2023-04-03 | Preprint
Contributors: Samanthi A. Perera; Johnny E. Kopinja; Yanhong Ma; Eric S. Muise; Jason Laskey; Kalyan Chakravarthy; Yiping Chen; Long Cui; Jeremy Presland; Manjiri Sathe et al.
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Crossref

Table S1 from STimulator of INterferon Genes Agonism Accelerates Antitumor Activity in Poorly Immunogenic Tumors

2023-04-03 | Preprint
Contributors: Samanthi A. Perera; Johnny E. Kopinja; Yanhong Ma; Eric S. Muise; Jason Laskey; Kalyan Chakravarthy; Yiping Chen; Long Cui; Jeremy Presland; Manjiri Sathe et al.
Source: check_circle
Crossref

Table S1 from STimulator of INterferon Genes Agonism Accelerates Antitumor Activity in Poorly Immunogenic Tumors

2023-04-03 | Preprint
Contributors: Samanthi A. Perera; Johnny E. Kopinja; Yanhong Ma; Eric S. Muise; Jason Laskey; Kalyan Chakravarthy; Yiping Chen; Long Cui; Jeremy Presland; Manjiri Sathe et al.
Source: check_circle
Crossref

STimulator of INterferon Genes Agonism Accelerates Antitumor Activity in Poorly Immunogenic Tumors

Molecular Cancer Therapeutics
2022-02-01 | Journal article
Contributors: Samanthi A. Perera; Johnny E. Kopinja; Yanhong Ma; Eric S. Muise; Jason Laskey; Kalyan Chakravarthy; Yiping Chen; Long Cui; Jeremy Presland; Manjiri Sathe et al.
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Crossref

An orally available non-nucleotide STING agonist with antitumor activity.

Science (New York, N.Y.)
2020-08-01 | Journal article
Source: Self-asserted source
Jeremy Presland
grade
Preferred source (of 2)‎

Determination of EPAC2 function using EPAC2 null Min6 sublines generated through CRISPR-Cas9 technology

Molecular and Cellular Endocrinology
2018 | Journal article
EID:

2-s2.0-85041615112

Part of ISBN:

18728057 03037207

Contributors: Xu, H.; Yang, Y.; Chen, Y.; Mueller, U.; Iyer, S.; Presland, J.; Yang, R.; Kariv, I.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Discovery of 3-morpholino-imidazole[1,5-a]pyrazine BTK inhibitors for rheumatoid arthritis

Bioorganic and Medicinal Chemistry Letters
2017 | Journal article
EID:

2-s2.0-85023648195

Part of ISBN:

14643405 0960894X

Contributors: Boga, S.B.; Alhassan, A.-B.; Liu, J.; Guiadeen, D.; Krikorian, A.; Gao, X.; Wang, J.; Yu, Y.; Anand, R.; Liu, S. et al.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Discovery of novel BTK inhibitors with carboxylic acids

Bioorganic and Medicinal Chemistry Letters
2017 | Journal article
EID:

2-s2.0-85013078020

Part of ISBN:

14643405 0960894X

Contributors: Gao, X.; Wang, J.; Liu, J.; Guiadeen, D.; Krikorian, A.; Boga, S.B.; Alhassan, A.-B.; Selyutin, O.; Yu, W.; Yu, Y. et al.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Identification of quinazoline based inhibitors of IRAK4 for the treatment of inflammation

Bioorganic and Medicinal Chemistry Letters
2017 | Journal article
EID:

2-s2.0-85019140510

Part of ISBN:

14643405 0960894X

Contributors: Smith, G.F.; Altman, M.D.; Andresen, B.; Baker, J.; Brubaker, J.D.; Chen, H.; Chen, Y.; Childers, M.; Donofrio, A.; Ferguson, H. et al.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Label-Free, LC-MS-Based Assays to Quantitate Small-Molecule Antagonist Binding to the Mammalian BLT1 Receptor

SLAS Discovery
2017 | Journal article
EID:

2-s2.0-85030251744

Part of ISBN:

24725560 24725552

Contributors: Chen, X.; Stout, S.; Mueller, U.; Boykow, G.; Visconti, R.; Siliphaivanh, P.; Spencer, K.; Presland, J.; Kavana, M.; Basso, A.D. et al.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Discovery of 8-Amino-imidazo[1,5-a]pyrazines as Reversible BTK Inhibitors for the Treatment of Rheumatoid Arthritis

ACS Medicinal Chemistry Letters
2016 | Journal article
EID:

2-s2.0-84958983955

Part of ISBN:

19485875

Contributors: Liu, J.; Guiadeen, D.; Krikorian, A.; Gao, X.; Wang, J.; Boga, S.B.; Alhassan, A.-B.; Yu, Y.; Vaccaro, H.; Liu, S. et al.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Discovery of 5-Amino- N -(1 H -pyrazol-4-yl)pyrazolo[1,5- a ]pyrimidine-3-carboxamide Inhibitors of IRAK4

ACS Medicinal Chemistry Letters
2015 | Journal article
EID:

2-s2.0-84931266819

Part of ISBN:

19485875

Contributors: Lim, J.; Altman, M.D.; Baker, J.; Brubaker, J.D.; Chen, H.; Chen, Y.; Fischmann, T.; Gibeau, C.; Kleinschek, M.A.; Leccese, E. et al.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Identification of N-(1H-pyrazol-4-yl)carboxamide inhibitors of interleukin-1 receptor associated kinase 4: Bicyclic core modifications

Bioorganic and Medicinal Chemistry Letters
2015 | Journal article
EID:

2-s2.0-84945898903

Part of ISBN:

14643405 0960894X

Contributors: Lim, J.; Altman, M.D.; Baker, J.; Brubaker, J.D.; Chen, H.; Chen, Y.; Kleinschek, M.A.; Li, C.; Liu, D.; Maclean, J.K.F. et al.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Identification and optimisation of novel sulfonamide, selective vasopressin V <inf>1B</inf> receptor antagonists

Bioorganic and Medicinal Chemistry Letters
2011 | Journal article
EID:

2-s2.0-79957823437

Part of ISBN:

0960894X 14643405

Contributors: Baker, J.; Bingham, M.; Blackburn-Munro, R.; Cai, J.; Craighead, M.; Gilfillan, R.; Goan, K.; Jaap, D.; Milne, R.; Richard Morphy, J. et al.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Optimisation of pharmacokinetic properties to afford an orally bioavailable and selective V <inf>1A</inf> receptor antagonist

Bioorganic and Medicinal Chemistry Letters
2011 | Journal article
EID:

2-s2.0-79960360059

Part of ISBN:

0960894X 14643405

Contributors: Arbuckle, W.; Baker, J.; Barn, D.; Bingham, M.; Brown, A.; Buchanan, K.; Craighead, M.; Goodwin, R.; Goutcher, S.; Kiczun, M. et al.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Synthesis and SAR studies of novel 2-(4-oxo-2-aryl-quinazolin-3(4H)-yl) acetamide vasopressin V<inf>1b</inf> receptor antagonists

Bioorganic and Medicinal Chemistry Letters
2011 | Journal article
EID:

2-s2.0-79952363767

Part of ISBN:

0960894X

Contributors: Napier, S.E.; Letourneau, J.J.; Ansari, N.; Auld, D.S.; Baker, J.; Best, S.; Campbell-Wan, L.; Chan, J.-H.; Craighead, M.; Desai, H. et al.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Synthesis and SAR studies of novel 2-(6-aminomethylaryl-2-aryl-4-oxo- quinazolin-3(4H)-yl)acetamide Vasopressin V <inf>1b</inf> receptor antagonists

Bioorganic and Medicinal Chemistry Letters
2011 | Journal article
EID:

2-s2.0-79957797698

Part of ISBN:

0960894X 14643405

Contributors: Napier, S.E.; Letourneau, J.J.; Ansari, N.; Auld, D.S.; Baker, J.; Best, S.; Campbell-Wan, L.; Chan, R.; Craighead, M.; Desai, H. et al.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

The discovery of novel 8-azabicyclo[3.2.1]octan-3-yl)-3-(4-chlorophenyl) propanamides as vasopressin V<inf>1A</inf> receptor antagonists

Bioorganic and Medicinal Chemistry Letters
2011 | Journal article
EID:

2-s2.0-79955555074

Part of ISBN:

0960894X

Contributors: Napier, S.; Wishart, G.; Arbuckle, W.; Baker, J.; Barn, D.; Bingham, M.; Brown, A.; Byford, A.; Claxton, C.; Craighead, M. et al.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

The discovery and SAR of indoline-3-carboxamides - A new series of 5-HT<inf>6</inf> antagonists

Bioorganic and Medicinal Chemistry Letters
2010 | Journal article
EID:

2-s2.0-77954218444

Part of ISBN:

0960894X

Contributors: Reid, M.; Carlyle, I.; Caulfield, W.L.; Clarkson, T.R.; Cusick, F.; Epemolu, O.; Gilfillan, R.; Goodwin, R.; Jaap, D.; O'Donnell, E.C. et al.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Characterization of a novel and selective V<inf>1B</inf> receptor antagonist

Progress in Brain Research
2008 | Book
EID:

2-s2.0-47549103890

Part of ISBN:

00796123

Contributors: Craighead, M.; Milne, R.; Campbell-Wan, L.; Watson, L.; Presland, J.; Thomson, F.J.; Marston, H.M.; MacSweeney, C.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

G-protein-coupled receptor heterodimerization: Assay technologies to clinical significance

Current Opinion in Drug Discovery and Development
2007 | Journal article
EID:

2-s2.0-34548421579

Part of ISBN:

13676733

Contributors: Kent, T.; McAlpine, C.; Sabetnia, S.; Presland, J.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Identifying novel modulators of G protein-coupled receptors via interaction at allosteric sites

Current Opinion in Drug Discovery and Development
2005 | Journal article
EID:

2-s2.0-24044493211

Part of ISBN:

13676733

Contributors: Presland, J.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

G-protein-coupled receptor accessory proteins: Their potential role in future drug discovery

Biochemical Society Transactions
2004 | Journal article
EID:

2-s2.0-8744302247

Part of ISBN:

03005127

Contributors: Presland, J.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Pharmacological characterisation of the D<inf>2</inf> dopamine receptor expressed in the yeast Schizosaccharomyces pombe

Biochemical Pharmacology
1998 | Journal article
EID:

2-s2.0-0032148392

Part of ISBN:

00062952

Contributors: Presland, J.; Strange, P.G.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

Expression of the rat D, dopamine receptor in the yeast Saccharomyces cerevisiae

Biochemical Society Transactions
1993 | Journal article
EID:

2-s2.0-0027600445

Part of ISBN:

03005127

Contributors: Presland, J.P.; Strange, P.G.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier

pH dependence of sulpiride binding to D<inf>2</inf> dopamine receptors in bovine brain

Biochemical Pharmacology
1991 | Journal article
EID:

2-s2.0-0025972154

Part of ISBN:

00062952

Contributors: Presland, J.P.; Strange, P.G.
Source: Self-asserted source
Jeremy Presland via Scopus - Elsevier