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Works (31)

Evaluating Cross-linking-driven integrative modeling in peptide-HLAII complexes prediction with insights for refining predictive accuracy

2024-09-03 | Preprint
Contributors: Andrea Di Ianni; Luca M. Barbero; Kyra Cowan; Federico Riccardi Sirtori
Source: check_circle
Crossref

Assessing MAPPs assay as a tool to predict the immunogenicity potential of protein therapeutics

Life Science Alliance
2024-01 | Journal article
Contributors: Andrea Di Ianni; Tiziana Fraone; Piercesare Balestra; Kyra Cowan; Federico Riccardi Sirtori; Luca Barbero
Source: check_circle
Crossref

Development of a Liquid Chromatography and High-Resolution and -Accuracy Mass Spectrometry Method to Evaluate New Biotherapeutic Entity Processing in Human Liver Lysosomes

ImmunoHorizons
2023 | Journal article
EID:

2-s2.0-85163273844

Part of ISSN: 25737732
Contributors: Colangelo, G.S.; Di Ianni, A.; Cowan, K.; Sirtori, F.R.; Barbero, L.M.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Hybrid liquid chromatography high resolution and accuracy mass spectrometry approach for quantification of antibody-drug conjugates at the intact protein level in biological samples

European Journal of Pharmaceutical Sciences
2023 | Journal article
EID:

2-s2.0-85163034343

Part of ISSN: 18790720 09280987
Contributors: Barbero, L.M.; Ianni, A.D.; Molinaro, F.; Cowan, K.J.; Sirtori, F.R.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Preclinical risk assessment strategy to mitigate the T-cell dependent immunogenicity of protein biotherapeutics: State of the art, challenges and future perspectives

Journal of Pharmaceutical and Biomedical Analysis
2023 | Journal article
EID:

2-s2.0-85163086860

Part of ISSN: 1873264X 07317085
Contributors: Di Ianni, A.; Barbero, L.; Fraone, T.; Cowan, K.; Sirtori, F.R.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

2022 White Paper on Recent Issues in Bioanalysis: ICH M10 BMV Guideline &amp; Global Harmonization; Hybrid Assays; Oligonucleotides &amp; ADC; Non-Liquid &amp; Rare Matrices; Regulatory Inputs (<u>Part 1A</u> – Recommendations on Mass Spectrometry, Chromatography and Sample Preparation, Novel Technologies, Novel Modalities, and Novel Challenges, ICH M10 BMV Guideline &amp; Global Harmonization <u>Part 1B</u> - Regulatory Agencies' Inputs on Regulated Bioanalysis/BMV, Biomarkers/CDx/BAV, Immunogenicity, Gene &amp; Cell Therapy and Vaccine)

Bioanalysis
2023-08 | Journal article
Part of ISSN: 1757-6180
Part of ISSN: 1757-6199
Contributors: Matt Szapacs; Wenying Jian; Daniel Spellman; Jennifer Cunliffe; Elizabeth Verburg; Surinder Kaur; John Kellie; Wenkui Li; John Mehl; Mark Qian et al.
Source: Self-asserted source
Federico Riccardi Sirtori

Assessing Major Histocompatibility Complex-Associated Peptide Proteomics assay as a tool to predict immunogenicity potential of protein therapeutics and antigens

Research Square
2022 | Other
EID:

2-s2.0-85167394010

Contributors: Barbero, L.; Ianni, A.D.; Fraone, T.; Balestra, P.; Cowan, K.; Sirtori, F.R.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Effect of Conjugation Site and Technique on the Stability and Pharmacokinetics of Antibody-Drug Conjugates

Journal of Pharmaceutical Sciences
2021 | Journal article
EID:

2-s2.0-85112846672

Part of ISSN: 15206017 00223549
Contributors: Kaempffe, A.; Dickgiesser, S.; Rasche, N.; Paoletti, A.; Bertotti, E.; De Salve, I.; Sirtori, F.R.; Kellner, R.; Könning, D.; Hecht, S. et al.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Identification of unprecedented ATP-competitive choline kinase inhibitors

Bioorganic and Medicinal Chemistry Letters
2021 | Journal article
EID:

2-s2.0-85114680705

Part of ISSN: 14643405 0960894X
Contributors: Quartieri, F.; Nesi, M.; Avanzi, N.R.; Borghi, D.; Casale, E.; Corti, E.; Cucchi, U.; Donati, D.; Fasolini, M.; Felder, E.R. et al.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Discovery of Stereospecific PARP-1 Inhibitor Isoindolinone NMS-P515

ACS Medicinal Chemistry Letters
2019 | Journal article
EID:

2-s2.0-85063157846

Part of ISSN: 19485875
Contributors: Papeo, G.; Orsini, P.; Avanzi, N.R.; Borghi, D.; Casale, E.; Ciomei, M.; Cirla, A.; Desperati, V.; Donati, D.; Felder, E.R. et al.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

MS methods to study macromolecule-ligand interaction: Applications in drug discovery

Methods
2018 | Journal article
EID:

2-s2.0-85048860371

Part of ISSN: 10959130 10462023
Contributors: Riccardi Sirtori, F.; Altomare, A.; Carini, M.; Aldini, G.; Regazzoni, L.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Virtual Cross-Linking of the Active Nemorubicin Metabolite PNU-159682 to Double-Stranded DNA

Chemical Research in Toxicology
2017 | Journal article
EID:

2-s2.0-85013243645

Part of ISSN: 15205010 0893228X
Contributors: Scalabrin, M.; Quintieri, L.; Palumbo, M.; Riccardi Sirtori, F.; Gatto, B.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Nemorubicin and doxorubicin bind the G-quadruplex sequences of the human telomeres and of the c-MYC promoter element Pu22

Biochimica et Biophysica Acta - General Subjects
2016 | Journal article
EID:

2-s2.0-84960156799

Part of ISSN: 18728006 03044165
Contributors: Scaglioni, L.; Mondelli, R.; Artali, R.; Sirtori, F.R.; Mazzini, S.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy

Journal of Medicinal Chemistry
2015 | Journal article
EID:

2-s2.0-84941551184

Part of ISSN: 15204804 00222623
Contributors: Papeo, G.; Posteri, H.; Borghi, D.; Busel, A.A.; Caprera, F.; Casale, E.; Ciomei, M.; Cirla, A.; Corti, E.; D'Anello, M. et al.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Effective immuno-targeting of the IDH1 mutation R132H in a murine model of intracranial glioma

Acta neuropathologica communications
2015 | Journal article
EID:

2-s2.0-85018199153

Part of ISSN: 20515960
Contributors: Pellegatta, S.; Valletta, L.; Corbetta, C.; Patanè, M.; Zucca, I.; Riccardi Sirtori, F.; Bruzzone, M.G.; Fogliatto, G.; Isacchi, A.; Pollo, B. et al.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Establish an automated flow injection ESI-MS method for the screening of fragment based libraries: Application to Hsp90

European Journal of Pharmaceutical Sciences
2015 | Journal article
EID:

2-s2.0-84929173141

Part of ISSN: 18790720 09280987
Contributors: Riccardi Sirtori, F.; Caronni, D.; Colombo, M.; Dalvit, C.; Paolucci, M.; Regazzoni, L.; Visco, C.; Fogliatto, G.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Insights into PARP inhibitors' selectivity using fluorescence polarization and surface plasmon resonance binding assays

Journal of Biomolecular Screening
2014 | Journal article
EID:

2-s2.0-84905594808

Part of ISSN: 1552454X 10870571
Contributors: Papeo, G.; Avanzi, N.; Bettoni, S.; Leone, A.; Paolucci, M.; Perego, R.; Quartieri, F.; Riccardi-Sirtori, F.; Thieffine, S.; Montagnoli, A. et al.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Mass spectrometric strategies for the identification and characterization of human serum albumin covalently adducted by amoxicillin: Ex Vivo Studies

Chemical Research in Toxicology
2014 | Journal article
EID:

2-s2.0-84918526640

Part of ISSN: 15205010 0893228X
Contributors: Garzon, D.; Ariza, A.; Regazzoni, L.; Clerici, R.; Altomare, A.; Sirtori, F.R.; Carini, M.; Torres, M.J.; Perez-Sala, D.; Aldini, G.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Preclinical characterization of the drug-delivery device dcbeads™ for transarterial chemoembolization of doxorubicin and nemorubicin, a methoxy-morpholinyl derivative

Doxorubicin: Biosynthesis, Clinical Uses and Health Implications
2014 | Book chapter
EID:

2-s2.0-84949034764

Contributors: Fiore, F.; Valota, O.; Ballinari, D.; Sirtori, F.R.; Colombo, M.; D'Antò, M.; Geroni, C.; Cappella, P.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Alkylsulfanyl-1,2,4-triazoles, a New Class of allosteric valosine containing protein inhibitors. Synthesis and structure-activity relationships

Journal of Medicinal Chemistry
2013 | Journal article
EID:

2-s2.0-84872815788

Part of ISSN: 15204804 00222623
Contributors: Polucci, P.; Magnaghi, P.; Angiolini, M.; Asa, D.; Avanzi, N.; Badari, A.; Bertrand, J.; Casale, E.; Cauteruccio, S.; Cirla, A. et al.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Development of biochemical assays for the identification of eIF4E-specific inhibitors

Journal of Biomolecular Screening
2012 | Journal article
EID:

2-s2.0-84861832788

Part of ISSN: 10870571 1552454X
Contributors: Visco, C.; Perrera, C.; Thieffine, S.; Sirtori, F.R.; D'Alessio, R.; Magnaghi, P.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Molecular Recognition of T:G Mismatched Base Pairs in DNA as Studied by Electrospray Ionization Mass Spectrometry

ChemMedChem
2012 | Journal article
EID:

2-s2.0-84861537606

Part of ISSN: 18607179 18607187
Contributors: Riccardi Sirtori, F.; Aldini, G.; Colombo, M.; Colombo, N.; Malyszko, J.; Vistoli, G.; D'Alessio, R.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

The interaction of nemorubicin metabolite PNU-159682 with DNA fragments d(CGTACG)<sub>2</sub>, d(CGATCG)<sub>2</sub> and d(CGCGCG)<sub>2</sub> shows a strong but reversible binding to G:C base pairs

Bioorganic and Medicinal Chemistry
2012 | Journal article
EID:

2-s2.0-84870038799

Contributors: Mazzini, S.; Scaglioni, L.; Mondelli, R.; Caruso, M.; Sirtori, F.R.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Thieno[3,2-c]pyrazoles: A novel class of Aurora inhibitors with favorable antitumor activity

Bioorganic and Medicinal Chemistry
2010 | Journal article
EID:

2-s2.0-77956652574

Part of ISSN: 09680896
Contributors: Bindi, S.; Fancelli, D.; Alli, C.; Berta, D.; Bertrand, J.A.; Cameron, A.D.; Cappella, P.; Carpinelli, P.; Cervi, G.; Croci, V. et al.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Cell division cycle 7 kinase inhibitors: 1H-pyrrolo[2,3-b]pyridines, synthesis and structure-activity relationships

Journal of Medicinal Chemistry
2009 | Journal article
EID:

2-s2.0-67650754045

Part of ISSN: 00222623
Contributors: Ermoli, A.; Bargiotti, A.; Brasca, M.G.; Ciavolella, A.; Colombo, N.; Fachin, G.; Isacchi, A.; Menichincheri, M.; Molinari, A.; Montagnoli, A. et al.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

User Reports

HPLC Made to Measure: A Practical Handbook for Optimization
2008 | Book chapter
EID:

2-s2.0-84889359741

Contributors: Schäfer, H.; Lohaus, C.; Meyer, H.E.; Marcus, K.; Bilke, H.; Wagner, K.; Arangio, M.; Sirtori, F.R.; Marcucci, K.; Razzano, G. et al.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

6-Substituted pyrrolo[3,4-c]pyrazoles: An improved class of CDK2 inhibitors

ChemMedChem
2007 | Journal article
EID:

2-s2.0-51049124334

Part of ISSN: 18607179 18607187
Contributors: Brasca, M.G.; Albanese, C.; Amici, R.; Ballinari, D.; Corti, L.; Croci, V.; Fancelli, D.; Fiorentini, F.; Nesi, M.; Orsini, P. et al.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

A fully automated method for accurate mass determination using high-performance liquid chromatography with a quadrupole/orthogonal acceleration time-of-flight mass spectrometer

Rapid Communications in Mass Spectrometry
2004 | Journal article
EID:

2-s2.0-1242316994

Part of ISSN: 09514198
Contributors: Colombo, M.; Sirtori, F.R.; Rizzo, V.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Synthesis of novel simplified eleutheside analogues with potent microtubule-stabilizing activity, using ring-closing metathesis as the key-step

Tetrahedron Letters
2003 | Journal article
EID:

2-s2.0-0037454986

Part of ISSN: 00404039
Contributors: Beumer, R.; Bayón, P.; Bugada, P.; Ducki, S.; Mongelli, N.; Sirtori, F.R.; Telser, J.; Gennari, C.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Synthesis of novel simplified sarcodictyin/eleutherobin analogs with potent microtubule-stabilizing activity, using ring closing metathesis as the key-step

Tetrahedron
2003 | Journal article
EID:

2-s2.0-0141961790

Part of ISSN: 00404020
Contributors: Beumer, R.; Bayón, P.; Bugada, P.; Ducki, S.; Mongelli, N.; Sirtori, F.R.; Telser, J.; Gennari, C.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

[GdPCP2A(H<sub>2</sub>O)<sub>2</sub>]<sup>-</sup>: A paramagnetic contrast agent designed for improved applications in magnetic resonance imaging

Journal of Medicinal Chemistry
2000 | Journal article
EID:

2-s2.0-0034687242

Contributors: Aime, S.; Botta, M.; Frullano, L.; Crich, S.G.; Giovenzana, G.; Pagliarin, R.; Palmisano, G.; Sirtori, F.R.; Sisti, M.
Source: Self-asserted source
Federico Riccardi Sirtori via Scopus - Elsevier

Peer review (5 reviews for 2 publications/grants)

Review activity for European journal of pharmaceutical sciences. (2)
Review activity for Journal of pharmaceutical & biomedical analysis. (3)