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Works (3)

Discovery and Characterization of a New Class of C5aR1 Antagonists Showing In Vivo Activity

Journal of Medicinal Chemistry
2024-03-14 | Journal article
Contributors: Francis Hubler; Dorte Renneberg; Hervé Siendt; Simon Stamm; Kurt Hilpert; Eva Caroff; Stephane Delahaye; Sylvie Froidevaux; Mark J. Murphy
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Design, Synthesis, and Pharmacological Evaluation of Benzimidazolo-thiazoles as Potent CXCR3 Antagonists with Therapeutic Potential in Autoimmune Diseases: Discovery of ACT-672125

Journal of Medicinal Chemistry
2022-09-08 | Journal article
Contributors: Eva Caroff; Emmanuel A. Meyer; Päivi Äänismaa; Sylvie Froidevaux; Marcel Keller; Luca Piali
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Discovery and In Vivo Evaluation of ACT-660602: A Potent and Selective Antagonist of the Chemokine Receptor CXCR3 for Autoimmune Diseases

Journal of Medicinal Chemistry
2022-09-08 | Journal article
Contributors: Emmanuel A. Meyer; Päivi Äänismaa; Sylvie Froidevaux; Marcel Keller; Luca Piali; Eva Caroff
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Peer review (4 reviews for 2 publications/grants)

Review activity for ACS medicinal chemistry letters. (1)
Review activity for Journal of medicinal chemistry. (3)