Personal information

No personal information available

Activities

Works (7)

Balancing Molecular Size, Activity, Permeability, and Other Properties: Drug Candidates in the Context of Their Chemical Structure Optimization

Journal of Chemical Information and Modeling
2024-08-26 | Journal article
Contributors: Maximilian Beckers; Finton Sirockin; Nikolas Fechner; Nikolaus Stiefl
Source: check_circle
Crossref

Prediction of Small-Molecule Developability Using Large-Scale In Silico ADMET Models

Journal of Medicinal Chemistry
2023-10-26 | Journal article
Contributors: Maximilian Beckers; Noé Sturm; Finton Sirockin; Nikolas Fechner; Nikolaus Stiefl
Source: check_circle
Crossref

PREFER: A New Predictive Modeling Framework for Molecular Discovery

Journal of Chemical Information and Modeling
2023-08-14 | Journal article
Contributors: Jessica Lanini; Gianluca Santarossa; Finton Sirockin; Richard Lewis; Nikolas Fechner; Hubert Misztela; Sarah Lewis; Krzysztof Maziarz; Megan Stanley; Marwin Segler et al.
Source: check_circle
Crossref

25 Years of Small-Molecule Optimization at Novartis: A Retrospective Analysis of Chemical Series Evolution

Journal of Chemical Information and Modeling
2022-12-12 | Journal article
Contributors: Maximilian Beckers; Nikolas Fechner; Nikolaus Stiefl
Source: check_circle
Crossref

Evolution of Novartis’ Small Molecule Screening Deck Design

Journal of Medicinal Chemistry
2020-12-10 | Journal article
Contributors: Ansgar Schuffenhauer; Nadine Schneider; Samuel Hintermann; Douglas Auld; Jutta Blank; Simona Cotesta; Caroline Engeloch; Nikolas Fechner; Christoph Gaul; Jerome Giovannoni et al.
Source: check_circle
Crossref

Automated Identification of Chemical Series: Classifying like a Medicinal Chemist

Journal of Chemical Information and Modeling
2020-06-22 | Journal article
Contributors: Franziska Kruger; Nikolas Fechner; Nikolaus Stiefl
Source: check_circle
Crossref

Chiral Cliffs: Investigating the Influence of Chirality on Binding Affinity

ChemMedChem
2018-07-06 | Journal article
Contributors: Nadine Schneider; Richard A. Lewis; Nikolas Fechner; Peter Ertl
Source: check_circle
Crossref

Peer review (1 review for 1 publication/grant)

Review activity for Journal of chemical information and modeling. (1)