Personal information

Countries

Japan

Activities

Collapse all

Employment (2)

Shionogi (Japan): Osaka, JP

2020-10-01 to present | Subgroup leader (API R&D Laboratory)
Employment
Source: Self-asserted source
Nobuaki Fukui

Shionogi (Japan): Osaka, JP

2012-04-01 to 2020-09-30 | Researcher (API R&D Laboratory))
Employment
Source: Self-asserted source
Nobuaki Fukui

Education and qualifications (1)

Tokyo Institute of Technology: Tokyo, JP

2009-04 to 2012-03 | Ph.D. in Science (Department of Chemistry)
Education
Source: Self-asserted source
Nobuaki Fukui

Professional activities (3)

The Japanese Society for Process Chemistry: Gifu, JP

2023-05 to present | 将来計画委員会
Service
Source: Self-asserted source
Nobuaki Fukui

The Society of Synthetic Organic Chemistry, Japan: Tokyo, JP

2023 | 有機合成化学協会賞(技術的なもの) / Synthetic Organic Chemistry Award, Japan
Distinction
Source: Self-asserted source
Nobuaki Fukui

The Chemical Society of Japan: Tokyo, JP

2012-04-12 | 日本化学会第 92 春季年会(2012)学生講演賞
Distinction
Source: Self-asserted source
Nobuaki Fukui

Works (19)

First-Generation Process Development for the Synthesis of Baloxavir Marboxil: Early-Stage Development of Synthetic Methods to Prepare Baloxavir Marboxil Intermediates

Organic Process Research & Development
2024-06-21 | Journal article
DOI: 10.1021/acs.oprd.3c00514
Contributors: Kosuke Anan; Masayoshi Miyagawa; Azusa Okano; Hideki Sugimoto; Naoki Miyake; Nobuaki Fukui; Akihito Kijima; Emi Tanimoto; Makoto Kawai
Source: check_circle
Crossref

Practical Manufacturing Process for Baloxavir Marboxil: Effective Selection and Replacement of Protective Group toward Enhancement of Crystallization-Induced Diastereomer Transformation

Organic Process Research & Development
2024-06-21 | Journal article
DOI: 10.1021/acs.oprd.3c00503
Contributors: Nobuaki Fukui; Setsuya Shibahara; Toshikatsu Maki; Tatsuhiko Ueno; Shuichi Yanagisawa; Kazuya Okamoto; Emi Tanimoto; Takafumi Ohara; Tatsuro Yasukata; Takayuki Tsuritani
Source: check_circle
Crossref

Practical Manufacturing Process for Baloxavir Marboxil: Efficient Route to a Tricyclic Triazinanone Scaffold

Organic Process Research & Development
2024-06-21 | Journal article
DOI: 10.1021/acs.oprd.3c00502
Contributors: Nobuaki Fukui; Toshikatsu Maki; Kazunori Ban; Akihito Kijima; Setsuya Shibahara; Kazuya Okamoto; Sho Kamiya; Tatsuro Yasukata; Takayuki Tsuritani
Source: check_circle
Crossref

バロキサビル マルボキシル中間体の実用的製造プロセスの開発：三環性トリアジナノン骨格の構築に関する研究

日本プロセス化学会2023サマーシンポジウム
2023-08-03 | Conference poster
Contributors: Nobuaki Fukui; Toshikatsu Maki; Takayuki Tsuritani
Source: Self-asserted source
Nobuaki Fukui

新規なホスホロアミダイトの開発とリガンド結合型オリゴヌクレオチドの効率的合成及び品質管理における利用

日本プロセス化学会2023サマーシンポジウム
2023-08-03 | Conference poster
Contributors: Nobuaki Fukui; Mitsuaki Sekiguchi; Shunsuke Ochi; Norikazu Kuroda; Takafumi Higuchi; Akira Kugimiya
Source: Self-asserted source
Nobuaki Fukui

ジアミン構造を有する安定なホスホロアミダイトの開発とリガンド結合型オリゴヌクレオチド合成への応用

日本核酸医薬学会第8回年会 / The 8th Annual Meeting of the Nucleic Acids Therapeutics Society of Japan
2023-07-12 | Conference abstract
Contributors: Nobuaki Fukui; Mitsuaki Sekiguchi; Shunsuke Ochi; Norikazu Kuroda; Takafumi Higuchi; Akira Kugimiya
Source: Self-asserted source
Nobuaki Fukui

Development of a Manufacturing Process toward the Convergent Synthesis of the COVID-19 Antiviral Ensitrelvir

ACS Central Science
2023-04-26 | Journal article | Author
DOI: 10.1021/acscentsci.2c01203
Part of ISSN: 2374-7943
Part of ISSN: 2374-7951
Contributors: Takahiro Kawajiri; Akihito Kijima; Atsuhiro Iimuro; Eisaku Ohashi; Katsuya Yamakawa; Kazushi Agura; Kengo Masuda; Kensuke Kouki; Koji Kasamatsu; Shuichi Yanagisawa et al.
Source: Self-asserted source
Nobuaki Fukui

Development of a manufacturing process toward the convergent synthesis of the COVID-19 antiviral Ensitrelvir

ChemRxiv
2022-10-05 | Preprint
DOI: 10.26434/chemrxiv-2022-wx3nl
Contributors: Takahiro Kawajiri; Akihito Kijima; Atsuhiro Iimuro; Eisaku Ohashi; Katsuya Yamakawa; Kazushi Agura; Kengo Masuda; Kensuke Kouki; Koji Kasamatsu; Shuichi Yanagisawa et al.
Source: Self-asserted source
Nobuaki Fukui

Production method for bifurcated lipid-linked oligonucleotide using cleavage reagent and deprotecting agent, and intermediate

2020-12-10 | Patent
Contributors: Tetsuya Tanino; Mitsuaki Sekiguchi; Shunsuke Ochi; Nobuaki Fukui
Source: Self-asserted source
Nobuaki Fukui

抗インフルエンザ薬 バロキサビル マルボキシルのプロセスの開発

日本プロセス化学会 2019ウインターシンポジウム
2019-12-06 | Conference abstract
Contributors: Nobuaki Fukui
Source: Self-asserted source
Nobuaki Fukui

Process Development for Large-scale Synthesis of Baloxavir marboxil (Xofluza®)

The 4th International Symposium on Process Chemistry [ISPC2019]
2019-07-26 | Conference poster
Contributors: Nobuaki Fukui; Setsuya Shibahara; Toshikatsu Maki; Tomohiro Fukuda; Kousuke Anan; Takayuki Tsuritani
Source: Self-asserted source
Nobuaki Fukui

Microwave‐Assisted Synthesis and Transformations of Cationic CpRu(II)(naphthalene) and CpRu(II)(naphthoquinone) Complexes

Helvetica Chimica Acta
2019-05-03 | Journal article
DOI: 10.1002/hlca.201900076
Part of ISSN: 0018-019X
Part of ISSN: 1522-2675
Contributors: Eva Bocekova‐Gajdošíkova; Bugra Epik; Jingyu Chou; Katsuhiro Akiyama; Nobuaki Fukui; Laure Guénée; E. Peter Kundig
Source: Self-asserted source
Nobuaki Fukui

Polycyclic pyridone derivative, crystal and preparation method thereof

2017-10-11 | Patent
Contributors: Setsuya Shibahara; Nobuaki Fukui; Toshikatsu Maki
Source: Self-asserted source
Nobuaki Fukui

ベンゾトロポロン型天然物goupiolone Aの合成と構造訂正

第32回有機合成若手セミナー: 明日の有機合成を担う人のために / The 32nd Organic Seminar for Young Chemists - For Those Who Take the Future of Syntheric Organic Chemistry -
2012-11-22 | Conference poster
Contributors: Nobuaki Fukui; Ken Ohmori; Keisuke Suzuki
Source: Self-asserted source
Nobuaki Fukui

Synthesis and Structure Revision of Goupiolone A: A Benzotropolone Natural Product

Helvetica Chimica Acta
2012-11-19 | Journal article
DOI: 10.1002/hlca.201200439
Part of ISSN: 0018-019X
Contributors: Nobuaki Fukui; Ken Ohmori; Keisuke Suzuki
Source: Self-asserted source
Nobuaki Fukui

シクロプロピルベンゾシクロブテンの環拡大による中員環形成法の開発に関する研究

日本化学会第92春季年会 / The 92nd CSJ Annual Meeting (2012)
2012-03-28 | Conference abstract
Contributors: Nobuaki Fukui; Ken Ohmori; Keisuke Suzuki
Source: Self-asserted source
Nobuaki Fukui

Ring Expansion of Cyclopropylbenzocyclobutenes En Route to Benzocycloheptenes

Chemistry Letters
2011-10-05 | Journal article
DOI: 10.1246/cl.2011.1198
Part of ISSN: 0366-7022
Part of ISSN: 1348-0715
Contributors: Nobuaki Fukui; Toshiyuki Hamura; Ken Ohmori; Keisuke Suzuki
Source: Self-asserted source
Nobuaki Fukui

ベンゾシクロブテン誘導体の新規環拡大反応に基づく中員環構築に関する研究

日本化学会第90春季年会 / The 90th CSJ Annual Meeting (2010)
2010-03-29 | Conference abstract
Contributors: Nobuaki Fukui; Ken Ohmori; Keisuke Suzuki
Source: Self-asserted source
Nobuaki Fukui

α,α'-ジアルコキシベンザインの反応の位置選択性における置換基効果

日本化学会第88春季年会 / The 88th CSJ Annual Meeting (2008)
2008-03-26 | Conference abstract
Contributors: Nobuaki Fukui; Takeaki Suzuki; Hideyuki Hamura; Takashi Matsumoto; Keisuke Suzuki
Source: Self-asserted source
Nobuaki Fukui
How many people are using ORCID?